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8 条记录 (耗时 0.017 秒)

    PESTICIDAL PYRIMIDINE-DERIVATIVES
    1.
    发明授权
    PESTICIDAL PYRIMIDINE-DERIVATIVES 有权
    PESTZIDES嘧啶衍生物

    公开(公告)号：EP1175407B1

    公开(公告)日：2009-12-09

    申请号：EP00931096.2

    申请日：2000-05-02

    申请人： Novartis AG

    发明人： EBERLE, Martin ,  JEANGUENAT, André ,  ZAMBACH, Werner ,  STEIGER, Arthur ,  FAROOQ, Saleem

    IPC分类号： C07D239/26 ,  C07D239/28 ,  C07D239/36 ,  C07D239/42 ,  C07D239/54 ,  C07D239/30 ,  C07D239/74 ,  A01N43/54

    CPC分类号： C07D239/26 ,  A01N43/54 ,  C07D239/28 ,  C07D239/34 ,  C07D239/36 ,  C07D239/42 ,  C07D239/54

    摘要： The invention relates to compounds of general formula (I), wherein R1 is unsubstituted or mono- to penta-substituted aryl, whereby the substituents are selected from the group consisting for instance of OH, halogen, CN, C1-C6-alkyl, optionally substituted C3-C8-cycloalkyl and optionally substituted C3-C8-cycloalkenyl; A is for instance a single bond, C1-C12-alkylene or O; X1 and X2, independently of one another, are R10; X3 is H or R10; R10 is for instance halogen, CN, NO2, C1-C6-alkyl, C3-C8-cycloalkyl or C1-C6-haloalkyl; R21 and R22, independently of one another are for instance H, halogen, CN, NO2, OH, SH, C1-C6-alkyl, C3-C8-cycloalkyl, C1-C6-alkyl-C3-C8-cycloalkyl or C3-C8-cycloalkyl-C1-C6-alkyl; R23 and R24, independently of one another, are for instance H, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, C1-C6-haloalkyl or C3-C8-halocycloalkyl; m is 1, 2, 3 or 4; and n is 0, 1 or 2; as well as the physiologically acceptable addition compounds, a method of producing these compounds and the usage of these compounds, pesticide compositions whose active ingredient is chosen from these compounds, each in free form or in agrochemically employable salt form, and a method of producing and using these compositions. The active ingredients, in free form or in agrochemically employable salt form, have advantageous pesticidal properties. They are especially suitable for the control of pests in agriculture and in storage, as well as in the care of domestic animals.

    PROCESS FOR THE PREPARATION OF PESTICIDES
    2.
    发明公开
    PROCESS FOR THE PREPARATION OF PESTICIDES 失效
    工艺对农药的研制

    公开(公告)号：EP0876333A1

    公开(公告)日：1998-11-11

    申请号：EP96939928.0

    申请日：1996-11-26

    申请人： Novartis AG

    发明人： FAROOQ, Saleem ,  TRAH, Stephan ,  ZIEGLER, Hugo ,  ZURFLÜH, René

    IPC分类号： C07C249 ,  C07C251

    CPC分类号： C07C249/12 ,  C07C251/48 ,  C07C251/60

    摘要： The invention relates to a process for the preparation of compounds of formula (I), or, if appropriate, a tautomer thereof, in each case in the free form or in salt form, in which A, X, Y, Z, R2, R3, R4, R5, R7, R9 and n are as defined in claim 1 and the C=N double bond marked with E has the E configuration, which comprises: a1) reacting either a compound of formula (II) mentioned in the description with a compound of formula (III) mentioned in the description, in which X1 is a leaving group; or a2) a compound of formula (IV) mentioned in the description, if appropriate in the presence of a base, with a compound of formula (V) mentioned in the description; or b1) reacting a compound of formula (IV) mentioned in the description with a compound of the formula R7-A-X2 (VII), in which X2 is a leaving group, and either further reacting the compound thus obtainable, of formula (IV), for example according to method a2); or b2) reacting it with hydroxylamine or a salt thereof, if appropriate in the presence of a basic or acid catalyst, and further reacting the compound thus obtainable, of formula (II), for example according to method a1); or c) reacting a compound of formula (VIII), mentioned in the description with a C1-C6alkyl nitrite and further reacting the compound thus obtainable, of formula (VI), for example according to method b), the E isomers of the compounds of the formulae (II), (IV) and (VI), a process for their preparation and their use for the preparation of compounds of formula (I).

    O-BENZYL OXIME ETHER DERIVATIVES AND THEIR USE AS PESTICIDES
    5.
    发明公开
    O-BENZYL OXIME ETHER DERIVATIVES AND THEIR USE AS PESTICIDES 失效
    O-苄基肟醚衍生物及其作为杀虫剂的用途

    公开(公告)号：EP0984924A1

    公开(公告)日：2000-03-15

    申请号：EP98932082.5

    申请日：1998-05-25

    申请人： Novartis AG ,  Novartis-Erfindungen Verwaltungsgesellschaft m.b.H.

    发明人： TRAH, Stephan ,  FAROOQ, Saleem

    IPC分类号： C07C251/60 ,  A01N37/50

    CPC分类号： C07C251/60

    摘要： Described are compounds of formula (I), wherein either X is CH or N, Y is OR1 and Z is O, or X is N, Y is NHR8 and Z is O, S or S(=O); R1 is C1-C4alkyl; R2 is C2-C4alkyl or C3-C6cycloalkyl; R3 and R4 are each independently of the other, for example, H, C1-C4alkyl or C1-C4-alkoxy; R8 is H or C1-C4alkyl; R9 is methyl, fluoromethyl or difluoromethyl; A is a direct bond, C1-C10alkylene, -C(=O)-, -C(=S)- or halo-C1-C10alkylene and R7 is a radical R10; or A is C1-C10alkylene, -C(=O)-, -C(=S)- or halo-C1-C10alkylene and R7 is -CN, OR10, N(R10)2 or -S(=O)pR10; p is 0, 1 or 2; G is O, S or -O-CH2-; R5 and R6 are each inter alia unsubstituted or substituted C1-C6alkyl, C3-C6cycloalkyl, C1-C6alkoxy, C1-C6alkylthio, C1-C6alkylsulfynyl, C1-C6alkylsulfonyl or C1-C6alkylsulfonyloxy and R10 is H or, for example, unsubstituted or substituted C1-C6alkyl, C2-C8alkenyl, C2-C8-alkynyl or C3-C6cycloalkyl; a process for the preparation of those compounds and their use; pesticides, the active ingredient of which is selected from those compounds; and a method of preparing those compositions and their use; intermediates in the preparation of those compounds; and a process for the preparation of those intermediates and their use.

    摘要翻译： 描述了式（I）的化合物，其中X为CH或N，Y为OR1且Z为O，或X为N，Y为NHR8且Z为O，S或S（= O）。 R1是C1-C4烷基; R2是C2-C4烷基或C3-C6环烷基; R3和R4各自相互独立，例如H，C1-C4烷基或C1-C4烷氧基; R8是H或C1-C4烷基; R9是甲基，氟甲基或二氟甲基; A是直接键，C 1 -C 10亚烷基，-C（= O） - ， - C（= S） - 或卤代-C 1 -C 10亚烷基并且R 7是基团R 10; 或者A是C 1 -C 10亚烷基，-C（= O） - ， - C（= S） - 或卤代-C 1 -C 10亚烷基和R 7是-CN，OR 10，N（R 10）2或-S（= O） p是0,1或2; G是O，S或-O-CH 2 - ; R5和R6各自为未取代的或取代的C1-C6烷基，C3-C6环烷基，C1-C6烷氧基，C1-C6烷硫基，C1-C6烷基亚磺酰基， -C 6烷基，C 2 -C 8烯基，C 2 -C 8炔基或C 3 -C 6环烷基; 制备这些化合物的方法及其用途; 农药，其活性成分选自那些化合物; 以及制备这些组合物及其用途的方法; 在制备这些化合物中的中间体; 以及制备这些中间体及其用途的方法。

    O-BENZYL OXIME ETHERS AND THEIR USE AS PESTICIDES
    7.
    发明公开
    O-BENZYL OXIME ETHERS AND THEIR USE AS PESTICIDES 失效
    O-苄基肟醚及其作为杀虫剂的用途

    公开(公告)号：EP0984923A1

    公开(公告)日：2000-03-15

    申请号：EP98932081.7

    申请日：1998-05-25

    申请人： Novartis AG ,  Novartis-Erfindungen Verwaltungsgesellschaft m.b.H.

    发明人： TRAH, Stephan ,  SZCZEPANSKI, Henry ,  HÜTER, Ottmar, Franz ,  HALL, Roger, Graham ,  FAROOQ, Saleem ,  PASCUAL, Alfons

    IPC分类号： C07C251/60 ,  C07D261/08 ,  C07D261/20 ,  A01N37/50

    CPC分类号： C07F9/4021 ,  C07C251/60 ,  C07D261/08 ,  C07D261/20 ,  C07F9/3229 ,  C07F9/5325

    摘要： Compounds of formula (I), wherein either X is CH or N, Y is OR1 and Z is O, or X is N, Y is NHR8 and Z is O, S or S (=O); R1, R2 and R3 are as defined according to the specification; m is 0, 1 or 2; R5 is, for example, halogen, C1-C6alkyl, halo-C1-C6alkyl or C3-C6cycloalkyl; n is 0, 1, 2, 3 or 4; R9 is methyl, fluoromethyl or difluoromethyl; A and R7 are as defined according to the specification; D is O, S, -S(=O) or S(=O)2; G is C1-C8alkylene; T-R6 is R6, -C(=N-O-A1-R77)-R6; -SiR14(R15)-R6; -C(=O)-R6; -C(R16)=C(R17)-R6, -C≡C-R6 or -D-R6; R6 is C1-C4alkyl or unsubstituted or substituted aryl or heteroaryl; A1 and R77 are as defined above for A and R7; L is U-R18, P(O)vR11R12, P(S)wR11R12 or N(aryl)R13; v and w are 0 or 1; U-R18 is -C(=O)-C(=O)-R18; -C(OH)-C(OH)-R18; -C(=N-O-A1-R7)-R18; (i) or (ii); a is 0 or 1; b is 0 or 1; R11, R12 and R13 are, for example, C1-C6alkyl, halo-C1-C6alkyl or C3-C6cycloalkyl; R14 and R15 are each independently of the other C1-C4alkyl; R16 and R17 are each independently of the other hydrogen, C1-C4alkyl or halogen and R18 is R5; and, where applicable, their possible E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form, a method of controlling pests, a process for the preparation of those compounds and their use are described.

    摘要翻译： 其中X是CH或N，Y是OR1且Z是O，或X是N，Y是NHR8且Z是O，S或S（= O）的式（I）化合物。 R1，R2和R3如根据说明书所定义; m是0,1或2; R5是例如卤素，C1-C6烷基，卤代-C1-C6烷基或C3-C6环烷基; n是0,1,2,3或4; R9是甲基，氟甲基或二氟甲基; A和R7如根据说明书所定义; D是O，S，-S（= O）或S（= O）2; G是C1-C8亚烷基; T-R6是R6，-C（= N-O-A1-R77）-R6; -SiR14（R15）-R 6; -C（= O）-R 6; -C（R 16）= C（R 17）-R 6，-C≡C-R 6或-D-R 6; R6是C1-C4烷基或未取代或取代的芳基或杂芳基; A1和R77如以上A和R7所定义; L是U-R18，P（O）vR11R12，P（S）wR11R12或N（芳基）R13; v和w是0或1; U-R18是-C（= O）-C（= O）-R18; -C（OH）-C（OH）-R18; -C（= N-O-A1-R7）-R18; （i）或（ii）; a是0或1; b是0或1; 例如，R 11，R 12和R 13是C 1 -C 6烷基，卤代-C 1 -C 6烷基或C 3 -C 6环烷基; R14和R15各自独立于另一个C1-C4烷基; R 16和R 17各自独立地为氢，C 1 -C 4烷基或卤素且R 18为R 5; 并且在适用的情况下，它们可能的E / Z异构体，E / Z异构体和/或互变异构体的混合物，各自以游离形式或盐形式存在，控制害虫的方法，制备这些化合物及其 描述使用。