Oxime derivatives, hydrazone derivatives and use thereof
    4.
    发明授权
    Oxime derivatives, hydrazone derivatives and use thereof 失效
    肟衍生物,腙衍生物及其用途

    公开(公告)号:US06251949B1

    公开(公告)日:2001-06-26

    申请号:US09457672

    申请日:1999-12-09

    IPC分类号: A61K3115

    摘要: Compounds having fungicidal activities and represented by general formula (I) and salts and hydrates thereof wherein R1 represents an optionally substituted aryl, an optionally substituted alkyl or the like; R2 represents an optionally substituted alkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted aryl, an optionally substituted heterocyclic group or the like; R3 represents an optionally substituted alkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted arylsulfonyl, an optionally substituted heterocyclic group or the like; R4 and R5, which may be the same or different, represent each a hydrogen atom, an optionally substituted alkyl, or an optionally substituted alkoxy, or R4 and R5 may form together with the adjacent nitrogen atom an optionally substituted monocycle or polycycle; X and Y, which may be the same or different, represents each an oxygen atom or NR6 wherein R6 represents a hydrogen atom, an optionally substituted alkyl, an optionally substituted aryl, an optionally substituted alkanoyl, or an optionally substituted aroyl; Z represents an oxygen atom or a sulfur atom; and a wavy line (˜) represents the configuration of an E isomer, a Z isomer, or a mixture thereof.

    摘要翻译: 具有杀真菌活性并由通式(I)表示的化合物及其盐和水合物,其中R 1表示任选取代的芳基,任选取代的烷基等; R 2表示任选取代的烷基,任选取代的烯基,任选取代的炔基,任选取代的芳基,任选取代的杂环基等; R 3表示任选取代的烷基,任选取代的烯基,任选取代的炔基,任选取代的芳基磺酰基,任选取代的杂环基团等; R 4和R 5可以相同或不同,表示氢原子,任选取代的烷基或任选取代的烷氧基,或者R 4和R 5可以与相邻的氮原子一起形成任选取代的单环或多环; X和Y可以相同或不同,表示每个氧原子或NR 6,其中R 6表示氢原子,任选取代的烷基,任选取代的芳基,任选取代的烷酰基或任选取代的芳酰基; Z表示氧原子或硫原子; 波浪线(〜)表示E异构体,Z异构体或其混合物的构型。