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公开(公告)号:EP3368516B1
公开(公告)日:2020-07-15
申请号:EP16860767.9
申请日:2016-10-27
Applicant: Merck Sharp & Dohme Corp.
Inventor: LAPOINTE, Blair, T. , FULLER, Peter, H. , GUNAYDIN, Hakan , LIU, Kun , MOLINARI, Danielle, F. , PU, Qinglin , SCOTT, Mark, E. , TROTTER, B., Wesley , ZHANG, Hongjun
IPC: C07D231/56 , C07D491/052 , C07D491/107 , C07D487/04 , C07D401/04 , A61K31/4162 , A61K31/416 , A61K31/4439 , A61K31/437 , A61P29/00 , A61P37/00
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2.
公开(公告)号:EP3694331A1
公开(公告)日:2020-08-19
申请号:EP18867261.2
申请日:2018-10-08
Applicant: Merck Sharp & Dohme Corp.
Inventor: ACTON, John , CANDITO, DavidAnnunziato , ELLIS, J. Michael , FULLER, Peter, H. , GUNAYDIN, Hakan , LAPOINTE, Blair, T. , LIU, Weiguo , METHOT, Joey, L. , NEELAMKAVIL, Santhosh, F. , PIO, Barbara , SIMOV, Vladimir , WOOD, Harold, B.
IPC: A01N43/42 , C07D487/04
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公开(公告)号:EP3368535A1
公开(公告)日:2018-09-05
申请号:EP16860770.3
申请日:2016-10-27
Applicant: Merck Sharp & Dohme Corp.
Inventor: ZHANG, Hongjun , BARR, Kenneth, Jay , LAPOINTE, Blair, T. , GUNAYDIN, Hakan , LIU, Kun , TROTTER, B., Wesley
IPC: C07D471/04 , A61K31/437 , A61P37/00 , A61P29/00
CPC classification number: C07D471/04
Abstract: The present invention relates to compounds according to Formula I and pharmaceutically acceptable salts thereof. Such compounds can be used in the treatment of RORgammaT-mediated diseases or conditions.
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4.
公开(公告)号:EP3873471A1
公开(公告)日:2021-09-08
申请号:EP19879334.1
申请日:2019-10-25
Applicant: Merck Sharp & Dohme Corp.
Inventor: SIMOV, Vladimir , KAPLAN, William, P. , ACTON, John, J., III , ARDOLINO, Michael, J. , CHEN, Joanna, L. , FULLER, Peter, H. , GUNAYDIN, Hakan , LI, Derun , LIU, Ping , LOGAN, Kaitlyn Marie , METHOT, Joey , MORRIELLO, Gregori, J. , NEELAMKAVIL, Santhosh, F. , TORRES, Luis , YAN, Xin , ZHOU, Hua
IPC: A61K31/4985 , A61K31/519 , C07D471/04
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公开(公告)号:EP3368539B1
公开(公告)日:2020-12-02
申请号:EP16860768.7
申请日:2016-10-27
Applicant: Merck Sharp & Dohme Corp.
Inventor: LAPOINTE, Blair, T. , FULLER, Peter, H. , GUNAYDIN, Hakan , LIU, Kun , SCOTT, Mark, E. , TROTTER, B., Wesley , ZHANG, Hongjun
IPC: C07D487/10 , C07D403/06 , C07D403/14 , C07D403/12 , C07D491/107 , C07D487/04 , C07D491/048 , C07D231/56 , C07D405/12 , A61K31/416 , A61K31/495 , A61K31/506 , A61K31/454 , A61K31/4439 , A61K31/4162 , A61K31/445 , A61P29/00 , A61P37/00 , A61P19/02 , A61P11/06
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6.
公开(公告)号:EP3694330A1
公开(公告)日:2020-08-19
申请号:EP18867260.4
申请日:2018-10-08
Applicant: Merck Sharp & Dohme Corp.
Inventor: CANDITO, David Annunziato , GRAHAM, Thomas, H. , ACTON, John , CHAU, Ryan Wing-Kun , CHEN, Joanna, L. , ELLIS, J. Michael , FULLER, Peter, H. , GULATI, Anmol , GUNAYDIN, Hakan , KATTAR, Solomon , KEYLOR, Mitchell Henry , LAPOINTE, Blair, T. , LIU, Ping , LIU, Weiguo , METHOT, Joey, L. , NEELAMKAVIL, Santhosh, F. , SIMOV, Vladimir , TONG, Ling , WOOD, Harold, B.
IPC: A01N43/42 , C07D487/04
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公开(公告)号:EP3525786A1
公开(公告)日:2019-08-21
申请号:EP17860647.1
申请日:2017-10-06
Applicant: Merck Sharp & Dohme Corp.
Inventor: MANSOOR, Umar Faruk , FISCHER, Christian , SILIPHAIVANH, Phieng , GUNAYDIN, Hakan
IPC: A61K31/4353 , C07D471/04
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公开(公告)号:EP3525785A1
公开(公告)日:2019-08-21
申请号:EP17859538.5
申请日:2017-10-06
Applicant: Merck Sharp & Dohme Corp.
Inventor: MANSOOR, Umar Faruk , FISCHER, Christian , SILIPHAIVANH, Phieng , TORRES, Luis , GUNAYDIN, Hakan , SLOMAN, David, L.
IPC: A61K31/4353 , C07D471/04
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公开(公告)号:EP3765006A1
公开(公告)日:2021-01-20
申请号:EP19767942.6
申请日:2019-03-08
Applicant: Merck Sharp & Dohme Corp.
Inventor: ACHAB, Abdelghani Abe , CHILDERS, Matthew, L. , CUMMING, Jared, N. , FISCHER, Christian , GATHIAKA, Symon , GUNAYDIN, Hakan , LESBURG, Charles, A. , LI, Derun , LU, Min , PALANI, Anandan , PALTE, Rachel, L. , PU, Qinglin , SLOMAN, David, L. , SO, Sung-Sau , SUN, Chunrui , ZHANG, Hongjun
IPC: A61K31/195 , A61K31/69 , C07F5/02
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公开(公告)号:EP3368535B1
公开(公告)日:2020-12-02
申请号:EP16860770.3
申请日:2016-10-27
Applicant: Merck Sharp & Dohme Corp.
Inventor: ZHANG, Hongjun , BARR, Kenneth, Jay , LAPOINTE, Blair, T. , GUNAYDIN, Hakan , LIU, Kun , TROTTER, B., Wesley
IPC: A61P11/06 , A61P19/02 , C07D471/04 , A61P29/00 , A61P37/00
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