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公开(公告)号：EP0653207B1
公开(公告)日：1997-09-24
申请号：EP93900436.2
申请日：1992-12-25
发明人： KONDO, Shinichi , IKEDA, Yoko Crescent Ikejiri Ohashi 502, 19 -16 , HAMADA, Masa , TAKEUCHI, Tomio , HOSHINO, Hiroo
IPC分类号： A61K31/16
CPC分类号： A61K31/16
摘要： D-β-Lysylmethanediamine represented by formula (I) or a salt or hydrate thereof has an activity of inhibiting the infection with AIDS virus or HIV, and hence an AIDS virus infection inhibitor containing the same as an active ingredient is prospective as one of the remedies for AIDS which is thought to be difficult to cure.
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公开(公告)号：EP0653207A1
公开(公告)日：1995-05-17
申请号：EP93900436.2
申请日：1992-12-25
发明人： KONDO, Shinichi , IKEDA, Yoko Crescent Ikejiri Ohashi 502, 19 -16 , HAMADA, Masa , TAKEUCHI, Tomio , HOSHINO, Hiroo
IPC分类号： A61K31/16
CPC分类号： A61K31/16
摘要： D-β-Lysylmethanediamine represented by formula (I) or a salt or hydrate thereof has an activity of inhibiting the infection with AIDS virus or HIV, and hence an AIDS virus infection inhibitor containing the same as an active ingredient is prospective as one of the remedies for AIDS which is thought to be difficult to cure.
摘要翻译： 由式（I）表示的D-β-赖氨酰基甲二胺或其盐或水合物具有抑制艾滋病病毒或HIV感染的活性，因此含有其作为活性成分的AIDS病毒感染抑制剂有望作为 被认为难以治愈的艾滋病补救措施。
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3.发明公开D-B-LYSYLMETHANEDIAMINE DERIVATIVES WITH BACTERIA, AIDS VIRUS AND TUMOR CELL GROWTH INHIBITING ACTIVITY AND PREPARATION THEREOF 失效WITH INHIBITIERENDEN EFFECT D-B-lysylmethanediamine衍生物对细菌，艾滋病病毒和肿瘤细胞生长及生产
公开(公告)号：EP0777644A1
公开(公告)日：1997-06-11
申请号：EP95929220.0
申请日：1995-08-24
发明人： KONDO, Shinichi Royal Heights Minami-Rokugo 608 , IKEDA, Yoko Crescent Ikejiri Ohashi 502 , TAKEUCHI, Tomio New Fuji Mansion 701 , SHINEI, Rie , GOMI, Shuichi , SHIBAHARA, Seiji , HOSHINO, Hiroo
CPC分类号： C07C237/10
摘要： Now are provided (R)-3,6-diamino-N-(φ-aminoalkyl)-hexanamides which are novel compounds having general formula (I), wherein n stands for 2-5, and which may be for example, (R)-3,6-diamino-N-(2-aminoethyl)hexanamide (n = 2) and (R)-3,6-diamino-N-(3-aminopropyl)hexanamide (n = 3). Their preparation process is also provided. These novel compounds and acid addition salts thereof have activities inhibitory against Gram-positive bacteria, Gram-negative bacteria and AIDS virus, as well as tumor cells and are chemically stable. These novel compounds and their salts are useful as chemotherapeutic agents for diseases caused by these bacteria or virus and also as antitumor agent.
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