Invention Application
- Patent Title: METHOD FOR PRODUCING A VADADUSTAT INTERMEDIATE
-
Application No.: US17605408Application Date: 2020-03-05
-
Publication No.: US20220204451A1Publication Date: 2022-06-30
- Inventor: Koji MACHIDA , Hiroaki YASUKOUCHI , Akira NISHIYAMA
- Applicant: KANEKA CORPORATION
- Applicant Address: JP Osaka-shi, Osaka
- Assignee: KANEKA CORPORATION
- Current Assignee: KANEKA CORPORATION
- Current Assignee Address: JP Osaka-shi, Osaka
- Priority: JP2019-086759 20190426
- International Application: PCT/JP2020/009453 WO 20200305
- Main IPC: C07D213/81
- IPC: C07D213/81

Abstract:
A method for producing a first vadadustat intermediate represented by the following formula (3) comprising reacting a compound represented by the following formula (1) with glycine or a glycine derivative represented by the following formula (2) or a salt of the glycine or the glycine derivative in the presence of carbon monoxide. The method produces a vadadustat intermediate through a clean reaction with high atom conversion efficiency.
Public/Granted literature
- US12134600B2 Method for producing a vadadustat intermediate Public/Granted day:2024-11-05
Information query
IPC分类: