Invention Application
WO0220526A3 CYCLIC AND ACYCLIC AMIDINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR USE AS PROGESTERONE RECEPTOR BINDING AGENTS
审中-公开
包含它们作为孕激素受体结合剂的循环和ACYCLIC和药物组合物
- Patent Title: CYCLIC AND ACYCLIC AMIDINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR USE AS PROGESTERONE RECEPTOR BINDING AGENTS
- Patent Title (中): 包含它们作为孕激素受体结合剂的循环和ACYCLIC和药物组合物
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Application No.: PCT/US0127007Application Date: 2001-08-30
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Publication No.: WO0220526A3Publication Date: 2002-05-30
- Inventor: BULLOCK WILLIAM H , KLUENDER HAROLD C E , COLLIBEE WILLIAM L , DALLY ROBERT , RODRIGUEZ MARTHA E , WANG MING
- Applicant: BAYER AG , BULLOCK WILLIAM H , KLUENDER HAROLD C E , COLLIBEE WILLIAM L , DALLY ROBERT , RODRIGUEZ MARTHA E , WANG MING
- Assignee: BAYER AG,BULLOCK WILLIAM H,KLUENDER HAROLD C E,COLLIBEE WILLIAM L,DALLY ROBERT,RODRIGUEZ MARTHA E,WANG MING
- Current Assignee: BAYER AG,BULLOCK WILLIAM H,KLUENDER HAROLD C E,COLLIBEE WILLIAM L,DALLY ROBERT,RODRIGUEZ MARTHA E,WANG MING
- Priority: US65685400 2000-09-07
- Main IPC: C07D295/12
- IPC: C07D295/12 ; A61K31/136 ; A61K31/155 ; A61K31/395 ; A61K31/40 ; A61K31/403 ; A61K31/426 ; A61K31/438 ; A61K31/439 ; A61K31/445 ; A61K31/47 ; A61K31/496 ; A61K31/5375 ; A61K31/55 ; A61P5/24 ; A61P5/42 ; A61P15/00 ; A61P15/02 ; A61P15/04 ; A61P15/06 ; A61P15/08 ; A61P15/12 ; A61P19/08 ; A61P19/10 ; A61P35/00 ; A61P43/00 ; C07C257/14 ; C07D207/22 ; C07D209/52 ; C07D209/54 ; C07D211/14 ; C07D211/72 ; C07D215/38 ; C07D221/20 ; C07D221/22 ; C07D223/12 ; C07D223/14 ; C07D223/32 ; C07D225/02 ; C07D235/26 ; C07D265/30 ; C07D277/04 ; C07D295/125 ; C07D453/06 ; C07D487/08 ; A61K31/435 ; C07D295/13
Abstract:
Disclosed are cyclic and acyclic amidines, pharmaceutical compositions containing such amidines, and their use in treating or preventing progesterone receptor mediated diseases or conditions, such as osteopenia and osteoporosis.
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