公开(公告)号：EP1863795B1

公开(公告)日：2008-10-29

申请号：EP06710566.8

申请日：2006-03-08

申请人： Pfizer Limited

发明人： CALABRESE, Andrew, Antony

IPC分类号： C07D401/14 ,  A61K31/497 ,  A61P5/10

CPC分类号： C07D401/14

摘要： The present invention relates to a class of substituted triazoles of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).

公开(公告)号：EP1758910A1

公开(公告)日：2007-03-07

申请号：EP05741010.2

申请日：2005-05-27

申请人： Pfizer Limited ,  Brown, Alan Daniel

发明人： BROWN, Alan Daniel ,  CALABRESE, Andrew, Antony ,  ELLIS, David ,  WATSON, Lesa

IPC分类号： C07D498/04 ,  C07D498/14 ,  C07D471/14 ,  A61K31/551 ,  A61K31/553 ,  A61P15/00

CPC分类号： C07D471/14 ,  C07D487/14 ,  C07D498/04

摘要： This invention relates to compounds of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).

公开(公告)号：EP1917257A1

公开(公告)日：2008-05-07

申请号：EP06795254.9

申请日：2006-07-31

申请人： Pfizer Limited

发明人： BROWN, Alan, Daniel ,  CALABRESE, Andrew, Antony ,  ELLIS, David ,  SCIAMMETTA, Nunzio

IPC分类号： C07D401/14 ,  A61K31/497 ,  A61P15/12

CPC分类号： C07D401/14

摘要： The present invention relates to a class of substituted triazoles of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).

公开(公告)号：EP1863795A1

公开(公告)日：2007-12-12

申请号：EP06710566.8

申请日：2006-03-08

申请人： Pfizer Limited

发明人： CALABRESE, Andrew, Antony

IPC分类号： C07D401/14 ,  A61K31/497 ,  A61P5/10

CPC分类号： C07D401/14

摘要： The present invention relates to a class of substituted triazoles of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).

摘要翻译： 本发明涉及具有作为催产素拮抗剂活性的一类具有式（I）的取代三唑，其用途，其制备方法和含有所述抑制剂的组合物。 这些抑制剂可用于多种治疗领域，包括性功能障碍，特别是早泄（P.E.）。