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公开(公告)号：EP2084126A1
公开(公告)日：2009-08-05
申请号：EP07862379.0
申请日：2007-11-30
发明人： TSIPERMAN, Evgeny , GOROHOVSKY ROSENBERG, Sofia , YURKOVSKI, Slavik , FINE, Sergei , KOLTAI, Tamàs , ARONHIME, Judith
IPC分类号： C07C237/26
CPC分类号： C07C237/26
摘要： The present invention provides substantially pure intermediates, 9- haloacetomidominocyclines, and process of preparing them that are useful for the preparation of glycylcyclines, specifically Tigecycline.
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公开(公告)号：EP1919453A2
公开(公告)日：2008-05-14
申请号：EP06845942.9
申请日：2006-12-22
IPC分类号： A61K9/14 , A61K31/496
CPC分类号： A61K31/496 , A61K9/14
摘要： Micronized aripiprazole Form II having a particle shape and wherein 90% or more of the particles have a particle size of about 30 μm and the micronized aripiprazole Form II does not have more than 10% by weight of aripiprazole Type C as determined by X-ray diffraction and processes for making thereof.
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公开(公告)号：EP1633364B1
公开(公告)日：2008-02-27
申请号：EP05705020.5
申请日：2005-01-05
IPC分类号： A61K31/519 , A61P15/10 , C07D487/04
CPC分类号： A61K31/519 , C07D487/04
摘要： Provided are processes for the preparation of sildenafil base and the citrate salt sildenafil. Also provided are sildenafil citrate water adduct and a method of preparing pharmaceutical compositions comprising combining the sildenafil citrate and/or sildenafil citrate water adduct with at least one pharmaceutically-acceptable excipient.
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公开(公告)号：EP1863806A1
公开(公告)日：2007-12-12
申请号：EP06734993.6
申请日：2006-02-13
IPC分类号： C07D417/12 , A61K31/496 , A61P25/18
CPC分类号： C07D417/12
摘要： Provided is amorphous form of ziprasidone mesylate and process for its preparation. Also provided is a process for preparing ziprasidone mesylate dihydrate needle crystals.
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5.发明授权PHARMACEUTICAL COMPOSITION CONTAINING LAMOTRIGINE PARTICLES OF DEFINED MORPHOLOGY 有权药物组合物含拉莫三嗪颗粒具有确定形态
公开(公告)号：EP1496864B1
公开(公告)日：2007-03-21
申请号：EP03728552.5
申请日：2003-04-23
发明人： ARONHIME, Judith , SAMBURSKI, Guy
IPC分类号： A61K9/14
CPC分类号： A61K9/0019 , A61K9/0095 , A61K9/14 , A61K31/53
摘要： The present invention provides a pharmaceutical composition comprising a plurality of lamotrigine particles having a specific surface area of from about two to about three and a half meters per gram. Pharmaceutical compositions falling within the surface area criteria for the lamotrigine particles include those having a particle diameter equal to or less than about 100 µm, preferably about 50 µm, and most preferably 10 µm. The pharmaceutical composition can be formulated into a wide variety of dosage forms.
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公开(公告)号：EP1720876A1
公开(公告)日：2006-11-15
申请号：EP05723683.8
申请日：2005-02-25
发明人： WIZEL, Shlomit , ARONHIME, Judith , NIDDAM-HILDESHEIM, Valerie , DOLITZKY, Ben-Zion , ETINGER, Marina, Yu , YUZEFOVICH, Michael , NISNEVICH, Gennady, A. , PERTSIKOV, Boris , TISHIN, Boris , BLASBERGER, Dina
IPC分类号： C07D473/18 , A61K31/522 , A61P31/18
CPC分类号： A61K31/522 , C07D473/00 , C07D473/18
摘要： Provided are novel polymorphs and pseudopolymorphs of valacyclovir hydrochloride and pharmaceutical compositions containing these. Also provided are methods for making the novel polymorphs and pseudopolymorphs, which include valacyclovir hydrochloride monohydrate and valacyclovir hydrochloride dihydrate.
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公开(公告)号：EP1708708A1
公开(公告)日：2006-10-11
申请号：EP05712362.2
申请日：2005-01-31
IPC分类号： A61K31/47 , C07D215/18 , A61P11/06
CPC分类号： C07D215/18
摘要： The present invention relates to amorphous and polymorphic forms of montelukast free acid.
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公开(公告)号：EP1685099A1
公开(公告)日：2006-08-02
申请号：EP05810281.5
申请日：2005-07-01
IPC分类号： C07C401/00 , A61K31/592
CPC分类号： C07C401/00
摘要： Provided are novel crystalline forms of 1,24-(S)-dihydroxy vitamin D2, including hydrates and solvates, and methods for making them. Also provided are pharmaceutical and nutraceutical compositions containing the novel crystalline forms.
摘要翻译： 提供了1,24-（S） - 二羟基维生素D 2的新型结晶形式，包括水合物和溶剂化物，以及制备它们的方法。 还提供了含有新颖结晶形式的药物和营养组合物。
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公开(公告)号：EP1594493A2
公开(公告)日：2005-11-16
申请号：EP04814954.6
申请日：2004-12-16
IPC分类号： A61K31/404
CPC分类号： C07D209/14 , A61K31/404
摘要： Provided are polymorphic forms of tegaserod base and maleate, and processes for their preparation.
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公开(公告)号：EP1292304B1
公开(公告)日：2005-11-02
申请号：EP01930705.7
申请日：2001-04-24
发明人： ARONHIME, Judith , LEONOV, David , MESZAROS-SOS, Erzebet , SALYI, Szaboles , SZABO, Csaba , ZAVUROV, Shlomo
IPC分类号： A61K31/44 , C07D471/02 , A61P43/00 , C07D471/04
CPC分类号： C07D471/04 , A61K31/44
摘要： The present invention provides for novel polymorphs of zolpidem hemitartrate and the preparation of the polymorphs.
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