Benzylamine derivatives, process for production thereof, and use thereof
    6.
    发明公开
    Benzylamine derivatives, process for production thereof, and use thereof 失效
    苯甲酰胺衍生物,其生产方法及其用途

    公开(公告)号:EP0221781A3

    公开(公告)日:1988-08-17

    申请号:EP86308505

    申请日:1986-10-31

    CPC分类号: A61K31/135

    摘要: Benzylamine derivative of the following general formula (I)
    wherein R₁ represents an alkyl group, R₂ represents a group of the formula
    in which R₄ represents a hydrogen atom, a lower alkyl group or a halogen atom, and
    R₃ represents an alkyl or alkenyl group, can be produced by reacting a compound represented by the general formula (III)
    R₂-NH-R₃ (III)
    wherein R₂ and R₃ are as defined above, with a compound represented by the general formula (IV)
    wherein R₁ is as defined and X represents a reactive residue, or reacting a compound represented by the general formula (V)
    wherein R₁ and R₃ are as defined, with a compound represented by the general formula (VI)
    X-R₂ (VI)
    wherein X and R₂ are as defined, or reacting a compound represented by the general formula (VII)
    wherein R₁ and R₂ are as defined above, with a compound represented by the general formula (VIII)
    X-R₃ (VIII)
    wherein R₃ and X are as defined above. These compounds are useful for the treatment of animal epidemics or infectious diseases induced by fungi as an antimycotic agent for humans and animals, for the control of plant diseases as an agricultural fungicide, and for the control of fungi and bacteria in industrial materials or products as an industrial fungicide.

    Benzylamine derivatives, process for production thereof, and use thereof
    7.
    发明公开
    Benzylamine derivatives, process for production thereof, and use thereof 失效
    苄胺衍生物,它们的制备和它们的用途。

    公开(公告)号:EP0221781A2

    公开(公告)日:1987-05-13

    申请号:EP86308505.6

    申请日:1986-10-31

    CPC分类号: A61K31/135

    摘要: Benzylamine derivative of the following general formula (I)
    wherein R₁ represents an alkyl group, R₂ represents a group of the formula
    in which R₄ represents a hydrogen atom, a lower alkyl group or a halogen atom, and
    R₃ represents an alkyl or alkenyl group, can be produced by reacting a compound represented by the general formula (III)
    R₂-NH-R₃ (III)
    wherein R₂ and R₃ are as defined above, with a compound represented by the general formula (IV)
    wherein R₁ is as defined and X represents a reactive residue,
    or reacting a compound represented by the general formula (V)
    wherein R₁ and R₃ are as defined, with a compound represented by the general formula (VI)
    X-R₂ (VI)
    wherein X and R₂ are as defined, or reacting a compound represented by the general formula (VII)
    wherein R₁ and R₂ are as defined above, with a compound represented by the general formula (VIII)
    X-R₃ (VIII)
    wherein R₃ and X are as defined above. These compounds are useful for the treatment of animal epidemics or infectious diseases induced by fungi as an antimycotic agent for humans and animals, for the control of plant diseases as an agricultural fungicide, and for the control of fungi and bacteria in industrial materials or products as an industrial fungicide.

    Amide derivatives, processes for production thereof, and agricultural-horticultural fungicide containing them
    9.
    发明公开
    Amide derivatives, processes for production thereof, and agricultural-horticultural fungicide containing them 失效
    酰胺衍生物,它们的制备方法和含有在农业和园艺这些化合物的杀真菌剂。

    公开(公告)号:EP0313091A2

    公开(公告)日:1989-04-26

    申请号:EP88117606.9

    申请日:1988-10-21

    摘要: An amide derivative represented by the following general formula (I)
    wherein one of X and Y represents a sulfur atom and the other represents a carbon atom, Z represents a nitrile or thioamide group, each of R 1 and R 2 represents a hydrogen atom, a halogen atom, an alkyl group having 1 to 6 carbon atoms, a halomethyl group or a phenyl group, and R 3 represents an alkenyl group having 2 to 6 carbon atoms, a haloalkenyl group having 2 to 4 carbon atoms, a furyl group, a thienyl group, an alkoxy group having 1 to 4 carbon atoms, an alkylthio group having 1 to 4 carbon atoms, an alkynyloxy group having 3 to 5 carbon atoms, an alkynylthio group having 3 to 5 carbon atoms, a pyrazolyl group, or an unsubstituted or halo-substituted phenyl group;
    processes for producing the amide derivative; an agricultural-horticultural fungicide comprising the amide derivative as an active ingredient; and to an agricultural-horticultural fungicidal composition comprising the amide derivative of general formula (I) as an active ingredient.

    摘要翻译: 由下述通式(I) worin X和Y中的一个表示的酰胺衍生物darstellt硫原子,另一个darstellt的碳原子,Z darstellt腈或硫代酰胺基团,每个R <1>和R <的 2>代表氢原子,卤原子,在具有1至6个碳原子,卤代甲基或苯基,且R烷基<3> darstellt具有2至6个碳原子的链烯基,具有2卤代烯基 至4个碳原子,呋喃基,噻吩基,在具有1至4个碳原子的具有1至4个碳原子的具有3-5个碳原子具有3至5炔硫基炔氧基烷硫基烷氧基 碳原子,吡唑基,或在unsubstituiertem或卤素取代的苯基; 用于制备酰胺衍生物过程; 农业园艺用杀菌剂,其包括作为活性成分的酰胺衍生物; 并在农业园艺用杀菌剂组合物包含通式(I)作为在活性成分的酰胺衍生物。