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    NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF
    5.
    发明公开
    NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF 审中-公开
    在NALROGENIERTE HETEROCYCLISCHE VERBINDUNG UND SALZ DAVON

    公开(公告)号：EP1900732A1

    公开(公告)日：2008-03-19

    申请号：EP06767173.5

    申请日：2006-06-22

    申请人： TOYAMA CHEMICAL CO., LTD. ,  TAISHO PHARMACEUTICAL CO., LTD

    发明人： KIYOTO, Taro ,  TANAKA, Tadashi ,  TSUTSUI, Yasuhiro ,  ANDO, Junichi ,  MOTONO, Mai ,  KAWAGUCHI, Yasuko ,  NOGUCHI, Toshiya ,  USHIKI, Yasunobu ,  USHIYAMA, Fumihito ,  URABE, Hiroki

    IPC分类号： C07D401/06 ,  A61K31/4709 ,  A61K31/496 ,  A61P31/04 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D491/056

    CPC分类号： C07D405/14 ,  C07D215/227 ,  C07D401/06 ,  C07D401/14 ,  C07D405/12 ,  C07D409/14 ,  C07D413/14 ,  C07D471/04 ,  C07D491/04 ,  C07D495/04 ,  C07D513/04 ,  C07D519/00

    摘要： A nitrogen-containing heterocyclic compound represented by the general formula: wherein the dashed line represents a single bond or a double bond; R 1 , R 2 , R 3 , R 4 and R 5 independently represent a hydrogen atom, halogen atom, a lower alkyl, aryl, lower alkoxy or monocyclic heterocyclic group which may be substituted or the like; R 6 represents a lower alkyl, aryl, monocyclic heterocyclic, bicyclic heterocyclic or tricyclic heterocyclic group which may be substituted; X 1 represents a lower alkylene group or the like; X 2 represents a lower alkylene, lower alkenylene or lower alkynylene group which may be substituted; X 3 represents an oxygen atom, sulfur atom, a sulfinyl group, sulfonyl group or the like; Y 1 represents a bivalent cyclic group, containing a nitrogen, which may be substituted or the like; and Z 1 represents a nitrogen atom, a carbon atom which may be substituted or the like, or a salt thereof. The compound or salt has a potent antibacterial activity and a high safety, and is therefore useful as an excellent antibacterial agent.

    摘要翻译： 一种由以下通式表示的含氮杂环化合物：其中虚线表示单键或双键; R 1，R 2，R 3，R 4和R 5独立地表示可以被取代的氢原子，卤素原子，低级烷基，芳基，低级烷氧基或单环杂环基等。 R 6表示可以被取代的低级烷基，芳基，单环杂环，双环杂环或三环杂环基; X 1表示低级亚烷基等; X 2表示可以被取代的低级亚烷基，低级亚烯基或低级亚烷基; X 3表示氧原子，硫原子，亚磺酰基，磺酰基等; Y 1表示可以被取代的氮的二价环状基团， Z 1表示氮原子，可被取代的碳原子等，或其盐。 该化合物或盐具有有效的抗菌活性和高安全性，因此可用作优异的抗菌剂。