in which A is fluoro, chloro, bromo, iodo, C₁₋₄ alkyl, C₁₋₄ alkoxy, halo(C₁₋₄)alkyl, C₁₋₄ alkoxylmethyl, C₁₋₄ alkylthiomethyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₁₋₄ alkoxycarbonyl, C₁₋₄ alkylcarbonyl, formyl, cyano, nitro or C₁₋₄ alkylthio; R¹ and R² are independently C₁₋₄ alkyl, C₃₋₆ alkenyl (optionally substituted with halogen), C₃₋₆ alkynyl (optionally substituted with halogen) C₁₋₄ alkoxy, halo(C₁₋₄)-alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalky(C₁₋₄)alkyl, C₁₋₄alkoxy(C₁₋₄)-alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano, or R¹ and R² together with the nitrogen to which they are atached join to form a morpholine, piperidine, pyrrolidine or azetidine ring, which may be optionally substitued with C₁₋₄ alkyl; R³ is H, or R³ and R⁴, together with the group C(0)N to which they are attached join to form an azetidin-2-one ring which is optionally substituted with C₁₋₄ alkyl; R⁴ is C₂₋₈ alkyl, C₂₋₈ alkenyl, C₂₋₈ alkynyl, or C₃₋₆ cycloalkyl, all of which may be optionally substituted with halogen, C₁₋₄ alkyl, C₁₋₄ alkoxy, C₁₋₄ alkylthio, cyano, C₁₋₄ alkylcarbonyl, C₁₋₄ alkoxycarbonyl, azido, nitro, isocyano or NR⁵R⁶ (where R⁵ and R⁶ are independently H, C₁₋₄ alkyl, C₁₋₄ alkylcarbonyl, or formyl); and X and Y are independently oxygen or sulphur.
in which D and E are independently H or F; X and Y are 0 or S; R¹ to R⁴ have various specified values; A and B are independently H, iodo, nitro, cyano, C₁₋₄ alkoxycarbonyl, C₁₋₄ alkoxy(C₁₋₄)alkyl, C₁₋₄ alkylthio(C₁₋₄)-alkyl, formyl, C₁₋₄ alkylthio, halo(C₁₋₄)alkylthio, halo(C₁₋₄)alkoxy, C₁₋₄alkylcarbonyl, -CR⁵=NOR⁶ (where R⁵ and R⁶ are independently H or C₁₋₄ alkyl), C₂₋₄ alkenyl or C₂₋₄ alkynyl, provided that A and B are not both H.
摘要翻译:具有式(I)的杀真菌化合物:其中D和E独立地为H或F; X和Y为0或S; R 1至R 4具有各种指定值; A和B独立地是H,碘,硝基,氰基,C 1-4烷氧基羰基,C 1-4烷氧基(C 1-4)烷基,C 1-4烷硫基(C 1-4) - 烷基,甲酰基,C 1-4烷硫基,卤代( C 1-4)烷硫基,卤代(C 1-4)烷氧基,C 1-4烷基羰基,-CR 5 = NOR 6(其中R 5和R 6独立地为H或C 1-4烷基),C 2 -4-烯基或C 2-4炔基,条件是A和B不同时为H.
in which A is fluoro, chloro, bromo, iodo, C₁₋₄ alkyl, C₁₋₄ alkoxy, halo(C₁₋₄)alkyl, C₁₋₄ alkoxylmethyl, C₁₋₄ alkylthiomethyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₁₋₄ alkoxycarbonyl, C₁₋₄ alkylcarbonyl, formyl, cyano, nitro or C₁₋₄ alkylthio; R¹ and R² are independently C₁₋₄ alkyl, C₃₋₆ alkenyl (optionally substituted with halogen), C₃₋₆ alkynyl (optionally substituted with halogen) C₁₋₄ alkoxy, halo(C₁₋₄)-alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalky(C₁₋₄)alkyl, C₁₋₄alkoxy(C₁₋₄)-alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano, or R¹ and R² together with the nitrogen to which they are atached join to form a morpholine, piperidine, pyrrolidine or azetidine ring, which may be optionally substitued with C₁₋₄ alkyl; R³ is H, or R³ and R⁴, together with the group C(0)N to which they are attached join to form an azetidin-2-one ring which is optionally substituted with C₁₋₄ alkyl; R⁴ is C₂₋₈ alkyl, C₂₋₈ alkenyl, C₂₋₈ alkynyl, or C₃₋₆ cycloalkyl, all of which may be optionally substituted with halogen, C₁₋₄ alkyl, C₁₋₄ alkoxy, C₁₋₄ alkylthio, cyano, C₁₋₄ alkylcarbonyl, C₁₋₄ alkoxycarbonyl, azido, nitro, isocyano or NR⁵R⁶ (where R⁵ and R⁶ are independently H, C₁₋₄ alkyl, C₁₋₄ alkylcarbonyl, or formyl); and X and Y are independently oxygen or sulphur.
in which D and E are independently H or F; X and Y are O or S; A, B, R¹ and R² have various specified values; and R⁴ is substituted C₂₋₈ alkyl or optionally substituted cyclobutyl, cyclopentyl or cyclohexyl.
in which D and E are independently H or fluoro; X and Y are O or S; A, B, R³ and R⁴ have various specified values R¹ is C₂₋₄ alkenyl (optionally substituted with halogen), C₂₋₄ alkynyl (optionally substituted with halogen), halo(C₁₋₄)alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalkyl(C₁₋₄)alkyl, C₁₋₄ alkoxy(C₁₋₄)alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano; and R² is C₁₋₄ alkyl, C₁₋₄ alkoxy, C₂₋₄ alkenyl (optionally substituted with halogen), C₂₋₄ alkynyl (optionally substituted with halogen), halo(C₁₋₄) alkyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalkyl(C₁₋₄)alkyl, C₁₋₄alkoxy(C₁₋₄)alkyl, C₁₋₄ alkylthio(C₁₋₄)alkyl or cyano.