Pesticidal 1-aryl-5-(substituted alkylideneimino)pyrazoles
    18.
    发明授权
    Pesticidal 1-aryl-5-(substituted alkylideneimino)pyrazoles 失效
    杀虫剂1-芳基-5-(取代的亚烷基亚氨基)吡唑

    公开(公告)号:US5360910A

    公开(公告)日:1994-11-01

    申请号:US842431

    申请日:1992-03-04

    摘要: The invention describes novel 1-aryl-5-(substituted alkylideneimino)pyrazoles of formula (I) ##STR1## wherein typically preferred substituents are: R.sup.1 is cyano, nitro, or halogen;R.sup.2 is R.sup.9 S(O).sub.n in which n is 0, 1 or 2 and R.sup.9 is alkyl, preferably methyl which is substituted by halogen atoms which are the same or different up to full substitution of the alkyl moiety;R.sup.3 is hydrogen or alkyl;R.sup.4 is phenyl or heteroaryl, optionally substituted by one or more hydroxy, halogen, alkoxy, alkylthio, cyano or alkyl or combinations thereof; preferably R.sup.4 is phenyl, which is at least substituted by 3-hydroxy or 4-hydroxy;R.sup.5 is hydrogen, alkyl or halogen;R.sup.6 and R.sup.8 are hydrogen;R.sup.7 is halogen, alkyl, haloalkyl or haloalkoxy; andX is a nitrogen atom or CR.sup.14 in which R.sup.14 is hydrogen, halogen, cyano, alkyl, alkylthio or alkoxy.The invention further describes processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (mites, aphids or insects), nematodes, helminths, or protozoa.

    摘要翻译: 本发明描述了式(I)的新型1-芳基-5-(取代的亚烷基亚氨基)吡唑其中通常优选的取代基是:R 1是氰基,硝基或卤素; R2是R9S(O)n,其中n是0,1或2,R9是烷基,优选被烷基部分完全取代的相同或不同的卤素原子取代的甲基; R3是氢或烷基; R4是任选被一个或多个羟基,卤素,烷氧基,烷硫基,氰基或烷基或其组合取代的苯基或杂芳基; 优选R4是至少被3-羟基或4-羟基取代的苯基; R5是氢,烷基或卤素; R6和R8是氢; R7是卤素,烷基,卤代烷基或卤代烷氧基; X为氮原子或CR 14,其中R 14为氢,卤素,氰基,烷基,烷硫基或烷氧基。 本发明还描述了使化合物,化合物的组合物和化合物用于控制节肢动物(螨虫,蚜虫或昆虫),线虫,蠕虫或原生动物的方法。