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1.发明授权NEW PROCESS FOR THE PREPARATIION OF CYCLOHEXANECARBOXYLIC ACID DERICATIVES 有权VERFAHREN ZUR HERSTELLUNG VONCYCLOHEXANCARBOXYLSÄURE-DERIVATEN
公开(公告)号：EP2274278B1
公开(公告)日：2016-08-17
申请号：EP09728035.8
申请日：2009-03-26
发明人： HARNETT, Gerard, John , HOFFMANN, Ursula , JANSEN, Michael , REENTS, Reinhard , SATTELKAU, Tim , SMITH, Dennis, A. , STAHR, Helmut
IPC分类号： C07C253/30 , C07C255/46 , C07C231/06 , C07C233/58 , C07C51/06 , C07C61/08 , C07C323/42 , C07C329/10
CPC分类号： C07C233/58 , C07C51/06 , C07C253/30 , C07C2601/14 , C07C61/08 , C07C255/46
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2.发明授权SOLID FORMS OF (S)-2-METHOXY-3-{4-[2-(5-METHYL-2-PHENYL-OXAZOL-4-YL)-ETHOXY]-BENZO[B]THIOPHEN-7-YL}-PROPIONIC ACID AND OF SALTS THEREOF 有权（S）-2-甲氧基-3- {4- [2-（5-甲基-2-苯基 - 恶唑-4-基） - 乙氧基] -BENZO [B]噻吩-7-基] - 丙酸的固体形式 酸及其盐
公开(公告)号：EP2895469B1
公开(公告)日：2017-10-18
申请号：EP13759215.0
申请日：2013-09-09
发明人： DREIER, Lukas , EGLI, André , FAEHNRICH, Karsten , GRASSMANN, Olaf , MOHR, Peter , SCHWITTER, Urs , STAHR, Helmut , WYTTENBACH, Nicole
IPC分类号： C07D263/22 , A61K31/421 , A61P3/10
CPC分类号： A61K31/422 , C07D263/22
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公开(公告)号：EP2274278A1
公开(公告)日：2011-01-19
申请号：EP09728035.8
申请日：2009-03-26
发明人： HARNETT, Gerard, John , HOFFMANN, Ursula , JANSEN, Michael , REENTS, Reinhard , SATTELKAU, Tim , SMITH, Dennis, A. , STAHR, Helmut
IPC分类号： C07C253/30 , C07C255/46 , C07C231/06 , C07C233/58 , C07C51/06 , C07C61/08 , C07C323/42 , C07C329/10
CPC分类号： C07C233/58 , C07C51/06 , C07C253/30 , C07C2601/14 , C07C61/08 , C07C255/46
摘要： A process for the preparation of a compound of formula (Ia): which are useful as intermediates in the preparation of i.a. pharmaceutically active compounds.
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公开(公告)号：EP2323981B1
公开(公告)日：2014-03-12
申请号：EP09781167.3
申请日：2009-07-28
IPC分类号： C07D209/44 , C07D487/04
CPC分类号： C07D209/44 , C07D487/04 , Y02P20/55
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5.发明授权NEW PROCESS FOR THE PREPARATION OF CYCLOHEXANECARBOXYLIC ACID DERIVATIVES VIA THE CORRESPONDING CYCLOHEXANECARBOXAMIDE DERIVATIVE 有权通过相应的环己烷氨基甲酰胺衍生物制备环己烷羧酸衍生物的新方法
公开(公告)号：EP2274264B1
公开(公告)日：2014-02-12
申请号：EP09727723.0
申请日：2009-03-26
IPC分类号： C07C51/06 , C07C51/08 , C07C53/134 , C07C323/40 , C07C327/30 , C07C319/06 , C07C319/22 , C07C233/58 , C07C253/30
CPC分类号： C07C327/30 , C07C51/06 , C07C51/08 , C07C233/58 , C07C253/30 , C07C319/06 , C07C319/22 , C07C2601/14 , C07C53/134 , C07C323/42 , C07C255/46
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6.发明公开PROCESS FOR THE PREPARATION OF INSULIN SENSITIZER AND INTERMEDIATE COMPOUND THEREOF 审中-公开用于生产胰岛素产品中降低和中间化合物
公开(公告)号：EP1641790A1
公开(公告)日：2006-04-05
申请号：EP04740116.1
申请日：2004-06-21
IPC分类号： C07D419/14 , C07D333/54
CPC分类号： C07D417/14
摘要： The present invention is concerned with a novel process for the preparation of compounds of formula (I) and optionally converting a compound of formula (I) into a pharmaceutically acceptable salt, wherein R1 and R 2 are as defined in the description and claims. The compounds of formula (I) and the corresponding salts, e.g. the sodium salts, are pharmaceutically active substances.
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公开(公告)号：EP2323981A1
公开(公告)日：2011-05-25
申请号：EP09781167.3
申请日：2009-07-28
IPC分类号： C07D209/44 , C07D487/04
CPC分类号： C07D209/44 , C07D487/04 , Y02P20/55
摘要： The present invention relates to a new process for the preparation of macrocyclic HCV protease inhibitor compounds of the formula (XXII) wherein R
1 is an amino protecting group and X is halogen by way of a ring closing metathesis approach.-
8.发明公开NEW PROCESS FOR THE PREPARATION OF CYCLOHEXANECARBOXYLIC ACID DERIVATIVES VIA THE CORRESPONDING CYCLOHEXANECARBOXAMIDE DERIVATIVE 有权通过相应的环己烷氨基甲酰胺衍生物制备环己烷羧酸衍生物的新方法
公开(公告)号：EP2274264A1
公开(公告)日：2011-01-19
申请号：EP09727723.0
申请日：2009-03-26
IPC分类号： C07C51/06 , C07C51/08 , C07C53/134 , C07C323/40 , C07C327/30
CPC分类号： C07C327/30 , C07C51/06 , C07C51/08 , C07C233/58 , C07C253/30 , C07C319/06 , C07C319/22 , C07C2601/14 , C07C53/134 , C07C323/42 , C07C255/46
摘要： A process for the preparation of a compound of Formula (I): which are useful as intermediates in the preparation of i.a. pharmaceutically active compounds.
摘要翻译： 用于制备式（I）化合物的方法：其可用作制备i.a.中的中间体。 药学活性化合物。
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公开(公告)号：EP2150548B1
公开(公告)日：2010-12-08
申请号：EP08736214.1
申请日：2008-04-15
发明人： GANTZ, François , STAHR, Helmut
IPC分类号： C07D403/12 , C07D487/04
CPC分类号： C07D487/04 , C07D403/12 , Y02P20/55
摘要： The present invention relates to a new process for the preparation of diene compounds of the formula (I) wherein R1 is an amino protecting group and X is a halogen atom which may serve as intermediates for the manufacture of macrocyclic HCV protease inhibitors.
摘要翻译： 本发明涉及用于制备式（I）的二烯化合物的新方法，其中R 1是氨基保护基，X是卤素原子，其可以用作制备大环HCV蛋白酶抑制剂的中间体。
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公开(公告)号：EP2150548A1
公开(公告)日：2010-02-10
申请号：EP08736214.1
申请日：2008-04-15
发明人： GANTZ, François , STAHR, Helmut
IPC分类号： C07D403/12 , C07D487/04
CPC分类号： C07D487/04 , C07D403/12 , Y02P20/55
摘要： The present invention relates to a new process for the preparation of diene compounds of the formula (I) wherein R1 is an amino protecting group and X is a halogen atom which may serve as intermediates for the manufacture of macrocyclic HCV protease inhibitors.
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