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    Acylamino-cephalosporanic acids
    1.
    发明授权
    Acylamino-cephalosporanic acids 失效
    酰氨基 - 头孢菌酸

    公开(公告)号：US3865820A

    公开(公告)日：1975-02-11

    申请号：US24428772

    申请日：1972-04-14

    Applicant: HOECHST AG

    Inventor： SCHORR MANFRED ,  SCHRINNER ELMAR

    IPC: A61K20060101 ,  A61K31/43 ,  C07D20060101 ,  C07D499/12 ,  C07D499/34 ,  C07D499/48 ,  C07D501/06 ,  C07D501/26 ,  C07D501/32 ,  C07D501/60 ,  C07D99/24

    CPC classification number: C07D499/00

    Abstract: Acylaminocephalosporanic acids of the formula I

    wherein R1, R2 and R3 each represents hydrogen or lower alkyl radicals in which case R1 and R2 may also form together an optionally substituted alkylene radical, A represents an optionally substituted phenylene or thienyl radical, and X represents an oxygen atom or a single bond, the physiologically tolerable salts thereof, pharmaceutical preparations effective against bacterial infections containing these compounds, and a process for the manufacture.

    Abstract translation: 式I的酰氨基头孢烷酸其中R 1，R 2和R 3各自表示氢或低级烷基，其中R 1和R 2也可以一起形成任选取代的亚烷基，A表示任选取代的亚苯基或噻吩基，X表示氧 原子或单键，其生理上可耐受的盐，对含有这些化合物的细菌感染有效的药物制剂及其制备方法。

    Phenyldithiocarbamic acid benzimidazolyl-(2)-methyl esters
    2.
    发明授权
    Phenyldithiocarbamic acid benzimidazolyl-(2)-methyl esters 失效
    （2）-METHYL ESTERS（苯甲酰胺）

    公开(公告)号：US3658834A

    公开(公告)日：1972-04-25

    申请号：US3658834D

    申请日：1969-11-21

    Applicant: HOECHST AG

    Inventor： SCHORR MANFRED ,  DURCKHEIMER WALTER ,  DUWEL DIETER

    IPC: C07D235/06 ,  C07D49/38

    CPC classification number: C07D235/06

    Abstract: DITHIOCARBAMIC ACID ESTERS OF THE FORMULA

    1-R3,2-((R4,R5-PHENYL)-NH-C(=S)-S-CH2-),R1,R2-

    BENZIMIDAZOLE

    IN WHICH R1 IS HYDROGEN, CHLORINE, BROMINE, TRIFLUOROMETHYL, NITRO OR CYANO, R2 IS HYDROGEN, CHLORINE, BROMINE, TRIFLUOROMETHYL OR NITRO, R3 IS HYRDROGEN OR ALKYL HAVING 1 TO 6 CARBON ATOMS, AND R4 AND R5 EACH IS HYDROGEN, CHLORINE, BROMINE, IODINE, TRIFLUOROMETHYL OR ALKYL HAVING 1 TO 6 CARBON ATOMS, WHICH COMPOUNDS ARE ACTIVE AGAINST HELMINTHIC DISEASES, AND A PROCESS FOR PREPARING THEM.

    Substituted p-hydroxyphenyl-hydrazones and process for their manufacture
    3.
    发明授权
    Substituted p-hydroxyphenyl-hydrazones and process for their manufacture 失效
    取代的对羟基苯酚和水解产物及其制备方法

    公开(公告)号：US3573287A

    公开(公告)日：1971-03-30

    申请号：US3573287D

    申请日：1968-08-07

    Applicant: HOECHST AG

    Inventor： SCHORR MANFRED ,  SCHRINNER ELMAR ,  TEICHMANN KARL HORST

    IPC: A61K31/44 ,  C09B26/04 ,  C07D31/42

    CPC classification number: A61K31/44 ,  C09B26/04

    Abstract: SUBSTITUTED P-HYDROXYPHENYL-HYDRAZONES OF THE FORMULA

    1-R4,3-((4-(HO-),R1,R2-PHENYL)-NH-N=C(-R3)-)PYRIDINIUM

    X(-)

    IN WHICH R1 AND R2 REPRESENT HYDROGEN, HALOGEN, LOWER ALKYL OR ALKOXY, CARBOXY, CARBAMOYL, LOWER CARBALKOXY, CARBOBENZOXY, SULFOXY OR SULFAMOUL; R3 REPRESNETS HYDROGEN OR LOWER ALKYL HAVING 1 TO 3 CARBON ATOMS, R4 REPRESENTS AN ALKYL RADICAL HAVING 1 TO 12 CARBON ATOMS, WHICH MAY CARRY ONE OR SEVERAL HYDROXY, LOWER ALKOXY, CARBOXY, LOWER CARBALKOXY, CARBAMOYL, NITRILE, SULFO, LOWER SULFALKOXY AND/OR SULFAMOYL GROUPS, AND X REPRESENTS THE ANION OF A NON-TOXIC ACID, WHICH COMPOUNDS HAVE BACTERIOSTATIC PROPERTIES.

    Acylamino-cephem-carboxylic acids and process for preparing them
    4.
    发明授权
    Acylamino-cephem-carboxylic acids and process for preparing them 失效
    酰氨基 - 头孢烯羧酸及其制备方法

    公开(公告)号：US3920640A

    公开(公告)日：1975-11-18

    申请号：US35646673

    申请日：1973-05-02

    Applicant: HOECHST AG

    Inventor： SCHORR MANFRED ,  WORM MANFRED ,  SCHRINNER ELMAR

    IPC: C07D233/22 ,  C07D233/26 ,  C07D239/06 ,  C07D333/38 ,  C07D501/20 ,  C07D501/22 ,  C07D501/24

    CPC classification number: C07D239/06 ,  C07D233/22 ,  C07D233/26 ,  C07D333/38

    Abstract: IN WHICH R1, R2 and R3 represent hydrogen or lower alkyl groups and R1 and R2 may form together an alkylene group which may be substituted, R4 represents a linear or branched alkyl radical of 1 to 5 carbon atoms, a cyclo-alkyl radical of 3 to 7 carbon atoms which may be interrupted by heteroatoms, X represents a single bond or NH, A represents a phenylene or thienylene group which may be substituted and Y represents a single bond or oxygen, and their physiologically tolerated salts; the novel compounds have very good anti-bacterial properties.

    Acylamino-cephem-carboxylic acids of the general formula

    Abstract translation: 酰基氨基 - 头孢烯羧酸，其通式为R 1，R 2和R 3表示氢或低级烷基，R 1和R 2可以一起形成可被取代的亚烷基，R 4表示1至5的直链或支链烷基 碳原子，可被杂原子中断的3-7个碳原子的环烷基，X表示单键或NH，A表示可被取代的亚苯基或亚噻吩基，Y表示单键或氧，以及 他们的生理耐受盐; 新型化合物具有非常好的抗菌性能。

    Thiophene-3-isonitriles
    6.
    发明授权
    Thiophene-3-isonitriles 失效
    三硝基-3-间苯二酚

    公开(公告)号：US3687977A

    公开(公告)日：1972-08-29

    申请号：US3687977D

    申请日：1969-09-05

    Applicant: HOECHST AG

    Inventor： RIPPEL ROBERT ,  DITTMAR WALTER ,  SCHORR MANFRED

    IPC: C07D333/36 ,  C07D333/38 ,  A61K27/00 ,  C07D63/16

    CPC classification number: C07D333/36 ,  C07D333/38

    Abstract: Thiophene-3-isonitriles of the formula IN WHICH R1 is hydrogen, alkyl, carbalkoxy, cyano or phenyl, R2 is hydrogen, alkyl, alkoxy, carbalkoxy, cyano or phenyl, R3 is hydrogen, alkyl, carbalkoxy or phenyl, or R2 and R3 together represent an alkylene chain, are disclosed as having antimycotic and antibacterial properties.

    Abstract translation: 噻吩-3-异腈，其中R1是氢，烷基，烷氧基，氰基或苯基，R2是氢，烷基，烷氧基，烷氧基，氰基或苯基，R3是氢，烷基，烷氧基或苯基，或R2和R3 一起表示亚烷基链，被公开为具有抗真菌性和抗菌性。

    1 4-phenylene-bis-dithiocarbamic acid esters
    7.
    发明授权
    1 4-phenylene-bis-dithiocarbamic acid esters 失效
    1 4-苯基双 - 二硫代酸酯

    公开(公告)号：US3660422A

    公开(公告)日：1972-05-02

    申请号：US3660422D

    申请日：1969-07-11

    Applicant: HOECHST AG

    Inventor： SCHORR MANFRED ,  DURCKHEIMER WALTER ,  DUWEL DIETER

    IPC: C07D235/24 ,  C07C333/24 ,  C07D235/06 ,  C07D49/38

    CPC classification number: C07D235/06 ,  Y10S514/893

    Abstract: WHEREIN X IS CHLORINE, BROMINE, OR IODINE.

    R3-CH(-X)-R4

    WHEREIN R1 AND R2 ARE HYDROGEN, HALOGEN, ALKYL HAVING 1-6 CARBON ATOMS, OR ALKOXY HAVING 1-6 CARBON ATOMS, R3 IS HYDROGEN OR ALKYL HAVING 1-6 CARBON ATOMS, AND R4 IS 2-BENZIMIDAZOLE OR 2-BENZAMIDAZOLE SUBSTITUTED WITH ONE OR MORE HALOGEN, LOWER ALKYL, TRIFLUOROMETHYL, LOWER ALKOXY, NITRO, SULFAMIDO, OR NITRILO GROUPS. THE ESTERS, WHICH ARE ACTIVE AGAINST LIVER FLUKES FOR EXAMPLE, ARE PREPARED BY REACTING A SALT OF A CORRESPONDING BIS-DITHIOCARBAMIC ACID WITH A COMPOUND OF THE FORMULA
    ANTHELMINTICALLY-ACTIVE BIS-DITHIOCARBAMIC ESTERS OF THE FORMULA

    1-R1,2,5-BIS(R3-CH(-R4)-S-C(=S)-NH-),4-R2-BENZENE

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