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公开(公告)号：EP2300465B1
公开(公告)日：2019-04-17
申请号：EP09761801.1
申请日：2009-06-12
发明人： BERDINI, Valerio , CARR, Maria, Grazia , CONGREVE, Miles, Stuart , FREDERICKSON, Martyn , GRIFFITHS-JONES, Charlotte, Mary , HAMLETT, Christopher, Charles, Frederick , MADIN, Andrew , MURRAY, Christopher, William , BENNING, Rajdeep Kaur , SAXTY, Gordon , VICKERSTAFFE, Emma , WOODHEAD, Andrew, James , WOODHEAD, Steven, John , FREYNE, Eddy, Jean, Edgard , GOVAERTS, Tom, Cornelis, Hortense , ANGIBAUD, Patrick, René , WILLIAMS, Brian, John
IPC分类号： C07D471/04 , C07D513/04 , A61P35/00 , A61K31/437 , A61K31/506 , A61K31/501 , A61K31/53 , A61K31/444 , A61K31/497 , A61K31/496 , A61K31/4545
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公开(公告)号：EP2776397B1
公开(公告)日：2017-11-29
申请号：EP12794744.8
申请日：2012-10-26
IPC分类号： C07D215/38 , C07D401/04 , C07D401/14 , C07D407/14 , C07D413/14 , A61K31/4709 , A61K31/47 , A61P35/00 , C07D405/14 , A61K45/06 , A61K31/506 , A61K31/5377
CPC分类号： A61K31/4709 , A61K31/47 , A61K31/506 , A61K31/5377 , A61K45/06 , C07D215/38 , C07D401/04 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/14
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公开(公告)号：EP2776397A1
公开(公告)日：2014-09-17
申请号：EP12794744.8
申请日：2012-10-26
IPC分类号： C07D215/38 , C07D401/04 , C07D401/14 , C07D407/14 , C07D413/14 , A61K31/4709 , A61K31/47 , A61P35/00
CPC分类号： A61K31/4709 , A61K31/47 , A61K31/506 , A61K31/5377 , A61K45/06 , C07D215/38 , C07D401/04 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/14
摘要： The invention relates to new quinoline derivative compounds of formula (I), to pharmaceutical compositions comprising said compounds, to processes for the preparation of said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer. Formula (I)
摘要翻译： 本发明涉及式（I）的新的喹啉衍生物化合物，包含所述化合物的药物组合物，所述化合物的制备方法以及所述化合物在治疗疾病中的用途。 癌症。 式（I）
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公开(公告)号：EP2563775A1
公开(公告)日：2013-03-06
申请号：EP11724710.6
申请日：2011-04-28
发明人： SAXTY, Gordon , MURRAY, Christopher William , BERDINI, Valerio , BESONG, Gilbert Ebai , HAMLETT, Christopher Charles Frederick , JOHNSON, Christopher Norbert , WOODHEAD, Steven John , READER, Michael , REES, David Charles , MEVELLEC, Laurence Anne , ANGIBAUD, Patrick René , FREYNE, Eddy Jean Edgard , GOVAERTS, Tom Cornelis Hortense , WEERTS, Johan Erwin Edmond , PERERA, Timothy Pietro Suren , GILISSEN, Ronaldus Arnodus Hendrika Joseph , WROBLOWSKI, Berthold , LACRAMPE, Jean Fernand Armand , PAPANIKOS, Alexandra , QUEROLLE, Oliver Alexis Georges , PASQUIER, Elisabeth Thérèse Jeanne , PILATTE, Isabelle Noëlle Constance , BONNET, Pascal Ghislain André , EMBRECHTS, Werner Constant Johan , AKKARI, Rhalid , MEERPOEL, Lieven
IPC分类号： C07D403/04 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D487/08 , A61K31/498 , A61P35/00
CPC分类号： C07D403/04 , A61K31/498 , A61K31/5377 , A61K45/06 , C07D401/14 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D487/08 , C07D491/113 , C07F9/6524
摘要： The invention relates to new quinoxaline derivative compounds, to pharmaceutical compositions comprising said compounds, to processes for the preparation of said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
摘要翻译： 本发明涉及新的喹喔啉衍生物化合物，涉及包含所述化合物的药物组合物，制备所述化合物的方法以及所述化合物在治疗疾病中的用途， 癌症。
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公开(公告)号：EP2300465A1
公开(公告)日：2011-03-30
申请号：EP09761801.1
申请日：2009-06-12
发明人： BERDINI, Valerio , CARR, Maria, Grazia , CONGREVE, Miles, Stuart , FREDERICKSON, Martyn , GRIFFITHS-JONES, Charlotte, Mary , HAMLETT, Christopher, Charles, Frederick , MADIN, Andrew , MURRAY, Christopher, William , BENNING, Rajdeep Kaur , SAXTY, Gordon , VICKERSTAFFE, Emma , WOODHEAD, Andrew, James , WOODHEAD, Steven, John , FREYNE, Eddy, Jean, Edgard , GOVAERTS, Tom, Cornelis, Hortense , ANGIBAUD, Patrick, René , WILLIAMS, Brian, John
IPC分类号： C07D471/04 , C07D513/04 , A61P35/00 , A61K31/437 , A61K31/506 , A61K31/501 , A61K31/53 , A61K31/444 , A61K31/497 , A61K31/496 , A61K31/4545
CPC分类号： C07D471/04 , C07D513/04
摘要： The invention relates to new bicyclic heterocyclic derivative compounds, to pharmaceutical compositions comprising the compounds and to the use of the compounds in the treatment of diseases, e.g. cancer.
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公开(公告)号：EP2776435B1
公开(公告)日：2018-06-27
申请号：EP12794745.5
申请日：2012-10-26
发明人： BERDINI, Valerio , SAXTY, Gordon , ANGIBAUD, Patrick René , QUEROLLE, Olivier Alexis Georges , PONCELET, Virginie Sophie , ROUX, Bruno , MEERPOEL, Lieven
IPC分类号： C07D471/04 , A61P35/00 , A61K31/4985
CPC分类号： A61K31/4985 , A61K31/506 , A61K31/5377 , C07D471/04
摘要： The invention relates to new pyridopyrazine derivative compounds, to pharmaceutical compositions comprising said compounds, to processes for the preparation of said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
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公开(公告)号：EP2563775B1
公开(公告)日：2017-01-04
申请号：EP11724710.6
申请日：2011-04-28
发明人： SAXTY, Gordon , MURRAY, Christopher William , BERDINI, Valerio , BESONG, Gilbert Ebai , HAMLETT, Christopher Charles Frederick , JOHNSON, Christopher Norbert , WOODHEAD, Steven John , READER, Michael , REES, David Charles , MEVELLEC, Laurence Anne , ANGIBAUD, Patrick René , FREYNE, Eddy Jean Edgard , GOVAERTS, Tom Cornelis Hortense , WEERTS, Johan Erwin Edmond , PERERA, Timothy Pietro Suren , GILISSEN, Ronaldus Arnodus Hendrika Joseph , WROBLOWSKI, Berthold , LACRAMPE, Jean Fernand Armand , PAPANIKOS, Alexandra , QUEROLLE, Olivier Alexis Georges , PASQUIER, Elisabeth Thérèse Jeanne , PILATTE, Isabelle Noëlle Constance , BONNET, Pascal Ghislain André , EMBRECHTS, Werner Constant Johan , AKKARI, Rhalid , MEERPOEL, Lieven
IPC分类号： C07D403/04 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D487/08 , A61K31/498 , A61P35/00
CPC分类号： C07D403/04 , A61K31/498 , A61K31/5377 , A61K45/06 , C07D401/14 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D487/08 , C07D491/113 , C07F9/6524
摘要： The invention relates to new quinoxaline derivative compounds, to pharmaceutical compositions comprising said compounds, to processes for the preparation of said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
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公开(公告)号：EP2203449B1
公开(公告)日：2016-04-27
申请号：EP08806575.0
申请日：2008-10-10
发明人： SAXTY, Gordon , BERDINI, Valerio , MURRAY, Christopher, William , GRIFFITHS-JONES, Charlotte, Mary , VICKERSTAFFE, Emma , BESONG, Gilbert, Ebai
IPC分类号： C07D471/04 , C07D487/04 , A61P35/00 , A61K31/437
CPC分类号： C07D471/04
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公开(公告)号：EP2114941B1
公开(公告)日：2015-03-25
申请号：EP07848659.4
申请日：2007-12-21
发明人： BERDINI, Valerio , BESONG, Gilbert, Ebai , CALLAGHAN, Owen , CARR, Maria, Grazia , CONGREVE, Miles, Stuart , GILL, Adrian, Liam , GRIFFITHS-JONES, Charlotte, Mary , MADIN, Andrew , MURRAY, Christopher, William , NIJJAR, Rajdeep, Kaur , O'BRIEN, Michael, Alistair , PIKE, Andrew , SAXTY, Gordon , TAYLOR, Richard, David , VICKERSTAFFE, Emma
IPC分类号： C07D471/04 , C07D487/04 , A61K31/437 , A61K31/519 , A61P35/00
CPC分类号： C07D487/04 , A61K31/437 , C07D471/04
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30.发明公开
公开(公告)号：EP2197880A1
公开(公告)日：2010-06-23
申请号：EP08806556.0
申请日：2008-10-10
发明人： SAXTY, Gordon , BERDINI, Valerio , MURRAY, Christopher, William , GRIFFITHS-JONES, Charlotte, Mary , VICKERSTAFFE, Emma , BESONG, Gilbert, Ebai , CARR, Maria, Grazia
IPC分类号： C07D471/04 , C07D487/04 , A61P35/00 , A61K31/437
CPC分类号： C07D471/04 , C07D487/04
摘要： The invention relates to new bicyclic heterocyclic derivative compounds of formula (I): wherein R1, A, X1, X2, X3, X4, X5 and R2 are as defined herein, to pharmaceutical compositions comprising said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
摘要翻译： 本发明涉及式（I）的新双环杂环衍生物化合物：其中R 1，A，X 1，X 2，X 3，X 4，X 5和R 2如本文所定义，涉及包含所述化合物的药物组合物以及所述化合物在 疾病的治疗，例如 癌症。
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