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    4-Amino-1,2,4-triazine-5-one novel compounds, a process for their production and herbicidal compositions
    1.
    发明授权
    4-Amino-1,2,4-triazine-5-one novel compounds, a process for their production and herbicidal compositions 失效
    4-氨基-1,2,4-三嗪-5-酮新化合物，其生产方法和除草组合物

    公开(公告)号：US3907543A

    公开(公告)日：1975-09-23

    申请号：US41066873

    申请日：1973-10-29

    Applicant: BAYER AG

    Inventor： DICKORE KARLFRIED ,  DRABER WILFRIED ,  EUE LUDWIG

    IPC: A01N43/707 ,  C07D253/07 ,  A01N9/22

    CPC classification number: A01N43/707 ,  C07D253/07

    Abstract: Certain novel 4-amino-1,2,4-triazine-5-one compounds of the formula:

    in which R1 and R4 are hydrogen, alkyl, cycloalkyl, substituted phenyl or phenyl; R2 is hydrogen or alkyl; R3 is hydrogen, alkyl, phenyl, haloalkyl, phenylalkyl, or alkylphenyl, alkoxyphenyl or alkylmercaptophenyl; ARE PREPARED BY A NOVEL PROCESS COMPRISING REACTING A GLYOXYLIC ACID ESTER 2-ACYLHYDRAZONE OF THE FORMULA
    in which R1 and R4 are defined as above, and R is alkyl of from 1 to 4 carbon atoms, IS REACTED WITH A HYDRAZINE DERIVATIVE OF THE FORMULA

    in which R2 and R3 are defined as above, IN THE PRESENCE OF AN ORGANIC SOLVENT. The novel compounds are outstandingly active as herbicides and are particularly useful as selective herbicides.

    Abstract translation: 某些新的4-氨基-1,2,4-三嗪-5-酮化合物，其中R 1和R 4为氢，烷基，环烷基，取代的苯基或苯基; R2是氢或烷基; R3是氢，烷基，苯基，卤代烷基，苯基烷基或烷基苯基，烷氧基苯基或烷基巯基; 通过包含反应式中R1和R4如上定义的式R 1 -CO-NH-N = C-COOR（II）| R4的GLYOXYLAC酸酯2-氰乙酯的新方法制备，R是 1至4个碳原子，与有机溶剂存在下，R2和R3定义如上所定义的式II R2 H2N-N型角（R3）的氢化衍生物反应。 新型化合物作为除草剂具有突出的活性，并且特别用作选择性除草剂。

    N-diaryl-pyridyl-methyl-imidazoles salts thereof
    2.
    发明授权
    N-diaryl-pyridyl-methyl-imidazoles salts thereof 失效
    N-二元 - 吡啶基 - 甲基咪唑烷钠盐

    公开(公告)号：US3629273A

    公开(公告)日：1971-12-21

    申请号：US3629273D

    申请日：1969-07-03

    Applicant: BAYER AG

    Inventor： DRABER WILFRIED ,  BUCHEL KARLHEINZ ,  PLEMPEL MANFRED

    IPC: C07D213/30 ,  C07D31/42

    CPC classification number: C07D213/30

    Abstract: N-DIARYL-PYRIDYL-METHYL-IMIDAZOLES OF THE FORMULA:

    1-(PYRIDYL-C(-PHENYLENE-(X)N)(-PHENYLENE-(X)N1)-),2-R,

    4-R1,5-R2-IMIDAZOLE

    WHEREIN

    R, R1 AND R2 ARE EACH HYDROGEN, STRAIGHT OR BRANCHED CHAIN LOWER ALKYL OR STRAIGHT OR BRANCHED CHAIN LOWER ALKENYL. X IS STRAIGHT OR BRANCHED CHAIN ALKYL OF 1 TO 12 CARBON ATOMS, STRAIGHT OR BRANCHED CHAIN ALKENYL OF 1 TO 12 CARBON ATOMS OR AN ELECTRONEGATIVE MOIETY, AND N AND N1 ARE EACH INTEGERS FROM 0 TO 2,

    OR PHARMACEUTICALLY ACCEPTABLE NON-TOXIC SALTS THEREOF ARE PRODUCED BY REACTING DIARYL-PYRIDYL CARBINOLS OF THE FORMULA:

    (HO-C(-PHENYLENE-(X)N)(-PHENYLENE-(X)N1)-)PYRIDINE

    WHEREIN X, N AND N1 ARE AS ABOVE DEFINED, IN AN INERT ORGANIC SOLVENT WITH A REAGENT SUITABLE FOR CHLORINATION OF TERTIARY ALCOHOLS AND REACTING THE DIARYL-PYRIDYL-METHYL CHLORIDE THUS PRODUCED WITH AN ACID-BINDING AGENT AND IMIDAZOLE OR LOWER ALKYL IMIDAZOLE. THE SALTS ARE OBTAINED BY REACTION OF THE COMPOUNDS WITH THE CORRESPONDING ACID. THESE COMPOUNDS ARE USEFUL AS ANTIMYCOTICS AND SHOULD GENERALLY BE ADMINISTERED IN THE RANGE OF ABOUT 20 TO 100 M./KG.

    N-methyl-imidazole derivatives and their production
    3.
    发明授权
    N-methyl-imidazole derivatives and their production 失效
    N-甲基咪唑衍生物及其制备

    公开(公告)号：US3928348A

    公开(公告)日：1975-12-23

    申请号：US31040072

    申请日：1972-11-29

    Applicant: BAYER AG

    Inventor： DRABER WILFRIED ,  BUCHEL KARL HEINZ ,  REGEL ERIK ,  PLEMPEL MANFRED

    IPC: A61K31/495 ,  A61K31/505 ,  C07D241/12 ,  C07D403/06 ,  C07D237/08

    CPC classification number: C07D403/06 ,  A61K31/495 ,  A61K31/505 ,  C07D241/12

    Abstract: N-methyl-imidazole derivatives of the formula:

    OR A PHARMACEUTICALLY ACCEPTABLE NON-TOXIC SALT THEREOF, WHEREIN X is an unsubstituted or substituted 6-membered hetero-aromatic moiety having two nitro heteroatoms, Y is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety or an unsubstituted or substituted aryl moiety, and Z is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety, an unsubstituted or substituted aryl moiety, an unsubstituted or substituted pyridyl moiety or an alkoxycarbonyl moiety, ARE USEFUL AS ANTIMYCOTIC AGENTS.

    Abstract translation: 下式的N-甲基 - 咪唑衍生物：

    Cyano substituted phenylhydrazones of 1 2-dicarbonyl compounds
    8.
    发明授权
    Cyano substituted phenylhydrazones of 1 2-dicarbonyl compounds 失效
    1,6-二氧化碳化合物的氰基取代苯乙烯

    公开(公告)号：US3641098A

    公开(公告)日：1972-02-08

    申请号：US3641098D

    申请日：1968-09-24

    Applicant: BAYER AG

    Inventor： BUCHEL KARL-HEINZ ,  DRABER WILFRIED ,  HAMMANN INGEBORG ,  UNTERSTENHOFER GUNTER

    IPC: C07C133/00

    Abstract: A-(HALO, CYANO, NITRO AND AZIDO)-A-(ALKANOYL, CARBOALKOXY (I.E. ALKOXY CARBONYL), AMINO AND MONO- AND DIALKYL AMINO)-CARBONYL-(UNSUBSTITUTED AND MONO TO PENTA ALKY AND/OR ELECTROEGATIVE SUBSTITUENT (E.G. HALO, NITRO, CYANO, TRIFFUOROMETHYL, TRIFLUOROMETHYL-, -MERCAPTO, -SULFONYL AND -SULFOXYL, ALKOXY, ALKYL SUFONYL AND/OR DIMETHYLMINO SULFONYL)-SUBSTITUTED) PHENYLHYDRAZONES AND THEIR CORRESPONDING ALKALI METAL, ALKALINE EARTH METAL AND AMINE SALTS, WHICH POSSESS PEDTICIDAL, ESPECIALLY ACARICIDAL AND INSECTICDAL, PROPERTIES AND WHICH MAY BE PRODUCED BY CONVENTIONAL METHODS.

    Diaryl-pyridyl-imidazole methanes and their production
    10.
    发明授权
    Diaryl-pyridyl-imidazole methanes and their production 失效
    二芳基 - 吡啶基 - 咪唑甲烷及其制备

    公开(公告)号：US3910936A

    公开(公告)日：1975-10-07

    申请号：US36784973

    申请日：1973-06-07

    Applicant: BAYER AG

    Inventor： DRABER WILFRIED ,  PLEMPEL MANFRED ,  BUCHEL KARL HEINZ

    IPC: C07D401/06 ,  A61K31/435 ,  A61K31/44 ,  A61K31/4427 ,  A61P31/04 ,  C07D213/06 ,  C07D233/56 ,  C07D521/00 ,  C07D213/32

    CPC classification number: C07D231/12 ,  A61K31/44 ,  C07D233/56 ,  C07D249/08

    Abstract: Diaryl-pyridyl-imidazolyl methanes of the formula

    AND PHARMACEUTICALLY ACCEPTABLE NON-TOXIC SALTS THEREOF, WHEREIN R1 and R2 are the same or different alkyl of 1 to 4 carbon atoms, ARE PRODUCED EITHER BY A. REACTING A (DIALKYLPHENYL-PHENYL-PYRIDYL)-METHANOL OF THE FORMULA

    WHEREIN R1 and R2 are as above defined, with thionyl-bis-imidazole in the presence of an inert organic diluent at a temperature of from -20* C to about 150* C; or B. REACTING A (DIALKYLPHENYL-PHENYL-PYRIDYL)-METHYL HALIDE OF THE FORMULA

    WHEREIN R1 and R2 are as above defined and Hal is chlorine or bromine, WITH IMIDAZOLE IN THE PRESENCE OF AN ACID BINDING AGENT AT A TEMPERATURE OF FROM 20* C to about 180* C. The diaryl-pyridyl-imidazole methanes of the present invention are useful for their antimycotic activity.

    Abstract translation: 具有下式的二芳基 - 吡啶基 - 咪唑基甲烷及其药学上可接受的非毒性盐，其中R 1和R 2是相同或不同的1至4个碳原子的烷基，由A产生A.反应A（对二苯基苯基 - 吡啶基） 在惰性有机稀释剂存在下，在-20℃至约150℃的温度下，在亚甲基 - 双 - 咪唑存在的情况下，R1和R2如上所定义。 或B.反应式（R 1和R 2如上所定义）的式（二烷基苯基 - 苯基 - 吡啶基） - 甲基卤化物，Hal是氯或溴，在酸性粘合剂存在下，在20℃的温度下存在咪唑 约180℃

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