公开(公告)号：EP1526896A1

公开(公告)日：2005-05-04

申请号：EP03766214.5

申请日：2003-07-18

申请人： Bayer HealthCare AG

发明人： LAMPE, Thomas ,  ADELT, Isabelle ,  BEYER, Dieter ,  BRUNNER, Nina ,  ENDERMANN, Rainer ,  EHLERT, Kerstin ,  KROLL, Hein-Peter ,  VON NUSSBAUM, Franz ,  RADDATZ, Siegfried ,  RUDOLPH, Joachim ,  SCHIFFER, Guido ,  SCHUMACHER, Andreas ,  CANCHO-GRANDE, Yolanda ,  MICHELS, Martin ,  WEIGAND, Stefan

IPC分类号： A61P31/00 ,  C07D245/06 ,  A61K31/395

CPC分类号： C07K5/0812 ,  A61K38/00

摘要： The invention relates to antibacterial ester macrocycles of formula (I), methods for the production thereof, and the use thereof for producing medicaments used for the treatment and/or prophylaxis of diseases, particularly bacterial infections.

公开(公告)号：EP1515983A1

公开(公告)日：2005-03-23

申请号：EP03738012.8

申请日：2003-06-10

申请人： Bayer HealthCare AG

发明人： LAMPE, Thomas ,  ADELT, Isabelle ,  BEYER, Dieter ,  BRUNNER, Nina ,  ENDERMANN, Rainer ,  EHLERT, Kerstin ,  KROLL, Hein-Peter ,  VON NUSSBAUM, Franz ,  RADDATZ, Siegfried ,  RUDOLPH, Joachim ,  SCHIFFER, Guido ,  SCHUMACHER, Andreas ,  CANCHO-GRANDE, Yolanda ,  MICHELS, Martin ,  WEIGAND, Stefan

IPC分类号： C07K5/00

CPC分类号： C07D245/04 ,  A61K38/00 ,  C07K5/0812

摘要： The invention relates to antibacterial amide macrocycles, to methods for the production thereof, and to the use of the same for producing pharmaceuticals for the treatment and/or prophylaxis of illness, especially bacterial infections.