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11.发明授权Chemo-enzymatic process for the preparation of opticaly enriched β-benzyl-γ-butyrolactones 有权用于制备光学富集的β-苄基-γ-丁内酯的化学 - 酶法公开(公告)号：US07153983B2
公开(公告)日：2006-12-26
申请号：US10376508
申请日：2003-03-03
IPC分类号： C07D307/20
CPC分类号： C07D307/33
摘要： The present invention relates to a novel synthetic process for the enriched preparation of substituted R(+)β-benzyl-γ-butyrolactone (1) as shown in the drawing wherein R1 and R2 independently or in combination represent the following groups: i.e. R1═R2═H, —OCnH2n+1 (where n=1 to 8); R1, and R2 together represents —O(CH2)mO— (where m=2 to 4)
摘要翻译： 本发明涉及用于富集制备取代的R（+） - β-苄基-γ-丁内酯（1）的合成方法，如图所示，其中R 1和R 2 独立地或组合地表示以下基团：即R 1 -R 2 -H，-OC n H， 2n + 1（其中n = 1至8）; R 1和R 2一起表示-O（CH 2）2 O - （其中m = 2 到4）
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12.发明授权Stereoselective chemoenzymatic process for the preparation of optically enriched phenylglycidates as precursors of taxol side chain 有权用于制备作为紫杉醇侧链前体的光学富集的苯基甘氨酸酯的立体选择性化学酶学方法公开(公告)号：US07060471B2
公开(公告)日：2006-06-13
申请号：US10798199
申请日：2004-03-10
申请人： Naveen Anand , Munish Kapoor , Subhash Chandra Taneja , Surrinder Koul , Rattan Lal Sharma , Ghulam Nabi Qazi
发明人： Naveen Anand , Munish Kapoor , Subhash Chandra Taneja , Surrinder Koul , Rattan Lal Sharma , Ghulam Nabi Qazi
IPC分类号： C12P17/02 , C07D301/26
CPC分类号： C12P41/004 , C12P7/62 , C12P17/02
摘要： The present invention relates to a novel and efficient chemoenzymatic process of preparation of optically active trans alkyl phenylglycidates. The invention particularly discloses a novel process for the chemoenzymatic synthesis of two enantiomers of trans alkyl phenylglycidate i.e. alkyl(2S,3R)-phenylglycidate and alkyl(2R,3S)-phenylglycidate of formulae 7 and 8 respectively
摘要翻译： 本发明涉及一种制备光学活性的反式烷基苯基缩水甘油酯的新颖有效的化学酶学方法。 本发明特别公开了分别反应式合成反式烷基苯基缩水甘油酯的对映异构体（即式7和8的（2S，3R） - 苯基缩水甘油酸酯和（2R，3S） - 苯基缩水甘油基）烷基酯的新方法
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公开(公告)号：US07262296B2
公开(公告)日：2007-08-28
申请号：US11300295
申请日：2005-12-15
IPC分类号： C07D295/192 , C07D265/30
CPC分类号： C07D295/185 , A23L27/205 , C07D311/58 , C07D319/18
摘要： The present invention relates to novel compounds possessing specific hot, pungent and spicy taste when subjected to direct pungency evaluation, which may be useful as food additives and anti-oxidants, however the said compounds do not add to any nutritional value but the synthesised compounds can possess useful pharmacological properties which is expected to find application in new test models for the development of anti-inflammatory drugs, bioavailability enhancers and for the study of hepatic drug metabolising mechanism; also relates to a process for preparing the said compounds.
摘要翻译： 本发明涉及当经受直接刺激性评估时具有特别热，刺鼻和辛辣味道的新化合物，其可用作食品添加剂和抗氧化剂，然而所述化合物不增加任何营养价值，但合成的化合物可以 具有有用的药理学性质，预计可用于新型抗炎药，生物利用度增强剂研发试验和肝脏药物代谢机制研究; 还涉及制备所述化合物的方法。
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14.发明授权Synergistic composition of bioactive fraction isolated from barleria prionitis linn and a method of treatment for hepatotoxicity, immuno-deficiency and fatigue and a process thereof 失效从barperia prionitis linn分离的生物活性成分的协同组成和肝毒性，免疫缺陷和疲劳的治疗方法及其过程公开(公告)号：US06664236B2
公开(公告)日：2003-12-16
申请号：US10100166
申请日：2002-03-19
申请人： J. L. Suri , S. K. Banerjee , Subhash Chandra Taneja , A. S. Anand , Anil Prabhakar , Bupinder Singh Jaggi , A. K. Saxena , Bal Krishan Chandan , Sukhdev Swami Handa
发明人： J. L. Suri , S. K. Banerjee , Subhash Chandra Taneja , A. S. Anand , Anil Prabhakar , Bupinder Singh Jaggi , A. K. Saxena , Bal Krishan Chandan , Sukhdev Swami Handa
IPC分类号： A01N6500
CPC分类号： A61K36/19 , A61K2300/00
摘要： The present invention provides a synergistic composition of bioactive fraction essentially constituting iridoid glucosides, acetyl barlerin and shanzhiside methyl ester isolated from a plant source Barleria prionitis linn along with a process for the isolation of the bioactive fraction, the present invention also relates to a method of treating mammals and humans for hepatotoxicity, stress and immuno-deficiency with the synergistic bioactive composition.
摘要翻译： 本发明提供了生物活性部分的协同组合物，其基本上构成了从植物来源的Barleria prionitis linn分离的环烯醚萜苷，乙酰大肠杆菌素和shanzhiside甲酯以及分离生物活性级分的方法，本发明还涉及一种方法 用协同生物活性组合物治疗哺乳动物和人类的肝毒性，应激和免疫缺陷。
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公开(公告)号：US07057040B2
公开(公告)日：2006-06-06
申请号：US10067546
申请日：2002-02-07
IPC分类号： C07D295/192
CPC分类号： C07D295/185 , A23L27/205 , C07D311/58 , C07D319/18
摘要： The present invention relates to novel compounds possessing specific hot, pungent and spicy taste when subjected to direct pungency evaluation, which may be useful as food additives and anti-oxidants, however the said compounds do not add to any nutritional value but the synthesised compounds can possess useful pharmacological properties which is expected to find application in new test models for the development of anti-inflammatory drugs, bioavailability enhancers and for the study of hepatic drug metabolising mechanism; also relates to a process for preparing the said compounds.
摘要翻译： 本发明涉及当经受直接刺激性评估时具有特别热，刺鼻和辛辣味道的新化合物，其可用作食品添加剂和抗氧化剂，然而所述化合物不增加任何营养价值，但合成的化合物可以 具有有用的药理学性质，预计可用于新型抗炎药，生物利用度增强剂研发试验和肝脏药物代谢机制研究; 还涉及制备所述化合物的方法。
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