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公开(公告)号：EP1786913B1
公开(公告)日：2011-08-17
申请号：EP05782434.4
申请日：2005-08-23
发明人： SALAGNAD, Christophe , ZOCHER, Frank , BURGARD, Andreas , JUNKER, Bernd , HOERLEIN, Rolf , STUEDEMANN, Thomas , MAIER, Claus-Jürgen , HACHTEL, Jochen , HOLLA, Wolfgang , TAPPERTZHOFEN, Christoph , KULITZSCHER, Berndt , MUTTI, Stéphane
IPC分类号： C12P7/62
CPC分类号： C07D413/12 , C07D263/62 , C07D309/12 , C12P17/14 , Y02P20/55
摘要： The invention relates to a method for producing diarylcycloalkyl derivatives of general formula (I), wherein the radicals have the indicated meanings. The invention further relates to novel intermediate products that are formed by means of the inventive method, methods for producing intermediate products of compounds of general formula (I), and a method for separating cis/trans isomer mixtures from starting materials used for the production of compounds of general formula (I).
摘要翻译： 本发明涉及用于生产通式（I）的二芳基环烷基衍生物的方法，其中基团具有所指出的含义。 本发明进一步涉及通过本发明方法形成的新颖中间产物，用于制备通式（I）化合物的中间产物的方法，以及从用于生产通式（I）化合物的原料中分离顺式/反式异构体混合物的方法 通式（I）的化合物。
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2.发明授权VERFAHREN ZUR HERSTELLUNG DER ENANTIOMEREN FORMEN VON CIS-3-HYDROXYCYCLOHEXANCARBONSÄURE-DERIVATEN UNTER VERWENDUNG VON HYDROLASEN 有权PROCESS FOR CIS-3羟基环己烷衍生物对映体形式制备使用HYDRO READ
公开(公告)号：EP1805316B1
公开(公告)日：2009-04-15
申请号：EP05778085.0
申请日：2005-07-23
CPC分类号： C12P41/004 , C12P7/00 , C12P17/00
摘要： The invention relates to a method for producing chiral, non-racemic, cis-configured cyclohexanols or cyclohexanol derivatives of formulae (la) and (Ib) wherein the radicals have the designations cited in the description, by means of enzymatic racemic splitting.
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3.发明授权VERFAHREN ZUR HERSTELLUNG VON OXAZOLEN DURCH KONDENSATION VON AROMATISCHEN ALDEHYDEN MIT ALFA-KETOXIMEN ZU N-OXIDEN UND NACHFOLGENDE REAKTION MIT AKTIVIERTEN SÄUREDERIVATEN 有权用于生产恶唑BY缩合ALFA-酮肟TO N氧化物和后续反应芳香醛与活性酸衍生物
公开(公告)号：EP1828149B1
公开(公告)日：2015-01-21
申请号：EP05817378.2
申请日：2005-12-01
发明人： HOLLA, Wolfgang , HOERLEIN, Rolf-Ludwig , KULITZSCHER, Berndt , LAUX, Wolfgang , STUEDEMANN, Thomas , TAPPERTZHOFEN, Christoph , SCHEFFER, Robert, J., H.
IPC分类号： C07D263/32 , A61K31/41 , A61P3/00
CPC分类号： C07D263/32
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公开(公告)号：EP1786913A2
公开(公告)日：2007-05-23
申请号：EP05782434.4
申请日：2005-08-23
发明人： SALAGNAD, Christophe , ZOCHER, Frank , BURGARD, Andreas , JUNKER, Bernd , HOERLEIN, Rolf , STUEDEMANN, Thomas , MAIER, Claus-Jürgen , HACHTEL, Jochen , HOLLA, Wolfgang , TAPPERTZHOFEN, Christoph , KULITZSCHER, Berndt , MUTTI, Stéphane
IPC分类号： C12P7/62
CPC分类号： C07D413/12 , C07D263/62 , C07D309/12 , C12P17/14 , Y02P20/55
摘要： The invention relates to a method for producing diarylcycloalkyl derivatives of general formula (I), wherein the radicals have the indicated meanings. The invention further relates to novel intermediate products that are formed by means of the inventive method, methods for producing intermediate products of compounds of general formula (I), and a method for separating cis/trans isomer mixtures from starting materials used for the production of compounds of general formula (I).
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5.发明公开VERFAHREN ZUR HERSTELLUNG VON OXAZOLEN DURCH KONDENSATION VON AROMATISCHEN ALDEHYDEN MIT ALFA-KETOXIMEN ZU N-OXIDEN UND NACHFOLGENDE REAKTION MIT AKTIVIERTEN SÄUREDERIVATEN 有权用于生产恶唑BY缩合ALFA-酮肟TO N氧化物和后续反应芳香醛与活性酸衍生物
公开(公告)号：EP1828149A1
公开(公告)日：2007-09-05
申请号：EP05817378.2
申请日：2005-12-01
发明人： HOLLA, Wolfgang , HOERLEIN, Rolf-Ludwig , KULITZSCHER, Berndt , LAUX, Wolfgang , STUEDEMANN, Thomas , TAPPERTZHOFEN, Christoph , SCHEFFER, Robert, J., H.
IPC分类号： C07D263/32 , A61K31/41 , A61P3/00
CPC分类号： C07D263/32
摘要： Disclosed is a method for producing oxazoles of formula IV by condensing aromatic aldehydes with a-ketoximes to N-oxides and then reacting the same with activated acid derivatives. The invention relates to a method for producing oxazoles by condensing aldehydes with a-ketoximes to N-oxides in the form of the salts thereof or as free bases and then reacting the same with activated acid derivatives so as to obtain oxazoles in the form of the salts thereof or as free bases.
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6.发明公开VERFAHREN ZUR HERSTELLUNG DER ENANTIOMEREN FORMEN VON CIS-KONFIGURIERTEN 3-HYDROXYCYCLOHEXANCARBONSÄURE-DERIVATEN UNTER VERWENDUNG VON HYDROLASEN 有权PROCESS FOR CIS-3羟基环己烷衍生物对映体形式制备使用HYDRO READ
公开(公告)号：EP1805316A2
公开(公告)日：2007-07-11
申请号：EP05778085.0
申请日：2005-07-23
CPC分类号： C12P41/004 , C12P7/00 , C12P17/00
摘要： The invention relates to a method for producing chiral, non-racemic, cis-configured cyclohexanols or cyclohexanol derivatives of formulae (la) and (Ib) wherein the radicals have the designations cited in the description, by means of enzymatic racemic splitting.
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