N-cycloalkyl-3-alkenybenzoyl-pyrazole derivatives
    1.
    发明授权
    N-cycloalkyl-3-alkenybenzoyl-pyrazole derivatives 失效
    N-环烷基-3-烯基苯甲酰基 - 吡唑衍生物

    公开(公告)号:US06475957B1

    公开(公告)日:2002-11-05

    申请号:US10019047

    申请日:2001-12-27

    IPC分类号: A01N4356

    CPC分类号: A01N43/56 C07D231/20

    摘要: Cycloalkyl-substituted benzoylpyrazoles of the formula I where the variables have, for example, the following meanings: R1 is hydrogen, nitro, halogen, cyano, thiocyanato, or an unsubstituted or substituted aliphatic radical; R2 is an unsubstituted or substituted aliphatic radical, halogen, nitro, or substituted sulfonyl or amino groups, R3 is hydrogen, halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl or C2-C6-alkynyl; R4, R5 are hydrogen, nitro, halogen, cyano, thiocyanato, an unsubstituted or substituted aliphatic radical or substituted sulfonyl or amino groups; R6 is hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkyl; R7 is a cyclic ring system having 3-14 ring atoms; R16 is hydroxyl or a substituted hydroxyl group; and their tautomers or agriculturally useful salts are described. Moreover, the invention describes processes for preparing compounds of the formula I, compositions comprising them, and the use of the compounds of the formula I and of the compositions comprising them for controlling harmful plants.

    摘要翻译: 式I的环烷基取代的苯甲酰基吡唑,其中变量具有例如以下含义:R 1是氢,硝基,卤素,氰基,氰硫基或未取代或取代的脂族基; R 2是未取代或取代的脂族基,卤素, 硝基或取代的磺酰基或氨基,R 3是氢,卤素,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 6 - 烷氧基,C 2 -C 6 - 烯基或C 2 -C 6 - 炔基; R 4,R 5是氢 硝基,卤素,氰基,氰硫基,未取代或取代的脂族基团或取代的磺酰基或氨基; R 6是氢,卤素,C 1 -C 6烷基,C 1 -C 6 - 烷氧基,C 3 -C 8环烷基; 具有3-14个环原子的环系; R 16是羟基或取代的羟基;并且描述了它们的互变异构体或农业上有用的盐。此外,本发明描述了制备式I化合物的方法,包含它们的组合物,以及使用 式I化合物和组合物的化合物 包括它们用于控制有害植物。

    Thiochromanoylpyrazolone derivatives
    5.
    发明授权
    Thiochromanoylpyrazolone derivatives 失效
    硫代色酰基吡唑啉酮衍生物

    公开(公告)号:US06352959B1

    公开(公告)日:2002-03-05

    申请号:US09857053

    申请日:2001-05-31

    IPC分类号: A01N4384

    CPC分类号: C07D409/06 C07D409/14

    摘要: Thiochromanoylpyrazolone derivatives of the formula I where: A is an unsubstituted or substituted, saturated or unsaturated alkyl chain; R1 is cyano, thiocyanato, nitro, OR4, SR5, SOR6, S02R6, ONR6NR7, ON═CR6R8, NR9R10, P(O)R11R12, P(S)R11R12, COR, CO2R6, unsubstituted or substituted phenyl or heterocyclyl; R2 is alkyl, haloalkyl, alkoxy or haloalkoxy; R3 is hydrogen, alkyl or halogen; X is oxygen, sulfur, S═O, S(═O)2, CR13R14, C═O or C═NR15; m is 0, 1 or 2; n is 0, 1, 2, 3 or 4; R16 is substituted pyrazol-4-yl-carbonyl or substituted (4,5-dihydro-5-oxo-pyrazol-4-yl)methylidene; and their agriculturally useful salts; Processes for preparing the thiochromanoylpyrazolone derivatives, compositions comprising them, and the use of these derivatives or of the compositions comprising them for controlling undesirable plants are described.

    摘要翻译: 其中:A为未取代或取代的饱和或不饱和烷基链; R1为氰基,氰硫基,硝基,OR4,SR5,SOR6,SO2R6,ONR6NR7,ON = CR6R8,NR9R10,P(O)R11R12, P(S)R 11 R 12,COR,CO 2 R 6,未取代或取代的苯基或杂环基; R 2是烷基,卤代烷基,烷氧基或卤代烷氧基; R 3是氢,烷基或卤素; X是氧,硫,S = O,S(= O) 2,CR 13 R 14,C = O或C = NR 15; m为0,1或2; n为0,1,2,3或4; R 16为取代的吡唑-4-基 - 羰基或取代的(4,5-二氢 描述了制备硫代色满酰基吡唑啉酮衍生物的方法,包含它们的组合物,以及这些衍生物或包含它们的组合物用于防治不期望的植物的用途。

    3-(heterocyclyl)-substituted benzolpyrazols
    6.
    发明授权
    3-(heterocyclyl)-substituted benzolpyrazols 失效
    3-(杂环基)取代的苯并吡唑

    公开(公告)号:US06831039B1

    公开(公告)日:2004-12-14

    申请号:US09857067

    申请日:2001-05-21

    IPC分类号: A01N4356

    CPC分类号: C07D413/10 C07D231/20

    摘要: The invention relates to 3-(heterocyclyl)-substituted benzoylpyrazois of formula (I), wherein the variables have the following meanings: X is O, NH or N-alkyl; R1 is alkyl; R2, R3, R4, R5 are hydrogen, alkyl or alkyl halide; R6 is halogen, nitro, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfonyl or halogenalkylsulfonyl; R7 is hydroxy, alkoxy, alkenyloxy, alkylsulfonyloxy, alkylcarboyloxy, alkylthiocarbonyloxy, phenylsulfonyloxy or phenylcarbonyloxy, and the phenyl radical can be substituted; R8, R9 are alkyl; R10 is hydrogen or alkyl; and R11 is hydrogen or alkyl; and to their agriculturally useable salts. The invention also relates to intermediate products and methods for producing the inventive compounds and to the use of these compounds or products containing them for combating undesirable plants.

    摘要翻译: 本发明涉及式(I)的3-(杂环基)取代的苯甲酰基吡啶,其中变量具有以下含义:X是O,NH或N-烷基; R 1是烷基; R 2,R 3,R 4,R 5是氢,烷基或烷基卤; R 6是卤素,硝基,烷基卤,烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,烷基磺酰基或卤代烷基磺酰基; R 7是羟基,烷氧基,烯氧基,烷基磺酰氧基,烷基羰氧基,烷硫基羰基氧基,苯基磺酰氧基或苯基羰基氧基,苯基可以被取代; R 8,R 9是烷基; R 10是氢或烷基; 和R 11是氢或烷基; 以及其农业上可用的盐类。 本发明还涉及用于生产本发明化合物的中间产物和方法以及含有它们的这些化合物或产品用于对抗不期望的植物的用途。

    TRICYCLIC BENZOYLPYRAZOLE DERIVATIVES
    10.
    发明申请
    TRICYCLIC BENZOYLPYRAZOLE DERIVATIVES 审中-公开
    三苯甲酰基吡唑衍生物

    公开(公告)号:US20070197393A1

    公开(公告)日:2007-08-23

    申请号:US11461491

    申请日:2006-08-01

    摘要: Tricyclic benzoylpyrazole derivatives of the formula I where: X is oxygen, sulfur, S═O, S(═O)2, CR6R7, NR8 or a bond; Y together with the two carbons to which it is attached forms a saturated, partially saturated or unsaturated 5- or 6-membered heterocycle; R1, R2, R6, R7 are hydrogen, alkyl, haloalkyl, alkoxy or haloalkoxy; R3 is halogen, alkyl, haloalkyl, alkoxy or haloalkoxy; R4 is hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, unsubstituted or substituted aminosulfonyl or unsubstituted or substituted sulfonylamino; R5 is hydrogen, alkyl or halogen; l is 0, 1 or 2; R8 is hydrogen, alkyl, haloalkyl, alkylcarbonyl, formyl, alkoxycarbonyl, haloalkoxycarbonyl, alkylsulfonyl or haloalkylsulfonyl; R9 is substituted pyrazol-4-ylcarbonyl or substituted 5-oxopyrazolin-4-ylmethylidene; and their agriculturally useful salts; processes and intermediates for preparing the tricyclic benzoylpyrazole derivatives; compositions comprising them and the use of these derivatives or of the compositions comprising them for controlling undesirable plants are described.

    摘要翻译: 式I的三环苯甲酰基吡唑衍生物其中:X是氧,硫,SO,S(-O)2,CR 6,R 7, NR 8或键; Y与连接的两个碳一起形成饱和的,部分饱和的或不饱和的5-或6-元杂环; R 1,R 2,R 6,R 7是氢,烷​​基,卤代烷基,烷氧基或卤代烷氧基; R 3是卤素,烷基,卤代烷基,烷氧基或卤代烷氧基; R 4是氢,硝基,卤素,氰基,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,烷基亚磺酰基,卤代烷基亚磺酰基,烷基磺酰基,卤代烷基磺酰基,未取代或取代的氨基磺酰基或未取代或取代的磺酰基氨基; R 5是氢,烷基或卤素; l为0,1或2; R 8是氢,烷基,卤代烷基,烷基羰基,甲酰基,烷氧基羰基,卤代烷氧基羰基,烷基磺酰基或卤代烷基磺酰基; R 9是取代的吡唑-4-基羰基或取代的5-氧代吡唑啉-4-基亚甲基; 及其农业用盐; 制备三环苯甲酰基吡唑衍生物的方法和中间体; 描述了包含它们的组合物以及这些衍生物或包含它们的组合物用于防治不期望的植物的用途。