Invention Grant
- Patent Title: Histamine H3-receptor ligands and their therapeutic applications
- Patent Title (中): 组胺H3受体配体及其治疗应用
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Application No.: US11912816Application Date: 2006-04-25
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Publication No.: US08076329B2Publication Date: 2011-12-13
- Inventor: Isabelle Bertrand , Marc Capet , Jeanne-Marie Lecomte , Nicolas Levoin , Xavier Ligneau , Olivia Poupardin-Olivier , Philippe Robert , Jean-Charles Schwartz , Olivier Labeeuw
- Applicant: Isabelle Bertrand , Marc Capet , Jeanne-Marie Lecomte , Nicolas Levoin , Xavier Ligneau , Olivia Poupardin-Olivier , Philippe Robert , Jean-Charles Schwartz , Olivier Labeeuw
- Applicant Address: FR Paris
- Assignee: Bioprojet
- Current Assignee: Bioprojet
- Current Assignee Address: FR Paris
- Agency: Stites & Harbison PLLC
- Agent B. Aaron Schulman, Esq.; Terry L. Wright, Esq.
- Priority: EP05290950 20050429; EP05291793 20050826
- International Application: PCT/IB2006/000991 WO 20060425
- International Announcement: WO2006/117609 WO 20061109
- Main IPC: A61K31/4418
- IPC: A61K31/4418 ; A61K31/4453 ; A61K31/4545 ; A61K31/5355 ; C07D213/30 ; C07D211/14 ; C07D413/12
Abstract:
The present patent application concerns compounds of formula (I) with R1 and R2 taken together with the nitrogen atom to which they are attached, form a mono or bicyclic saturated nitrogen-containing ring; their preparation and their use as a H3 receptor ligand for treating e.g. CNS disorders like Alzheimer's disease.
Public/Granted literature
- US20090111808A1 NOVEL HISTAMINE H3-RECEPTOR LIGANDS AND THEIR THERAPEUTIC APPLICATIONS Public/Granted day:2009-04-30
Information query
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