Invention Application
- Patent Title: SMALL MOLECULE INHIBITORS OF A PROTEIN COMPLEX
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Application No.: US17611036Application Date: 2020-06-04
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Publication No.: US20220304958A1Publication Date: 2022-09-29
- Inventor: Alexandre GINGRAS , Mark GINSBERG, , Carlo BALLATORE , Larry SKLAR , Karol Rogelle Karagdag FRANCISCO
- Applicant: THE REGENTS OF THE UNIVERSITY OF CALIFORNIA , THE UNIVERSITY OF NEW MEXICO
- Applicant Address: US CA Oakland; US NM Albuquerque
- Assignee: THE REGENTS OF THE UNIVERSITY OF CALIFORNIA,THE UNIVERSITY OF NEW MEXICO
- Current Assignee: THE REGENTS OF THE UNIVERSITY OF CALIFORNIA,THE UNIVERSITY OF NEW MEXICO
- Current Assignee Address: US CA Oakland; US NM Albuquerque
- International Application: PCT/US2020/036093 WO 20200604
- Main IPC: A61K31/166
- IPC: A61K31/166 ; A61K31/196 ; A61K31/41 ; A61K31/4196 ; A61K31/4406 ; A61K31/245 ; A61K31/44 ; A61K31/135 ; A61K31/423 ; A61K31/472 ; A61K31/235 ; A61K31/05 ; A61K31/192 ; A61K31/337 ; A61K31/085 ; A61K31/095 ; A61K31/10 ; A61K31/055 ; A61K31/121 ; A61K31/451 ; A61K31/136 ; A61K31/397 ; A61K31/222 ; A61K31/137 ; A61K31/381 ; A61K31/11 ; A61P9/14 ; C07C251/24 ; C07D249/14 ; C07D257/06 ; C07D213/74 ; C07C229/56 ; C07C233/81 ; C07C251/48 ; C07D261/20 ; C07D217/16 ; C07C215/50 ; C07C65/19 ; C07C65/105 ; C07D305/08 ; C07C317/22 ; C07C39/38 ; C07C49/83 ; C07D295/112 ; C07D205/08 ; C07C69/738 ; C07C255/56 ; C07C47/575 ; C07D333/22

Abstract:
Compositions and methods for treating thrombosis, inflammation, and atherosclerosis by administration of a compound that binds to KRIT1 to inhibit binding with HEG1.
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