发明授权
- 专利标题: Triazole derivatives and salts thereof and antifungal agent containing the same
- 专利标题(中): 三唑衍生物及其盐和含有它们的抗真菌剂
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申请号: US986800申请日: 1992-12-08
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公开(公告)号: US5366989A公开(公告)日: 1994-11-22
- 发明人: Hiroyuki Imaizumi , Tetsuya Kajita , Kenichi Takashima , Minako Yotsuji , Keiko Takakura , Akira Yotsuji , Junichi Mitsuyama , Katsumi Shimizu , Hiroshi Sakai , Hirokazu Narita
- 申请人: Hiroyuki Imaizumi , Tetsuya Kajita , Kenichi Takashima , Minako Yotsuji , Keiko Takakura , Akira Yotsuji , Junichi Mitsuyama , Katsumi Shimizu , Hiroshi Sakai , Hirokazu Narita
- 申请人地址: JPX Tokyo
- 专利权人: Toyama Chemical Co., Ltd.
- 当前专利权人: Toyama Chemical Co., Ltd.
- 当前专利权人地址: JPX Tokyo
- 优先权: JPX3-350318 19911209; JPX4-293961 19921008
- 主分类号: A61K31/41
- IPC分类号: A61K31/41 ; A61P31/04 ; A61P31/10 ; C07D249/08 ; C07D401/12 ; C07D417/06 ; C07D521/00 ; A01N43/653
摘要:
The present invention relates to a compound represented by the general formula (1) or its salt, a process for producing the same, and an antifungal agent comprising the same as an effective component: ##STR1## wherein R.sup.1 represents a substituted or unsubstituted aryl group or a substituted or unsubstituted heterocyclic group bonded through a carbon atom in the ring to the main chain; R.sup.2 presents a hydrogen atom, a fluorine atom or a substituted or unsubstituted alkyl group; and R.sup.3 represents a cyano group, a thioamido group or a group represented by the formula ##STR2## in which R.sup.4 is a hydroxyl group or a group of the formula ##STR3## (R.sup.7 and R.sup.8, which may be the same or different, are hydrogen atoms or substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, aryl, amino, alkoxy, hydroxyl or heterocyclic groups, and may form a substituted or unsubstituted heterocyclic group together with the nitrogen atom to which R.sup.7 and R.sup.8 attach), R.sup.5 is a substituted or unsubstituted alkoxy group or a group of the formula ##STR4## (R.sup.7 and R.sup.8 are as defined above), and R.sup.6 is a hydrogen atom or a substituted or unsubstituted alkyl group.
公开/授权文献
- US05998788A Ion mobility spectrometer 公开/授权日:1999-12-07
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