Patent search ap:("Merck Sharp & Dohme Corp.") AND inv:"FULLER Page Peter

1.

发明授权
SUBSTITUTED BICYCLIC PYRAZOLE COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF 有权

公开(公告)号：EP3368516B1

公开(公告)日：2020-07-15

申请号：EP16860767.9

申请日：2016-10-27

Applicant: Merck Sharp & Dohme Corp.

Inventor： LAPOINTE, Blair, T. , FULLER, Peter, H. , GUNAYDIN, Hakan , LIU, Kun , MOLINARI, Danielle, F. , PU, Qinglin , SCOTT, Mark, E. , TROTTER, B., Wesley , ZHANG, Hongjun

IPC: C07D231/56 , C07D491/052 , C07D491/107 , C07D487/04 , C07D401/04 , A61K31/4162 , A61K31/416 , A61K31/4439 , A61K31/437 , A61P29/00 , A61P37/00

2.

发明公开
N-HETEROARYL INDAZOLE DERIVATIVES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF 审中-公开

公开(公告)号：EP3873471A1

公开(公告)日：2021-09-08

申请号：EP19879334.1

申请日：2019-10-25

Applicant: Merck Sharp & Dohme Corp.

Inventor： SIMOV, Vladimir , KAPLAN, William, P. , ACTON, John, J., III , ARDOLINO, Michael, J. , CHEN, Joanna, L. , FULLER, Peter, H. , GUNAYDIN, Hakan , LI, Derun , LIU, Ping , LOGAN, Kaitlyn Marie , METHOT, Joey , MORRIELLO, Gregori, J. , NEELAMKAVIL, Santhosh, F. , TORRES, Luis , YAN, Xin , ZHOU, Hua

IPC: A61K31/4985 , A61K31/519 , C07D471/04

3.

发明授权
SUBSTITUTED INDAZOLE COMPOUNDS AS ROR GAMMA T INHIBITORS AND USES THEREOF 有权

公开(公告)号：EP3368539B1

公开(公告)日：2020-12-02

申请号：EP16860768.7

申请日：2016-10-27

Applicant: Merck Sharp & Dohme Corp.

Inventor： LAPOINTE, Blair, T. , FULLER, Peter, H. , GUNAYDIN, Hakan , LIU, Kun , SCOTT, Mark, E. , TROTTER, B., Wesley , ZHANG, Hongjun

IPC: C07D487/10 , C07D403/06 , C07D403/14 , C07D403/12 , C07D491/107 , C07D487/04 , C07D491/048 , C07D231/56 , C07D405/12 , A61K31/416 , A61K31/495 , A61K31/506 , A61K31/454 , A61K31/4439 , A61K31/4162 , A61K31/445 , A61P29/00 , A61P37/00 , A61P19/02 , A61P11/06

4.

发明公开
INDAZOLYL-SPIRO[2.2]PENTANE-CARBONITRILE DERIVATIVES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF 审中-公开

公开(公告)号：EP3694330A1

公开(公告)日：2020-08-19

申请号：EP18867260.4

申请日：2018-10-08

Applicant: Merck Sharp & Dohme Corp.

Inventor： CANDITO, David Annunziato , GRAHAM, Thomas, H. , ACTON, John , CHAU, Ryan Wing-Kun , CHEN, Joanna, L. , ELLIS, J. Michael , FULLER, Peter, H. , GULATI, Anmol , GUNAYDIN, Hakan , KATTAR, Solomon , KEYLOR, Mitchell Henry , LAPOINTE, Blair, T. , LIU, Ping , LIU, Weiguo , METHOT, Joey, L. , NEELAMKAVIL, Santhosh, F. , SIMOV, Vladimir , TONG, Ling , WOOD, Harold, B.

IPC: A01N43/42 , C07D487/04

5.

发明公开
1-PYRAZOLYL, 5-, 6- DISUBSTITUTED INDAZOLE DERIVATIVES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF 审中-公开

公开(公告)号：EP3980412A2

公开(公告)日：2022-04-13

申请号：EP20817991.1

申请日：2020-06-01

Applicant: Merck Sharp & Dohme Corp.

Inventor： ZHOU, Hua , ACTON, John, J., III , ARDOLINO, Michael, J. , CHEN, Yi-Heng , FULLER, Peter, H. , GULATI, Anmol , JOHNSON, Rebecca Elizabeth , KAPLAN, William, P. , KATTAR, Solomon, D. , KEYLOR, Mitchell, H. , LI, Derun , LOGAN, Kaitlyn Marie , LU, Min , MORRIELLO, Gregori, J. , NEELAMKAVIL, Santhosh, F. , PIO, Barbara , SCIAMMETTA, Nunzio , SIMOV, Vladimir , SU, Jing , TORRES, Luis , YAN, Xin

IPC: C07D401/14 , C07D403/12 , C07D403/14

6.

发明公开
SUBSTITUTED INDAZOLE COMPOUNDS AS RORGAMMAT INHIBITORS AND USES THEREOF 审中-公开

公开(公告)号：EP3368539A1

公开(公告)日：2018-09-05

申请号：EP16860768.7

申请日：2016-10-27

Applicant: Merck Sharp & Dohme Corp.

Inventor： LAPOINTE, Blair, T. , FULLER, Peter, H. , GUNAYDIN, Hakan , LIU, Kun , SCOTT, Mark, E. , TROTTER, B., Wesley , ZHANG, Hongjun

IPC: C07D487/10 , C07D403/06 , C07D403/14 , C07D403/12 , C07D491/107 , C07D487/04 , C07D491/048 , C07D231/56 , C07D405/12 , A61K31/416 , A61K31/495 , A61K31/506 , A61K31/454 , A61K31/4439 , A61K31/4162 , A61K31/445 , A61P29/00 , A61P37/00 , A61P19/02 , A61P11/06

CPC classification number: C07D403/08 , A61P19/02 , C07D231/56 , C07D401/06 , C07D401/12 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/12 , C07D487/04 , C07D487/10 , C07D491/048 , C07D491/107

Abstract: The present invention relates to compounds according to Formula (I) and pharmaceutically acceptable salts thereof. Such compounds can be used in the treatment of RORgammaT-mediated diseases or conditions.

7.

发明公开
SUBSTITUTED BICYCLIC PYRAZOLE COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF 审中-公开

公开(公告)号：EP3368516A1

公开(公告)日：2018-09-05

申请号：EP16860767.9

申请日：2016-10-27

Applicant: Merck Sharp & Dohme Corp.

Inventor： LAPOINTE, Blair, T. , FULLER, Peter, H. , GUNAYDIN, Hakan , LIU, Kun , MOLINARI, Daneille, F. , PU, Qinglin , SCOTT, Mark, E. , TROTTER, B., Wesley , ZHANG, Hongjun

IPC: C07D231/56 , C07D491/052 , C07D491/107 , C07D487/04 , C07D401/04 , A61K31/4162 , A61K31/416 , A61K31/4439 , A61K31/437 , A61P29/00 , A61P37/00

CPC classification number: C07D231/56 , A61K2121/00 , A61P11/06 , A61P17/06 , A61P19/02 , A61P29/00 , A61P37/02 , C07D401/04 , C07D471/04 , C07D491/052 , C07D491/107

Abstract: The present invention relates to compounds according to Formula I: and pharmaceutically acceptable salts thereof. Such compounds can be used in the treatment of RORgammaT-mediated diseases or conditions.

8.

发明公开
INDAZOLYL-SPIRO[2.3]HEXANE-CARBONITRILE DERIVATIVES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF 审中-公开

公开(公告)号：EP3694331A1

公开(公告)日：2020-08-19

申请号：EP18867261.2

申请日：2018-10-08

Applicant: Merck Sharp & Dohme Corp.

Inventor： ACTON, John , CANDITO, DavidAnnunziato , ELLIS, J. Michael , FULLER, Peter, H. , GUNAYDIN, Hakan , LAPOINTE, Blair, T. , LIU, Weiguo , METHOT, Joey, L. , NEELAMKAVIL, Santhosh, F. , PIO, Barbara , SIMOV, Vladimir , WOOD, Harold, B.

IPC: A01N43/42 , C07D487/04

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