专利检索 ap:("Incyte Corporation") AND inv:"LIU, Pingli" 第 1 页

1.

发明公开
PROCESS AND INTERMEDIATES FOR PREPARING A JAK1 INHIBITOR 审中-公开

公开(公告)号：EP4200278A1

公开(公告)日：2023-06-28

申请号：EP21766776.5

申请日：2021-08-17

申请人： Incyte Corporation

发明人： ZHOU, Jiacheng , CHEN, Shili , LIU, Pingli , MELONI, David J. , PAN, Yongchun , SU, Naijing , XIA, Michael

IPC分类号： C07D205/04 , C07D401/14

2.

发明授权
1,2,5-OXADIAZOLES AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE 有权
标题翻译： 1,2,5-恶二唑AS吲哚胺2,3-双加氧酶的抑制剂

公开(公告)号：EP2315756B9

公开(公告)日：2015-07-22

申请号：EP09790108.6

申请日：2009-07-07

申请人： Incyte Corporation

发明人： COMBS, Andrew, P. , YUE, Eddy, W. , SPARKS, Richard, B. , ZHU, Wenyu , ZHOU, Jiacheng , LIN, Qiyan , WENG, Lingkai , YUE, Tai-Yuen , LIU, Pingli

IPC分类号： C07D271/08 , A61K31/4245 , A61P1/00 , A61P11/00 , A61P17/00 , A61P19/00 , A61P25/00 , A61P27/00 , A61P29/00 , A61P31/00 , A61P35/00 , A61P37/00 , A61P43/00

CPC分类号： A61K31/4245 , A61K39/0011 , A61K39/3955 , C07D271/08 , C07D413/04 , C07D413/12

3.

发明公开
CRYSTALLINE SOLID FORMS OF A BET INHIBITOR 审中-公开

公开(公告)号：EP4234554A3

公开(公告)日：2023-12-27

申请号：EP23160938.9

申请日：2017-06-19

申请人： Incyte Corporation

发明人： CHEN, Shili , JIA, Zhongjiang , LIU, Pingli , QIAO, Lei , WU, Yongzhong , ZHOU, Jiacheng , LI, Qun

IPC分类号： C07D471/04 , A61K31/538 , A61P35/00

摘要： The present application relates to crystalline solid forms of an inhibitor of BET proteins such as BRD2, BRD3, BRD4, and BRD-t, including methods of preparation thereof, and intermediates in the preparation thereof, where the compound is useful in the treatment of diseases such as cancer.

4.

发明公开
PROCESSES OF PREPARING A JAK1 INHIBITOR AND NEW FORMS THERETO 审中-公开
标题翻译： PROCESS其制造JAK1抑制剂和新形式

公开(公告)号：EP3137471A1

公开(公告)日：2017-03-08

申请号：EP15724406.2

申请日：2015-04-29

申请人： Incyte Corporation

发明人： ZHOU, Jiacheng , LIU, Pingli , CHEN, Shili , WU, Yongzhong , WANG, Dengjin , JIA, Zhongjiang , QIAO, Lei , FRIETZE, William , XIA, Michael , DAI, Yingrui

IPC分类号： C07D495/14 , A61K31/437 , A61P25/00 , A61P35/00 , A61P37/00

CPC分类号： C07D495/14 , C07D309/14 , C07D495/04

摘要： This invention relates to processes for preparing a JAK1 inhibitor having Formula Ia: as well as new forms of the inhibitor.

摘要翻译： 本发明涉及用于制备具有式Ia一个JAK1抑制剂：以及所述抑制剂的新形式。

5.

发明公开
PROCESS AND INTERMEDIATES FOR PREPARING BARICITINIB 审中-实审

公开(公告)号：EP4370504A1

公开(公告)日：2024-05-22

申请号：EP22748725.3

申请日：2022-07-11

申请人： Incyte Corporation

发明人： ZHOU, Jiacheng , CHEN, Shili , JIA, Zhongjiang , LIU, Pingli , MELONI, David , PAN, Yongchun , SU, Naijing , XIA, Michael

IPC分类号： C07D205/04 , C07D487/04

CPC分类号： C07D205/04 , C07D487/04

6.

发明授权
SALTS OF PI3K INHIBITOR AND PROCESSES FOR THEIR PREPARATION 有权

公开(公告)号：EP3262046B1

公开(公告)日：2020-11-04

申请号：EP16718921.6

申请日：2016-02-26

申请人： Incyte Corporation

发明人： QIAO, Lei , WENG, Lingkai , SHI, ChongSheng Eric , MELONI, David , LIN, Qiyan , XIA, Michael , SHARIEF, Vaqar , FRIETZE, William , JIA, Zhongjiang , PAN, Yongchun , LIU, Pingli , YUE, Tai-Yuen , ZHOU, Jiacheng

IPC分类号： C07D487/04 , A61K31/519 , A61P35/00

7.

发明公开
SALTS AND SOLID FORMS OF AN FGFR INHIBITOR AND PROCESSES OF PREPARING THEREOF 审中-公开

公开(公告)号：EP4452982A1

公开(公告)日：2024-10-30

申请号：EP22854263.5

申请日：2022-12-21

申请人： Incyte Corporation

发明人： LIU, Pingli , JIA, Zhongjiang , LIN, Qiyan , SU, Naijing , MARTIN, Timothy , XIA, Michael , ZHOU, Jiacheng , MI, Baoyu

IPC分类号： C07D487/04 , A61P35/00 , A61K31/498

8.

发明公开
CRYSTALLINE SOLID FORMS OF A BET INHIBITOR 审中-公开

公开(公告)号：EP4234554A2

公开(公告)日：2023-08-30

申请号：EP23160938.9

申请日：2017-06-19

申请人： Incyte Corporation

发明人： CHEN, Shili , JIA, Zhongjiang , LIU, Pingli , QIAO, Lei , WU, Yongzhong , ZHOU, Jiacheng , LI, Qun

IPC分类号： C07D471/04

摘要： The present application relates to crystalline solid forms of an inhibitor of BET proteins such as BRD2, BRD3, BRD4, and BRD-t, including methods of preparation thereof, and intermediates in the preparation thereof, where the compound is useful in the treatment of diseases such as cancer.

9.

发明公开
PROCESSES FOR PREPARING INTERMEDIATES FOR THE SYNTHESIS OF A JAK INHIBITOR 审中-公开

公开(公告)号：EP4086245A1

公开(公告)日：2022-11-09

申请号：EP22157237.3

申请日：2019-01-29

申请人： Incyte Corporation

发明人： WANG, Dengjin , LIU, Pingli , WU, Yongzhong , ZHOU, Jiacheng

IPC分类号： C07D401/04 , C07D213/61

摘要： This invention relates to processes and intermediates for making {1-{1-[3-fluoro-2-(trifluoromethyl)isonicotinoyl]piperidin-4-yl}-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile, useful in the treatment of diseases related to the activity of Janus kinases (JAK) including inflammatory disorders, autoimmune disorders, cancer, and other diseases.

10.

发明公开
SALTS OF A PD-1/PD-L1 INHIBITOR 审中-公开

公开(公告)号：EP4010342A1

公开(公告)日：2022-06-15

申请号：EP20760703.7

申请日：2020-08-07

申请人： Incyte Corporation

发明人： JIA, Zhongjiang , LIU, Pingli , MELONI, David J. , PAN, Yongchun , WU, Yongzhong , ZHOU, Jiacheng , LI, Qun

IPC分类号： C07D471/04 , A61K31/4375 , A61P31/04 , A61P31/10 , A61P31/12 , A61P33/00 , A61P35/00