Plant growth regulant compositions
    11.
    发明授权
    Plant growth regulant compositions 失效
    植物生长调节剂组合物

    公开(公告)号:US4350520A

    公开(公告)日:1982-09-21

    申请号:US213704

    申请日:1980-12-05

    摘要: The imidazole-2-carboxylic acid amides of the general formula ##STR1## in which R represents alkyl, have powerful growth-regulating properties.The invention provides a method of regulating the growth of plants, which comprises applying to the plants, or to a habitat thereof, a compound of the formula (I) alone or in the form of a composition containing as active ingredient a compound of the formula (I) in admixture with a diluent or carrier.

    摘要翻译: 通式为其中R代表烷基的通式为“IMAGE”(I)的咪唑-2-羧酸酰胺具有强大的生长调节性质。 本发明提供了一种调节植物生长的方法,其包括向植物或其栖息地施用式(I)化合物单独或以包含作为活性成分的化合物形式的化合物施用式 (I)与稀释剂或载体混合。

    N-(1,2,2,2-tetrachloroethyl)-formimide-chloride for synthesizing
trichlorothiazole
    12.
    发明授权
    N-(1,2,2,2-tetrachloroethyl)-formimide-chloride for synthesizing trichlorothiazole 失效
    N-(1,2,2,2-四氯乙基) - 用于合成三氯噻唑的酰胺氯

    公开(公告)号:US4013674A

    公开(公告)日:1977-03-22

    申请号:US639137

    申请日:1975-12-09

    IPC分类号: C07D277/32 C07D263/30

    CPC分类号: C07D277/32

    摘要: The new compound N-(1,2,2,2-tetrachloroethyl)-formimide chloride of the formula ##STR1## is produced by reacting a substituted formamide of the formula ##STR2## wherein X is OH or Cl,With approximately the stoichiometrically required amount of a highly reactive inorganic acid chloride, e.g. phosphorus pentachloride. The compound (I) can be reacted with sulfur at about 150.degree. to 250.degree. C to produce trichlorothiazole of the formula ##STR3## which is known to have insecticidal activity.

    Process for the preparation of tetrachloropyrimidine
    16.
    发明授权
    Process for the preparation of tetrachloropyrimidine 失效
    四氯嘧啶的制备方法

    公开(公告)号:US4125723A

    公开(公告)日:1978-11-14

    申请号:US851309

    申请日:1977-11-14

    CPC分类号: C07D239/30

    摘要: Process for the preparation of tetrachloropyrimidine, characterized in that compounds of the formula ##STR1## wherein R = a radical which can be split off under the reaction conditions andR' = optionally substituted lower allyl radical, are reacted with chlorine or agents which release chlorine, preferably at temperatures from 0.degree. to 150.degree. C and using more than 7.5 mols of chlorine, preferably 8 to 9 mols of chlorine.

    摘要翻译: 制备四氯嘧啶的方法,其特征在于其中R =可在反应条件下分离的基团和R'=任选取代的低级烯丙基的式“IMAGE”化合物与氯或释放氯的试剂反应 ,优选在0℃至150℃的温度下,使用大于7.5摩尔的氯,优选8至9摩尔的氯。

    Benzodiazepine-diones, a process for their production and their use as
medicaments
    18.
    发明授权
    Benzodiazepine-diones, a process for their production and their use as medicaments 失效
    苯二氮卓类药物,其生产过程及其用作药物

    公开(公告)号:US4187306A

    公开(公告)日:1980-02-05

    申请号:US922419

    申请日:1978-07-06

    摘要: The invention covers compounds of the formula ##STR1## in which R.sup.1 and R.sup.5 each represents 0, 1, 2, 3 or 4 of the following substituents: alkyl, hydroxyl, acyloxy, alkoxy, nitro, amino, alkylamino, dialkylamino, acylamino, acylalkylamino, alkoxycarbonylamino, halogen, trifluoromethyl, cyano, carboxyl, alkoxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, aminosulphonyl, alkylaminosulphonyl, dialkylaminoamino, R.sup.2 is hydrogen, optionally substituted alkyl, aralkyl or aryl or heterocyclo-alkyl, acyl or alkoxycarbonyl, and R.sup.3 and R.sup.4 are each hydrogen, or optionally substituted alkyl, aralkyl, aryl or hetero-aryl, are useful as medicaments which have an action on the central nervous system, in particular as, for example, tranquilizers and/or antiamnesics. Also included in the invention are methods for preparing said compounds, compositions containing them and methods for the use of said compounds and compositions.

    摘要翻译: 本发明涵盖下式的化合物,其中R 1和R 5各自表示0,1,2,3或4个以下取代基:烷基,羟基,酰氧基,烷氧基,硝基,氨基,烷基氨基,二烷基氨基,酰氨基,酰基烷基氨基 烷氧基羰基,氨基羰基,氨基磺酰基,烷基氨基磺酰基,二烷基氨基氨基,R2是氢,任意取代的烷基,芳烷基或芳基或杂环烷基,酰基或烷氧基羰基,R3和R4是 每个氢或任选取代的烷基,芳烷基,芳基或杂芳基可用作对中枢神经系统具有作用的药物,特别是例如镇定剂和/或抗病毒药物。 本发明还包括制备所述化合物的方法,含有它们的组合物和使用所述化合物和组合物的方法。