Invention Grant
- Patent Title: Heterocyclic derivatives as GPCR receptor agonists
- Patent Title (中): 杂环衍生物作为GPCR受体激动剂
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Application No.: US10584025Application Date: 2004-12-23
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Publication No.: US08207147B2Publication Date: 2012-06-26
- Inventor: Matthew Colin Thor Fyfe , Lisa Sarah Gardner , John King-Underwood , Martin James Procter , Chrystelle Marie Rasamison , Karen Lesley Schofield , Gerard Hugh Thomas
- Applicant: Matthew Colin Thor Fyfe , Lisa Sarah Gardner , John King-Underwood , Martin James Procter , Chrystelle Marie Rasamison , Karen Lesley Schofield , Gerard Hugh Thomas
- Applicant Address: GB Oxford
- Assignee: Prosidion Limited
- Current Assignee: Prosidion Limited
- Current Assignee Address: GB Oxford
- Agency: Mintz Levin Cohn Ferris Glovsky and Popeo, P.C.
- Agent Ivor R. Elrifi; Heidi A. Erlacher
- International Application: PCT/GB2004/050046 WO 20041223
- International Announcement: WO2005/061489 WO 20050707
- Main IPC: A61K31/66
- IPC: A61K31/66 ; A61K31/497 ; A61K31/4523 ; C07D401/14 ; C07F9/02 ; C07D211/00 ; C07D413/14
Abstract:
Compounds of Formula (I), R1-A-V—B—R2; or pharmaceutically acceptable salts thereof, are agonists of GPR116 and are useful as regulators of satiety, e.g. for the treatment of obesity, and for the treatment of diabetes.
Public/Granted literature
- US20090281060A1 HETEROCYCLIC DERIVATIVES AS GPCR RECEPTOR AGONISTS Public/Granted day:2009-11-12
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