SOIL- OR SEED-TREATING AGENT COMPRISING QUINOLINE COMPOUND OR SALT THEREOF AS ACTIVE INGREDIENT, OR METHOD FOR CONTROL OF PLANT DISEASE USING THE SAME
    1.
    发明公开
    SOIL- OR SEED-TREATING AGENT COMPRISING QUINOLINE COMPOUND OR SALT THEREOF AS ACTIVE INGREDIENT, OR METHOD FOR CONTROL OF PLANT DISEASE USING THE SAME 有权
    使用喹或其盐在土壤和种子处理是指主动和方法防治植物病害

    公开(公告)号:EP2103214A1

    公开(公告)日:2009-09-23

    申请号:EP07832840.8

    申请日:2007-11-30

    CPC分类号: A01N43/42 A01N43/90

    摘要: A soil treating agent or a seed treating agent having excellent prevention effects against various plant pathogens (particularly against rice blast) is provided. A soil treating agent or seed treating agent, comprising one or more compounds of the general formula (Ia), (Ib) or (Ic):

    (wherein R 1 , R 2 : C 1 -C 6 alkyl (may be substituted), aryl (may be substituted), heteroaryl (may be substituted), aralkyl (may be substituted) and the like; R 3 , R 4 : H, C 1 -C 6 alkyl (may be substituted), halogen, C 1 -C 6 alkoxy and the like; X: halogen, C 1 -C 6 alkyl (may be substituted), C 2 -C 6 alkenyl (may be substituted), C 2 -C 6 alkynyl (may be substituted), aryl (may be substituted), heteroaryl (may be substituted), C 1 -C 6 alkoxy and the like; Y: halogen, C 1 -C 6 alkyl, C 1 -C 6 alkoxy, OH; n: 0 to 4; m: 0 to 6)
    or salts thereof as an active ingredient.

    摘要翻译: 提供土壤处理剂或具有抗各种植物病原体的优良效果预防种子处理剂(特别是对稻瘟病)。 土壤处理剂处理或种子剂,其中含有通式(Ia),(Ib)或(Ic)的一种或多种化合物:(其中,R 1,R 2:C 1个-C 6烷基(可以是substituiertem) 芳基(可以是substituiertem),杂芳基(可以是substituiertem),芳烷基(可以是substituiertem)等; R 3,R 4:H,C 1个-C 6烷基(可以是substituiertem),卤素,C 1个-C 6烷氧基等; X:卤素,C 1 -C 6烷基(可以是substituiertem),C 2 -C 6链烯基(可以是substituiertem),C 2 -C 6炔基(可以是substituiertem),芳基(可以是 取代),杂芳基(可以是substituiertem),C 1 -C 6烷氧基等; Y:卤素,C 1 -C 6烷基,C 1 -C 6烷氧基,OH,N:0〜4; m = 0时,以 6)或其盐在其作为活性成分。

    N-HETEROARYLNICOTINAMIDE DERIVATIVES
    3.
    发明公开
    N-HETEROARYLNICOTINAMIDE DERIVATIVES 有权
    N-杂芳酰基二酰胺衍生物

    公开(公告)号:EP1460071A1

    公开(公告)日:2004-09-22

    申请号:EP02803536.8

    申请日:2002-11-19

    摘要: An N-heteroaryl-4-(haloalkyl)nicotinamide derivative represented by formula (I):
    [wherein R represents a C 1 -C 6 haloalkyl group; R 1 represents a hydrogen atom, a C 1 -C 6 alkyl group which may be substituted a C 2 -C 6 alkenyl group or an acyl group; X represents a group represented by formula C-R 2 , or a nitrogen atom; R 2 and R 3 each independently represent a hydrogen atom, a halogen atom, a C 1 -C 6 alkyl group which may be substituted, a C 3 -C 7 cycloalkyl group, a C 2 -C 6 alkenyl group, a C 3 -C 7 cycloalkenyl group, a formyl group, a group represented by formula CH=NOR 4 , a cyano group, a phenyl group which may be substituted, a heterocyclic group which may be substituted, a C 1 -C 6 alkoxy group which may be substituted, a C 1 -C 6 alkylthio group or a phenoxy group]; or a salt thereof, a pesticide containing it as an active component, a method for producing it and intermediates thereof.

    摘要翻译: 由式(I)表示的N-杂芳基-4-(卤代烷基)烟酰胺衍生物:[其中R表示C1-C6卤代烷基; R 1表示氢原子,可以被C 2 -C 6烯基或酰基取代的C 1 -C 6烷基; X表示由式C-R2表示的基团或氮原子; R2和R3各自独立地表示氢原子,卤素原子,可被取代的C1-C6烷基,C3-C7环烷基,C2-C6烯基,C3-C7环烯基,甲酰基, 由式CH = NOR4表示的基团,氰基,可被取代的苯基,可被取代的杂环基,可被取代的C1-C6烷氧基,C1-C6烷硫基或苯氧基 ]。 或其盐,含有它作为活性组分的农药,其制备方法及其中间体。

    PROCESS FOR PRODUCING CYCLOPROPYLPHENOL DERIVATIVE
    7.
    发明公开
    PROCESS FOR PRODUCING CYCLOPROPYLPHENOL DERIVATIVE 审中-公开
    生产环丙基苯酚衍生物的方法

    公开(公告)号:EP1880987A1

    公开(公告)日:2008-01-23

    申请号:EP06730754.6

    申请日:2006-03-31

    摘要: An object of the present invention is to find a method for easily synthesizing cyclopropylphenol derivatives. The object of the present invention is to find a process for producing a cyclopropylphenol derivative represented by general formula (10):

    [wherein R 1 , R 2 , R 3 and R 4 each independently represent a hydrogen atom or the like; Z represents a hydrogen atom or the like; and Y 1 , Y 2 and Y 3 each independently represent a hydrogen atom or the like];
    and solved by the process comprising reacting a compound represented by general formula (7):

    [wherein each of the symbols are the same as previously defined; X represents a halogen atom; and V represents a hydrogen atom or the like],
    with a metal, metal salt or organometallic compound represented by general formula (8): M 2 to obtain a compound represented by general formula (9):

    [wherein each of the symbols are the same as previously defined] and obtaining a compound represented by general formula (10) by hydrolysis in the case V represents the group, -W-R 5 .

    摘要翻译: 本发明的一个目的是找到一种容易合成环丙基苯酚衍生物的方法。 本发明的目的是找到一种制备通式(10)表示的环丙基苯酚衍生物的方法:[其中R1,R2,R3和R4各自独立地代表氢原子等; Z表示氢原子等; Y 1,Y 2和Y 3各自独立地表示氢原子等]。 并通过包括使由通式(7)表示的化合物:[其中每个符号与前​​述定义相同; X代表卤素原子; (8)表示的金属,金属盐或有机金属化合物与通式(9)表示的化合物反应,得到通式(9)所示的化合物,式中,各符号相同 如前所定义],并且在V表示基团-W-R5的情况下通过水解获得通式(10)表示的化合物。

    3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES
    8.
    发明公开
    3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES 有权
    3-(二氢(四氢)ISOCHINOLIN -1-基)喹

    公开(公告)号:EP1736471A1

    公开(公告)日:2006-12-27

    申请号:EP05704224.4

    申请日:2005-01-21

    摘要: A compound is provided which is useful as an active ingredient of an agricultural chemical having superior antimicrobial activity against various plant diseases and capable of controlling rice blast and so on at a low dose.
    A compound or salt thereof represented by the following general formula:


    (wherein, R 1 and R 2 represent a C 1 -C 6 alkyl group, aryl group, heteroaryl group, aralkyl group or R 1 and R 2 together represent a C 3 -C 10 cycloalkyl group, R 3 and R 4 represent a hydrogen atom, a C 1 -C 6 alkyl group or R 3 and R 4 together represent a C 3 -C 10 cycloalkyl group, R 5 represents a hydrogen atom, C 1 -C 6 alkyl group or acyl group, X represents a halogen atom, a C 1 -C 6 alkyl group, C 2 -C 6 alkenyl group, C 2 -C 6 alkynyl group, aryl group, heteroaryl group, C 1 -C 6 alkoxy group, amino group, acyl group, cyano group or N-hydroxyalkaneimidoyl group, Y represents a substituent selected from the group consisting of a halogen atom, C 1 -C 6 alkyl group, C 1 -C 6 alkoxy group and hydroxyl group, n represents an integer of 0 to 4, and m represents an integer of 0 to 6).

    摘要翻译: 提供了一种化合物,其可用作农药的有效成分,对各种植物疾病具有优异的抗微生物活性,并且能够以低剂量控制稻瘟病等。 由下列通式表示的化合物或其盐:其中R 1和R 2表示C 1 -C 6烷基,芳基,杂芳基,芳烷基或R 1和R 2一起表示C 3 - C 10环烷基,R 3和R 4表示氢原子,C 1 -C 6烷基或R 3和R 4一起表示C 3 -C 10环烷基,R 5表示氢原子,C 1〜 C 6烷基或酰基,X表示卤素原子,C 1〜C 6烷基,C 2〜C 6烯基,C 2〜C 6炔基,芳基,杂芳基,C 1 -C 6 烷氧基,氨基,酰基,氰基或N-羟基亚氨基亚氨基,Y表示选自卤素原子,C 1 -C 6烷基,C 1 -C 6烷氧基和羟基的取代基, n表示0〜4的整数,m表示0〜6的整数。

    METHOD OF PREVENTING WHEAT FROM MYCOTOXIN CONTAMINATION
    9.
    发明公开
    METHOD OF PREVENTING WHEAT FROM MYCOTOXIN CONTAMINATION 有权
    VERFAHREN ZUM SCHUTZ VON WEIZEN VOR MYKOTOXINBEFALL

    公开(公告)号:EP1568277A1

    公开(公告)日:2005-08-31

    申请号:EP03777255.5

    申请日:2003-12-04

    IPC分类号: A01N57/12 A01N59/06

    摘要: We search for a cultivation method for reducing the amount of mycotoxin contamination in wheat which has been an important pending question for the quality in actual producing field of wheat and the health hazard risk for customers.
    The present invention discloses a method of reducing the contamination amount of mycotoxin in cereals characterized in that one or more compounds A selected from the group consisting of ammonium salts, primary to quaternary ammonium salts, alkali metal salts, alkaline earth metal salts and polyvalent metal salts of phosphorous acid and phosphite ester are given to the cereals.

    摘要翻译: 我们寻求减少小麦真菌毒素污染量的培养方法,这是小麦实际生产领域质量的重要问题,也是客户的健康危害风险。 本发明公开了一种减少谷物中霉菌毒素的污染量的方法,其特征在于一种或多种选自铵盐,伯 - 季铵盐,碱金属盐,碱土金属盐 并向谷物提供亚磷酸和亚磷酸酯的多价金属盐。