公开(公告)号：US07148227B2

公开(公告)日：2006-12-12

申请号：US10508409

申请日：2003-03-19

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schöfl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schöfl

IPC分类号： A61K31/519 ,  C07D487/04 ,  C07C69/738

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C255/57

摘要： The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L1 represents cyano, S(═O)nA1 or C(═O)A2, wherein A1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A2 stands for C1–C8 alkoxy, C1–C6 haloalkoxy or one of the groups named in A1; and n stands for 0, 1 or 2; L2, L3 represent hydrogen or halogen; L4, L5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R2 represents hydrogen or R1; R1 and R2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R1 and/or R2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.

摘要翻译： 本发明涉及式（I）的三唑并嘧啶，其中取代基定义如下：L 1表示氰基，S（-O）n A 1 或其中A 1代表氢，羟基，烷基，烷基氨基或二烷基氨基;或C（= O） A 2代表C 1 -C 8烷氧基，C 1 -C 6烷基，C 1 -C 6 - >卤代烷氧基或在A 中命名的基团之一; 而n代表0,1或2; L 2，L 3表示氢或卤素; L 4，L 5代表氢，卤素或烷基; X表示卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1表示烷基，卤代烷基，环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环 含有一个至四个来自含有O，N或S的基团的杂原子; R 2表示氢或R 1; R 1和R 2可以与它们所键合的氮原子一起形成五元或六元环，其可被中断和/或被 来自O，N和S族的原子; 其中R 1和/或R 2可以根据描述被取代。 本发明还涉及用于生产所述化合物的方法和中间产物，含有后者的试剂和所述化合物用于防治有害真菌的用途。

公开(公告)号：US06767923B2

公开(公告)日：2004-07-27

申请号：US10282023

申请日：2002-10-29

申请人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

发明人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

IPC分类号： A61K31215

CPC分类号： C07C323/25 ,  A01N31/16 ,  C07C43/23 ,  C07C69/017

摘要： Benzhydryl derivatives of the formula I, where the index and the variables are as defined below: X is oxygen or sulfur; R1, R3 are halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylcarbonyloxy, formyloxy, alkylthio, alkenylthio, alkynylthio, alkylamino, dialkylamino, alkylcarbonyl or formyl, where the carbon atoms in the radicals mentioned may be partially or fully halogenated; R2 is halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkoxy, haloalkyl or haloalkoxy, where the groups R2 may be different if n=2; R4 is alkyl, alkenyl or alkynyl, where the carbon atoms in these radicals may be unsubstituted or partially or fully halogenated; R5, R6 are hydroxyl, alkyl, alkenyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, cycloalkyl, cycloalkylalkyl, cycloalkoxy or cycloalkylalkoxy; n is 0, 1 or 2; processes for preparing the compounds I, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的二苯甲基衍生物，其中指数和变量如下定义：X是氧或硫; R 1，R 3是卤素，氰基，硝基，羟基，巯基，氨基，烷基，烯基， 炔基，烷氧基，烯氧基，炔氧基，烷基羰基氧基，甲酰氧基，烷硫基，烯硫基，炔硫基，烷基氨基，二烷基氨基，烷基羰基或甲酰基，其中所述基团中的碳原子可以被部分或完全卤化; R 2是卤素，氰基， 硝基，羟基，巯基，氨基，烷基，烷氧基，卤代烷基或卤代烷氧基，其中如果n = 2，基团R 2可以不同; R 4是烷基，烯基或炔基，其中这些基团中的碳原子 R 5为羟基，烷基，烯基，卤代烷基，卤代烯基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，环烷基，环烷基烷基，环烷氧基或环烷基烷氧基; n为0,1或 2;制备化合物I的方法，包含它们的组合物及其用途 描述了植物病原性有害真菌。

公开(公告)号：US07307172B2

公开(公告)日：2007-12-11

申请号：US10484250

申请日：2002-07-16

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Günter Krummel

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Günter Krummel

IPC分类号： A61K31/41 ,  A01N43/653 ,  C07D249/00

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

摘要翻译： 本发明涉及式（I）的7-氨基三唑并嘧啶，其中取代基具有以下含义：R 1，R 2表示氢，烷基，烯基，炔基 ，环烷基，苯基，萘基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂环基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂芳基，或R 1和R 2可以， 与它们结合的氮原子一起形成含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的五元或六元环; R 3表示烷基，烯基，炔基，环烷基，苯基烷基和烷基卤; 根据描述，R 3和R 2可以是未取代的或部分或完全取代的; X表示卤素，氰基，烷氧基，烷基卤，苯基或被R a取代的苯基。 本发明还涉及用于生产所述化合物的方法和中间产物，含有该化合物的试剂及其用途。

公开(公告)号：US07282503B2

公开(公告)日：2007-10-16

申请号：US10532769

申请日：2003-11-14

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schöfl

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schöfl

IPC分类号： A01N43/50 ,  A01N43/76 ,  A01N43/80 ,  A01N43/90

CPC分类号： A01N43/90 ,  A01N2300/00

摘要： Disclosed are fungicidal mixtures containing a synergistically effective amount of A) a triazolopyrimidine of formula I, and B) imidazole derivatives of formula II, wherein X1 and X2 represent halogen and phenyl which can be substituted by halogen or alkyl, or X1 and X2 form a difluoromethylendioxyphenyl group along with the bridging C═C double bond, X3 represents cyano or halogen, and X4 represents dialkylamino or isoxazol-4yl that can carry two alkyl radicals. The invention also relates to methods for controlling destructive fungi by means of mixtures of compounds I and II, agents containing said mixtures, and the use of compounds I and II for producing such mixtures.

摘要翻译： 公开了含有协同有效量的A）式I的三唑并嘧啶和B）式II的咪唑衍生物的杀真菌混合物，其中X 1和X 2代表卤素和 可被卤素或烷基取代的苯基或X 1和X 2 2与桥连CC双键一起形成二氟甲基内酰氧基苯基，X 3 O >表示氰基或卤素，X 4表示可带有两个烷基的二烷基氨基或异恶唑-4-基。 本发明还涉及通过化合物I和II的混合物控制破坏性真菌的方法，含有所述混合物的试剂以及化合物I和II用于制备这种混合物的方法。

公开(公告)号：US07038047B2

公开(公告)日：2006-05-02

申请号：US10483599

申请日：2002-07-08

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  C07C69/612 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Substituted 6-(2-methoxy-phenyl)-triazolopyrimidines of formula I in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or substituted as defined in the description, or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; L1, L2 independently denote hydrogen or halogen, provided that at least one from L1 or L2 is halogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

摘要翻译： 其中R 1和R 2的取代的6-（2-甲氧基 - 苯基） - 三唑并嘧啶独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的卤代烯基，环烷基，苯基，萘基或5-或6-元杂环基，或含有一至四个的5-或6-元杂芳基 氮原子或一至三个氮原子和一个硫或氧原子，或其中R 1和R 2基团可以是未取代的或如说明书中定义的取代的，或R R 1和R 2与中间的氮原子一起表示含有1-4个氮原子或一至三个氮原子和一个硫原子的5-或6-元杂环 或氧原子，其可以被取代; L 1，L 2，L 2独立地表示氢或卤素，条件是至少一个L 1或L 2， 是卤素; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US06593315B2

公开(公告)日：2003-07-15

申请号：US09896971

申请日：2001-07-02

申请人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N3736

CPC分类号： C07C251/86 ,  A01N37/50

摘要： Salicylic acid derivatives of the formula I, where the index and the substituents have the following meanings: X is halogen, NO2, cyano, alkyl or alkoxy; m is 0, 1, 2 or 3, it being possible for the substituents X to be different from each other if n is greater than 1; A is OH, alkoxy, NH2, NHCH3 or N(CH3)2; R1 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, comprising one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted; R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio, processes for the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.

摘要翻译： 式I的水杨酸衍生物，其中指数和取代基具有以下含义：X是卤素，NO 2，氰基，烷基或烷氧基; m是0,1,2或3，取代基X可以是 如果n大于1，A是不同的; A是OH，烷氧基，NH2，NHCH3或N（CH3）2; R1是苯基，萘基，环烷基，5元或6元杂芳基或5元或6- 包括一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未取代或取代的; R2是氢，氰基，烷基，烯基，炔基，卤代烷基， 烷氧基或烷硫基，制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US06576595B1

公开(公告)日：2003-06-10

申请号：US10251783

申请日：2002-09-23

申请人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann

发明人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann

IPC分类号： A01N4316

CPC分类号： C07D311/86 ,  A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84

摘要： Xanthone derivatives of the formula I where the index and the variables are as defined below: n is 0, 1 or 2; R1 is alkyl or haloalkyl; R2,R3 are alkoxy, alkenyloxy or alkynyloxy, or R2 and R3 together form an unsubstituted or substituted oxyalkyleneoxy group; R4 is halogen, cyano, hydroxyl, amino, mercapto, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylcarbonyloxy or alkylcarbonylthio; R5 is a group R4, where the groups R5 may be different if n=2; X, Y are oxygen or sulfur; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的呫吨酮衍生物，其中指数和变量如下：n为0,1或2; R 1为烷基或卤代烷基; R 2为烷氧基，烯氧基或炔氧基，或者R 2和R 3一起形成未取代或取代的 氧基亚烷基氧基; R4是卤素，氰基，羟基，氨基，巯基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基羰基氧基或烷基羰基硫基; R5是R4基团，其中如果n = 2，基团R5可以不同; X ，Y为氧或硫;制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US06696607B2

公开(公告)日：2004-02-24

申请号：US10297287

申请日：2002-12-04

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Norbert Götz ,  Thorsten Volk ,  Gisela Lorenz ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Norbert Götz ,  Thorsten Volk ,  Gisela Lorenz ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann

IPC分类号： C07C23309

CPC分类号： A01N37/36 ,  A01N37/18 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22

摘要： Use of phenethylacrylamides of the formula I: in which the substituents have the following meanings: X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and —O—C(Ra,Rb)—C≡C—R6; Ra,Rb and Rc have the meanings given in the description; m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1; Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl; R1,R2 independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3; R3,R4,R5,R6 independently of one another are hydrogen, halogen, alkyl, alkoxy, or R3 and R4 together form a cyclopropyl ring, it being possible for the C—R5— and C—R6 bonds can be in the E- or Z-position relative to each other; for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.

摘要翻译： 使用式I的苯乙基丙烯酰胺：其中取代基具有以下含义：X是卤素，烷基，卤代烷基，烷氧基，卤代烷氧基和-OC（R a，R b）-C = CR 6; R a，R b和R c具有说明书中给出的含义; m，n彼此独立地为1至4，如果m或n可以使基团X或Y不同 大于1; Y是卤素，硝基，氰基，烷基，CF 3，烷氧基和苯基; R 1，R 2彼此独立地是氢，卤素，烷基，烷氧基，卤代烷氧基和CF 3; R 3 R 4，R 5，R 6彼此独立地是氢，卤素，烷基，烷氧基或R 3和R 4一起形成环丙基环，其中CR <5> - 和CR 6键可以相对于彼此位于E-或Z-位;用于控制植物病原性真菌害虫，新型苯乙基丙烯酰胺，它们的制备和包含它们的组合物。

公开(公告)号：US06482984B2

公开(公告)日：2002-11-19

申请号：US09760710

申请日：2001-01-17

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Arne Ptock ,  Bernd Müller ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Arne Ptock ,  Bernd Müller ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： C07C23305

CPC分类号： C07C251/48 ,  A01N37/50

摘要： Iminooxy-substituted benzyl phenyl ethers of the formula I in which the substituents and the index are as defined below: Y is H, CH3, F or Cl; Q is C(═CHOCH3)—COOCH3, C(═CHCH3)—COOCH3, C(═NOCH3)—COOCH3, C(═NOCH3)—CONHCH3 or N(—OCH3)—COOCH3; X is hydrogen, halogen, alkyl, alkoxy or CF3; m is 1 or 2, where the radicals X may be different if m=2; R1 is alkyl and R2 is hydrogen or alkyl; or R1 and R2 together are cyclopropyl, cyclopentyl or cyclohexyl; R3 is alkyl or CF3; and R4 is alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl or haloalkynyl; processes and intermediates for their preparation, compositions comprising them, and their use, are described.

摘要翻译： 取代基和指数如下定义的式Iin的亚氨氧基取代的苄基苯基醚：Y是H，CH 3，F或Cl; Q是C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C （= NOCH 3）-COOCH 3，C（= NOCH 3）-CONHCH 3或N（-OCH 3）-COOCH 3; X是氢，卤素，烷基，烷氧基或CF 3; m是1或2，其中基团X可以不同，如果m = 2; R 1是烷基，R 2是氢或烷基; 或者R 1和R 2一起是环丙基，环戊基或环己基; R 3是烷基或CF 3; 和R 4是烷基，烯基，炔基，卤代烷基，卤代烯基或卤代炔基;其制备方法和中间体，包含它们的组合物及其用途。

公开(公告)号：US20060079537A1

公开(公告)日：2006-04-13

申请号：US10531898

申请日：2003-11-14

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(═O)-A or S(═O)pA′; A and A′ are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR1R2 or S(O)nR31, where n and R31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，-C（ - O） - 取代的取代基如下： -A或S（-O） A'; A和A'如说明书所定义; p为0,1或2; m为0,1,2,3,4或5; X是氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 - 至十元饱和的，部分不饱和的或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1和R 2连同 它们所连接的氮原子也可以形成可被来自O，N和S的原子间隔的五元或六元环，其中R 1和/或 R 2可以如说明书中定义的取代; 和R 3是氰基，羟基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，NR 1 R 2或S（O）n 其中n和R 31如在说明书中所定义的; 描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。