公开(公告)号：US3887556A

公开(公告)日：1975-06-03

申请号：US31042372

申请日：1972-11-29

Applicant: BAYER AG

Inventor： DRABER WILFRIED ,  BUCHEL KARL HEINZ ,  REGEL ERIK ,  PLEMPEL MANFRED

IPC: A61K31/495 ,  A61K31/505 ,  C07D241/12 ,  C07D403/06 ,  C07D51/36

CPC classification number: C07D403/06 ,  A61K31/495 ,  A61K31/505 ,  C07D241/12

Abstract: N-methyl-imidazole derivatives of the formula:

OR A PHARMACEUTICALLY ACCEPTABLE NON-TOXIC SALT THEREOF, WHEREIN X is an unsubstituted or substituted six-membered heteroaromatic moiety having two nitro heteroatoms, Y is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety or an unsubstituted or substituted aryl moiety, and Z is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety, an unsubstituted or substituted aryl moiety, an unsubstituted or substituted pyridyl moiety or an alkoxycarbonyl moiety, ARE USEFUL AS ANTIMYCOTIC AGENTS.

Abstract translation: 下式的N-甲基 - 咪唑衍生物：

公开(公告)号：US3689664A

公开(公告)日：1972-09-05

申请号：US3689664D

申请日：1971-04-06

Applicant: BAYER AG

Inventor： BUCHEL KARL HEINZ ,  DRABER WILFRIED ,  HAMMANN INGEBORG

IPC: A01N47/08 ,  A01N47/24 ,  A01N9/14 ,  A01N9/20

CPC classification number: A01N47/08 ,  A01N47/24

Abstract: N-carbonic acid derivatives of 1,2-dicarbonylphenylhydrazones, i.e. N-((alkoxy, phenoxy, alkylmercapto, cyclohexyloxy and dialkylamino- -carbonyl and -thiono)-N-(alkyl- and/or electronegative substituent (e.g. halo, haloalkyl, nitro and/or alkyl sulfonyl)- -substituted phenyl)-N''-( Alpha -cyano- Alpha (alkanoyl and carboalkoxyl)-carbonyl)-hydrazones, which possess arthropodicidal, especially acaricidal and insecticidal, properties and which may be produced by reacting the corresponding alkali metal salt of a 1,2dicarbonylphenylhydrozone, or such 1,2-dicarbonylphenylhydrozone in the presence of an acid-binding agent, with the corresponding carbonic acid chloride.

Abstract translation: N-（（烷氧基，苯氧基，烷基巯基，环己氧基和二烷基氨基 - 羰基和 - 硫杂）-N-（烷基 - 和/或电 - 负 - 取代基[例如卤素， 卤代烷基，硝基和/或烷基磺酰基] - 取代的苯基）-N' - （α-氰基-α-[烷酰基和烷氧羰基] - 羰基） - 腙，其具有杀虫，特别是杀螨和杀虫的性质， 通过使相应的1,2-二羰基苯基氢区的碱金属盐或这样的1,2-二羰基苯基氢区在酸结合剂的存在下与相应的碳酰氯反应而制备。

公开(公告)号：US3636112A

公开(公告)日：1972-01-18

申请号：US3636112D

申请日：1969-07-02

Applicant: BAYER AG

Inventor： DRABER WILFRIED ,  BUCHEL KARL HEINZ ,  HAMMANN INGEBORG ,  UNTERSTENHOFER GUNTER

IPC: A01N20060101 ,  C07C20060101 ,  C07C251/74 ,  C07C119/00

CPC classification number: C07C251/74

Abstract: A-HALO - A - FORMLY-CARBONYL-PHENYL-HYDRAZONES, I.E. A-(CHLORO AND BROMO)-A-(FORMYL, DIOXA-PENTAMETHYLENE AND OXA-THIA-PENTAMETHYLENE)-CARBONYL - (MONO TO TRI ALKYL, CHLORO, TRIFLUOROMETHYL, TRIFLUOROMETHYL MERCAPTO AND/OR ALKYL SULFONYL-SUBSTITUTED PHENYL)-HYDRAZONES, WHICH POSSESS ARTHROPOLICIDAL, ESPECIALLY ACARICIDAL AND INSECTICIDAL, PROPERTIES, AND WHICH MAY BE PRODUCED BY CONVENTIONAL METHODS.