发明授权
- 专利标题: Guanidine mimics as factor Xa inhibitors
- 专利标题(中): 胍类似物作为因子Xa抑制剂
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申请号: US09924381申请日: 2001-08-08
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公开(公告)号: US06906070B2公开(公告)日: 2005-06-14
- 发明人: Patrick Y. Lam , Charles G. Clark , Celia Dominguez , John M. Fevig , Qi Han , Renhua Li , Donald J. P. Pinto , James R. Pruitt , Mimi L. Quan
- 申请人: Patrick Y. Lam , Charles G. Clark , Celia Dominguez , John M. Fevig , Qi Han , Renhua Li , Donald J. P. Pinto , James R. Pruitt , Mimi L. Quan
- 申请人地址: US NJ Princeton
- 专利权人: Bristol-Myers Squibb Pharma Company
- 当前专利权人: Bristol-Myers Squibb Pharma Company
- 当前专利权人地址: US NJ Princeton
- 代理商 David H. Vance; Jing S. Belfield
- 主分类号: C07D231/14
- IPC分类号: C07D231/14 ; C07D231/56 ; C07D233/54 ; C07D233/61 ; C07D261/20 ; C07D401/04 ; C07D403/04 ; C07D405/04 ; C07D413/04 ; C07D413/14 ; A61K31/4725
摘要:
The present application describes nitrogen containing heteroaromatics and derivatives thereof of formula I: or pharmaceutically acceptable salt forms thereof, wherein rings D-E represent guanidine mimics, which are useful as inhibitors of factor Xa.
公开/授权文献
- US20020025963A1 Novel guanidine mimics as factor Xa inhibitors 公开/授权日:2002-02-28