PESTICIDAL PYRIMIDINE-DERIVATIVES
    3.
    发明授权
    PESTICIDAL PYRIMIDINE-DERIVATIVES 有权
    PESTZIDES嘧啶衍生物

    公开(公告)号:EP1175407B1

    公开(公告)日:2009-12-09

    申请号:EP00931096.2

    申请日:2000-05-02

    申请人: Novartis AG

    摘要: The invention relates to compounds of general formula (I), wherein R1 is unsubstituted or mono- to penta-substituted aryl, whereby the substituents are selected from the group consisting for instance of OH, halogen, CN, C1-C6-alkyl, optionally substituted C3-C8-cycloalkyl and optionally substituted C3-C8-cycloalkenyl; A is for instance a single bond, C1-C12-alkylene or O; X1 and X2, independently of one another, are R10; X3 is H or R10; R10 is for instance halogen, CN, NO2, C1-C6-alkyl, C3-C8-cycloalkyl or C1-C6-haloalkyl; R21 and R22, independently of one another are for instance H, halogen, CN, NO2, OH, SH, C1-C6-alkyl, C3-C8-cycloalkyl, C1-C6-alkyl-C3-C8-cycloalkyl or C3-C8-cycloalkyl-C1-C6-alkyl; R23 and R24, independently of one another, are for instance H, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, C1-C6-haloalkyl or C3-C8-halocycloalkyl; m is 1, 2, 3 or 4; and n is 0, 1 or 2; as well as the physiologically acceptable addition compounds, a method of producing these compounds and the usage of these compounds, pesticide compositions whose active ingredient is chosen from these compounds, each in free form or in agrochemically employable salt form, and a method of producing and using these compositions. The active ingredients, in free form or in agrochemically employable salt form, have advantageous pesticidal properties. They are especially suitable for the control of pests in agriculture and in storage, as well as in the care of domestic animals.

    PESTICIDAL PYRIDINE THIOAMIDES
    4.
    发明公开
    PESTICIDAL PYRIDINE THIOAMIDES 失效
    吡啶硫酰胺AS农药

    公开(公告)号:EP0790983A1

    公开(公告)日:1997-08-27

    申请号:EP95937839.0

    申请日:1995-10-25

    申请人: Novartis AG

    摘要: Compounds of formula (I), wherein, R1 and R2 are each independently of the other C1-C6alkyl, halo-C1-C6alkyl containing 1-5 halogen atoms, C1-C2alkoxy-C1-C6alkyl, nitro-C1-C6alkyl, cyano-C1-C6alkyl, C1-C2alkanoyl-C1-C6alkyl, C1-C2akloxycarbonyl-C1-C6alkyl, C1-C2alkylthio-C1-C6alkyl, C1-C2alkanesulfinyl-C1-C6alkyl, C1-C2alkanesulfonyl-C1-C6alkyl, C2-C6alkenyl, halo-C2-C6alkenyl containing 1-5 halogen atoms, C2-C6alkynyl, halo-C2-C6alkynyl containing 1-5 halogen atoms, C3-C7cycloalkyl or halogen; or R1 and R2, taken together, form a saturated or unsaturated 5- to 7-membered unsubstituted or substituted carbocyclic or heterocyclic ring which may contain one or two hetero atoms selected from O and S; R3 and R4 are each independently of the other hydrogen, C1-C6alkyl or halogen; R5 is hydrogen, C1-C6alkyl which is unsubstituted or substituted by cyano, nitro, halogen, carboxyl, C1-C2alkoxycarbonyl, C1-C2alkanoyl, C1-C2alkanesulfonyl or phenylsulfonyl, C2-C6alkenyl, C2-C6alkynyl or benzyl; X is (CH2)n, CH=CH, or C≡C; Y is an unsubstituted or substituted 5-8-membered carbocyclic or heterocyclic ring which can be saturated or unsaturated, aromatic or nonaromatic and which may contain 1 or 2 hetero atoms selected from O, S and/or N and to which a further aromatic group can be fused; n is 1, 2, 3 or 4; or tautomers thereof, in the free form or in the form of a salt, are pesticidal compounds. Said compounds can be used for the control of pests, in particular as microbicides, insecticides and acaracides in agriculture, horticulture and in the hygiene sector.