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公开(公告)号:US10167300B2
公开(公告)日:2019-01-01
申请号:US15914884
申请日:2018-03-07
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: A01N43/40 , A01N43/54 , A01N43/713 , A01N43/78 , A01N55/00 , A61K31/4439 , A61K31/444 , A61K31/506 , A61K31/695 , A61K45/06 , C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/06 , C07F7/08
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20180298038A1
公开(公告)日:2018-10-18
申请号:US15914884
申请日:2018-03-07
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07F7/08 , C07D405/14 , A01N55/00 , C07D409/14 , A01N43/78 , C07D417/06 , A01N43/40 , A01N43/54 , A61K31/506 , A61K31/444 , C07D401/14 , A01N43/713 , A61K31/4439 , C07D401/06 , A61K45/06 , A61K31/695
CPC classification number: C07F7/0812 , A01N43/40 , A01N43/54 , A01N43/713 , A01N43/78 , A01N55/00 , A61K31/4439 , A61K31/444 , A61K31/506 , A61K31/695 , A61K45/06 , C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/06
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US09944664B2
公开(公告)日:2018-04-17
申请号:US14683907
申请日:2015-04-10
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/06 , A61K45/06 , A61K31/444 , A61K31/506 , A61K31/695 , A01N43/54 , A01N43/78 , A01N43/713 , A01N47/02 , A01N55/00 , C07F7/08 , A61K31/4439 , A01N43/40
CPC classification number: C07F7/0812 , A01N43/40 , A01N43/54 , A01N43/713 , A01N43/78 , A01N55/00 , A61K31/4439 , A61K31/444 , A61K31/506 , A61K31/695 , A61K45/06 , C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/06
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20180290998A1
公开(公告)日:2018-10-11
申请号:US15945334
申请日:2018-04-04
Applicant: DOW AGROSCIENCES LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07D401/10 , A61K45/06 , A01N53/00 , C07D213/57 , C07D213/32 , A61K31/4406 , C07D213/30 , A01N47/02 , A61K31/506 , A61K31/505 , C07D239/26 , A01N43/54 , C07D239/34
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US09957252B2
公开(公告)日:2018-05-01
申请号:US15586657
申请日:2017-05-04
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07D401/10 , C07D239/26 , C07D213/30 , C07D213/32 , C07D213/57 , C07D239/34 , A61K31/505 , A01N47/02 , A01N43/54 , A61K31/4406 , A61K31/506
CPC classification number: C07D401/10 , A01N43/54 , A01N47/02 , A01N53/00 , A61K31/4406 , A61K31/505 , A61K31/506 , A61K45/06 , C07D213/30 , C07D213/32 , C07D213/57 , C07D239/26 , C07D239/34 , A61K2300/00
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20170233369A1
公开(公告)日:2017-08-17
申请号:US15586657
申请日:2017-05-04
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07D401/10 , C07D239/34 , C07D213/32 , C07D213/57 , C07D239/26 , C07D213/30
CPC classification number: C07D401/10 , A01N43/54 , A01N47/02 , A01N53/00 , A61K31/4406 , A61K31/505 , A61K31/506 , A61K45/06 , C07D213/30 , C07D213/32 , C07D213/57 , C07D239/26 , C07D239/34 , A61K2300/00
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US09663491B2
公开(公告)日:2017-05-30
申请号:US14683857
申请日:2015-04-10
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07D401/10 , A01N43/54 , C07D239/26 , A61K31/505 , A61K31/506 , A01N47/02 , C07D213/30 , A61K31/4406 , C07D213/32 , C07D213/57 , C07D239/34 , A61K45/06 , A01N53/00
CPC classification number: C07D401/10 , A01N43/54 , A01N47/02 , A01N53/00 , A61K31/4406 , A61K31/505 , A61K31/506 , A61K45/06 , C07D213/30 , C07D213/32 , C07D213/57 , C07D239/26 , C07D239/34 , A61K2300/00
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20150291632A1
公开(公告)日:2015-10-15
申请号:US14683907
申请日:2015-04-10
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07F7/08 , C07D401/06 , A61K31/4439 , A01N43/713 , C07D401/14 , A61K31/444 , A61K31/506 , A01N43/54 , A01N47/02 , A01N43/40 , C07D417/06 , A01N43/78 , C07D409/14 , A01N55/00 , A61K31/695 , C07D405/14 , A61K45/06
CPC classification number: C07F7/0812 , A01N43/40 , A01N43/54 , A01N43/713 , A01N43/78 , A01N55/00 , A61K31/4439 , A61K31/444 , A61K31/506 , A61K31/695 , A61K45/06 , C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/06
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20150291557A1
公开(公告)日:2015-10-15
申请号:US14683857
申请日:2015-04-10
Applicant: Dow AgroSciences LLC
Inventor: Michael R. Loso , Gary D. Gustafson , Asako Kubota , Maurice C. Yap , Zachary A. Buchan , Kimberly M. Steward , Michael T. Sullenberger , William J. Hoekstra , Christopher M. Yates
IPC: C07D401/10 , C07D239/26 , A61K31/505 , A61K31/506 , A01N47/02 , A61K45/06 , C07D213/30 , A61K31/4406 , C07D213/32 , C07D213/57 , C07D239/34 , A01N43/54 , A01N43/40
CPC classification number: C07D401/10 , A01N43/54 , A01N47/02 , A01N53/00 , A61K31/4406 , A61K31/505 , A61K31/506 , A61K45/06 , C07D213/30 , C07D213/32 , C07D213/57 , C07D239/26 , C07D239/34 , A61K2300/00
Abstract: The instant invention describes compounds of Formula I having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
Abstract translation: 本发明描述了具有金属酶调节活性的式I化合物,以及治疗由这些金属酶介导的疾病,病症或症状的方法。
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