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1.发明公开STEREOSELECTIVE PROCESS FOR PREPARING CYCLOHEXYL AMINE DERIVATIVES 审中-公开STEREO选择性工艺用于生产CYCLOHEXYLAMINDERIVATEN
公开(公告)号：EP1322652A1
公开(公告)日：2003-07-02
申请号：EP01975165.0
申请日：2001-09-13
IPC分类号： C07D498/04
CPC分类号： C07D498/04
摘要： A process for preparing (1R,3S)-3-(9-chloro-3-methyl-4-oxo-5H-(isoxazoloquinolin-5-yl))cyclohexanecarboxylic acid and esters thereof, as represented by formulas II and III, wherein R is a lower alkyl groups, and A and B are N or O, provided that when A is N, B is O, or when A is O, B is N: Formula (III) and Formula (II).
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公开(公告)号：EP1054859A1
公开(公告)日：2000-11-29
申请号：EP99903432.5
申请日：1999-01-27
发明人： BARNETT, Charles, Jackson , DUNLAP, Steven, Eugene , KOBIERSKI, Michael, Edward , WERNER, John, Arnold
IPC分类号： C07C255/00 , C07D207/02 , C07D211/04 , C07D213/02 , C07D231/02 , C07D231/04 , C07D231/06 , C07D231/10 , C07D233/02 , C07D233/04 , C07D233/54
CPC分类号： C07D471/04 , C07D333/38 , Y02P20/55
摘要： The present invention concerns intermediates, and processes directed to and from those intermediates, to a series of pyrimidine derivatives of formula (V), which are intermediates to useful antifolate compounds or are themselves useful antifolate compounds.
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3.发明授权PROCESS FOR PREPARING A 10,11-METHANODIBENZOSUBERANE DERIVATIVE 有权用于生产10,11METHANODIBENZOSUBERANDERIVATEN
公开(公告)号：EP1198462B1
公开(公告)日：2004-09-29
申请号：EP00935852.4
申请日：2000-05-30
发明人： ASTLEFORD, Bret, Anthony , BARNETT, Charles, Jackson , KOBIERSKI, Michael, Edward , WILSON, Thomas, Michael
IPC分类号： C07D401/04 , C07D295/02
CPC分类号： C07D295/073 , C07D215/20
摘要： This invention provides a process to prepare (2R)-anti-5-{3-[4-(10,11-difluoromethanodibenzosuber-5-yl)piperazin-1-yl]-2-hydroxypropoxy}quinoline.
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公开(公告)号：EP1198462A1
公开(公告)日：2002-04-24
申请号：EP00935852.4
申请日：2000-05-30
发明人： ASTLEFORD, Bret, Anthony , BARNETT, Charles, Jackson , KOBIERSKI, Michael, Edward , WILSON, Thomas, Michael
IPC分类号： C07D401/04 , C07D295/02
CPC分类号： C07D295/073 , C07D215/20
摘要： This invention provides a process to prepare (2R)-anti-5-{3-[4-(10,11-difluoromethanodibenzosuber-5-yl)piperazin-1-yl]-2-hydroxypropoxy}quinoline.
摘要翻译： 本发明提供了制备（2R） - 抗-5- {3- [4-（10,11-二氟甲基二苯并环戊烯-5-基）哌嗪-1-基] -2-羟基丙氧基}喹啉的方法。
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