Acylaminopyridinecarboxamides, process for their preparation and their use as fungicides
    1.
    发明公开
    Acylaminopyridinecarboxamides, process for their preparation and their use as fungicides 失效
    酰基氨基吡啶甲酰胺,Verfahren zu ihrer Herstellung und ihre Verwendung als Fungizide。

    公开(公告)号:EP0473267A2

    公开(公告)日:1992-03-04

    申请号:EP91306444.0

    申请日:1991-07-16

    申请人: ZENECA LIMITED

    摘要: Fungicidal compounds of formula (I):

    in which A is fluoro, chloro, bromo, iodo, C₁₋₄ alkyl, C₁₋₄ alkoxy, halo(C₁₋₄)alkyl, C₁₋₄ alkoxylmethyl, C₁₋₄ alkylthiomethyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₁₋₄ alkoxycarbonyl, C₁₋₄ alkylcarbonyl, formyl, cyano, nitro or C₁₋₄ alkylthio; R¹ and R² are independently C₁₋₄ alkyl, C₃₋₆ alkenyl (optionally substituted with halogen), C₃₋₆ alkynyl (optionally substituted with halogen) C₁₋₄ alkoxy, halo(C₁₋₄)-alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalky(C₁₋₄)alkyl, C₁₋₄alkoxy(C₁₋₄)-alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano, or R¹ and R² together with the nitrogen to which they are atached join to form a morpholine, piperidine, pyrrolidine or azetidine ring, which may be optionally substitued with C₁₋₄ alkyl; R³ is H, or R³ and R⁴, together with the group C(0)N to which they are attached join to form an azetidin-2-one ring which is optionally substituted with C₁₋₄ alkyl; R⁴ is C₂₋₈ alkyl, C₂₋₈ alkenyl, C₂₋₈ alkynyl, or C₃₋₆ cycloalkyl, all of which may be optionally substituted with halogen, C₁₋₄ alkyl, C₁₋₄ alkoxy, C₁₋₄ alkylthio, cyano, C₁₋₄ alkylcarbonyl, C₁₋₄ alkoxycarbonyl, azido, nitro, isocyano or NR⁵R⁶ (where R⁵ and R⁶ are independently H, C₁₋₄ alkyl, C₁₋₄ alkylcarbonyl, or formyl); and X and Y are independently oxygen or sulphur.

    摘要翻译: 式(I)的杀真菌化合物:其中X和Y独立地为0或S,且A和R 1至R 4具有各种规定值。

    Acylaminopyridinecarboxamides, process for their preparation and their use as fungicides
    5.
    发明公开
    Acylaminopyridinecarboxamides, process for their preparation and their use as fungicides 失效
    ACYLAMINOPRIDINECARBOXAMIDES,其制备方法及其作为防腐剂的使用

    公开(公告)号:EP0473267A3

    公开(公告)日:1992-10-28

    申请号:EP91306444.0

    申请日:1991-07-16

    申请人: ZENECA LIMITED

    摘要: Fungicidal compounds of formula (I):

    in which A is fluoro, chloro, bromo, iodo, C₁₋₄ alkyl, C₁₋₄ alkoxy, halo(C₁₋₄)alkyl, C₁₋₄ alkoxylmethyl, C₁₋₄ alkylthiomethyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₁₋₄ alkoxycarbonyl, C₁₋₄ alkylcarbonyl, formyl, cyano, nitro or C₁₋₄ alkylthio; R¹ and R² are independently C₁₋₄ alkyl, C₃₋₆ alkenyl (optionally substituted with halogen), C₃₋₆ alkynyl (optionally substituted with halogen) C₁₋₄ alkoxy, halo(C₁₋₄)-alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalky(C₁₋₄)alkyl, C₁₋₄alkoxy(C₁₋₄)-alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano, or R¹ and R² together with the nitrogen to which they are atached join to form a morpholine, piperidine, pyrrolidine or azetidine ring, which may be optionally substitued with C₁₋₄ alkyl; R³ is H, or R³ and R⁴, together with the group C(0)N to which they are attached join to form an azetidin-2-one ring which is optionally substituted with C₁₋₄ alkyl; R⁴ is C₂₋₈ alkyl, C₂₋₈ alkenyl, C₂₋₈ alkynyl, or C₃₋₆ cycloalkyl, all of which may be optionally substituted with halogen, C₁₋₄ alkyl, C₁₋₄ alkoxy, C₁₋₄ alkylthio, cyano, C₁₋₄ alkylcarbonyl, C₁₋₄ alkoxycarbonyl, azido, nitro, isocyano or NR⁵R⁶ (where R⁵ and R⁶ are independently H, C₁₋₄ alkyl, C₁₋₄ alkylcarbonyl, or formyl); and X and Y are independently oxygen or sulphur.

    Fungicidal acylaminbezamides, their production and use
    8.
    发明公开
    Fungicidal acylaminbezamides, their production and use 失效
    杀真菌酰基氨基苯甲酰胺,它们的生产和使用

    公开(公告)号:EP0468682A1

    公开(公告)日:1992-01-29

    申请号:EP91306445.7

    申请日:1991-07-16

    申请人: ZENECA LIMITED

    摘要: Fungicidal compounds of formula (I):

    in which D and E are independently H or fluoro; X and Y are O or S; A, B, R³ and R⁴ have various specified values R¹ is C₂₋₄ alkenyl (optionally substituted with halogen), C₂₋₄ alkynyl (optionally substituted with halogen), halo(C₁₋₄)alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalkyl(C₁₋₄)alkyl, C₁₋₄ alkoxy(C₁₋₄)alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano; and R² is C₁₋₄ alkyl, C₁₋₄ alkoxy, C₂₋₄ alkenyl (optionally substituted with halogen), C₂₋₄ alkynyl (optionally substituted with halogen), halo(C₁₋₄) alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalkyl(C₁₋₄)alkyl, C₁₋₄alkoxy(C₁₋₄)alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano.

    摘要翻译: 式(I)的杀真菌化合物:其中D和E独立地为H或氟; X和Y是O或S; A,B,R 3和R 4具有各种规定值,R 1是C 2-4链烯基(任选被卤素取代),C 2-4炔基(任选被卤素取代),卤代(C 1-4)烷基,C 3-6环烷基, (C 1-4)烷基,C 1-4烷氧基(C 1-4)烷基,C 1-4烷硫基(C 1-4)烷基或氰基; 和R 2是C 1-4烷基,C 1-4烷氧基,C 2-4链烯基(任意被卤素取代),C 2-4炔基(任选被卤素取代),卤代(C 1-4)烷基,C 3-6环烷基, (C 1-4)烷基,C 1-4烷氧基(C 1-4)烷基,C 1-4烷硫基(C 1-4)烷基或氰基。