Invention Grant
- Patent Title: Guanidine mimics as factor Xa inhibitors
- Patent Title (中): 胍类似物作为因子Xa抑制剂
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Application No.: US09924381Application Date: 2001-08-08
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Publication No.: US06906070B2Publication Date: 2005-06-14
- Inventor: Patrick Y. Lam , Charles G. Clark , Celia Dominguez , John M. Fevig , Qi Han , Renhua Li , Donald J. P. Pinto , James R. Pruitt , Mimi L. Quan
- Applicant: Patrick Y. Lam , Charles G. Clark , Celia Dominguez , John M. Fevig , Qi Han , Renhua Li , Donald J. P. Pinto , James R. Pruitt , Mimi L. Quan
- Applicant Address: US NJ Princeton
- Assignee: Bristol-Myers Squibb Pharma Company
- Current Assignee: Bristol-Myers Squibb Pharma Company
- Current Assignee Address: US NJ Princeton
- Agent David H. Vance; Jing S. Belfield
- Main IPC: C07D231/14
- IPC: C07D231/14 ; C07D231/56 ; C07D233/54 ; C07D233/61 ; C07D261/20 ; C07D401/04 ; C07D403/04 ; C07D405/04 ; C07D413/04 ; C07D413/14 ; A61K31/4725

Abstract:
The present application describes nitrogen containing heteroaromatics and derivatives thereof of formula I: or pharmaceutically acceptable salt forms thereof, wherein rings D-E represent guanidine mimics, which are useful as inhibitors of factor Xa.
Public/Granted literature
- US20020025963A1 Novel guanidine mimics as factor Xa inhibitors Public/Granted day:2002-02-28
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