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37 条记录 (耗时 0.043 秒)

    Isoxazoline derivatives and their use as herbicides
    32.
    发明授权
    Isoxazoline derivatives and their use as herbicides 失效
    异恶唑啉衍生物及其作为除草剂的用途

    公开(公告)号：US08680290B2

    公开(公告)日：2014-03-25

    申请号：US11574648

    申请日：2005-08-17

    申请人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

    发明人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

    IPC分类号： C07D261/10 ,  A61K31/421

    CPC分类号： C07D261/10 ,  C07D413/12 ,  C07D417/12

    摘要： Compounds of formula (I) wherein the substituents are as defined in claim 1, are suitable for use as herbicides. Also claimed is a process for the preparation of compounds of the formula I, wherein m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ia) by reacting a compound of the formula Ia in a single step or stepwise in succession with compounds of the formula R5—X and/or R6—X, wherein R5 and R6 are as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R6 is C1-C10alkyl or halogen, m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ib) by reacting a compound of the formula Ib with a compound of the formula R5—X, wherein R5 is as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R5 is chlorine, bromine or iodine, m is 1 or 2, and n is 1, and the other substituents are defined as in claim 1, formula (Ic) by reacting a compound of the formula 1e with an N-halosuccinimide and an oxidising agent.

    摘要翻译： 其中取代基如权利要求1中所定义的式（I）化合物适合用作除草剂。 还要求保护的是制备式I化合物的方法，其中m为2且n为1，其它取代基如权利要求1，式（Ia）所定义，通过使式Ia化合物在单一 与式R 5 -X和/或R 6 -X的化合物连续进行步骤或分步步骤，其中R 5和R 6如权利要求1中所定义，X为离去基团，以及制备式I化合物的方法 其中R 6为C 1 -C 10烷基或卤素，m为2且n为1，其它取代基如权利要求1所定义，式（Ib）通过式Ib化合物与式R 5 -X 其中R 5如权利要求1所定义，X为离去基团，以及制备式Ⅰ化合物的方法，其中R 5为氯，溴或碘，m为1或2，n为1， 并且其它取代基如权利要求1所定义，式（Ic）通过使式1e的化合物与N-卤代琥珀酰亚胺和氧化剂反应。

    Isoxazoline Derivatives and Their Use as Herbicides
    33.
    发明申请
    Isoxazoline Derivatives and Their Use as Herbicides 失效
    异恶唑啉衍生物及其作为除草剂的用途

    公开(公告)号：US20080139390A1

    公开(公告)日：2008-06-12

    申请号：US11574648

    申请日：2005-08-17

    申请人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

    发明人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

    IPC分类号： A01N43/80 ,  A01P13/00 ,  C07D261/10 ,  C07D413/12 ,  C07D417/12

    CPC分类号： C07D261/10 ,  C07D413/12 ,  C07D417/12

    摘要： Compounds of formula (I) wherein the substituents are as defined in claim 1, are suitable for use as herbicides. Also claimed is a process for the preparation of compounds of the formula I, wherein m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ia) by reacting a compound of the formula Ia in a single step or stepwise in succession with compounds of the formula R5—X and/or R6—X, wherein R5 and R6 are as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R6 is C1-C10alkyl or halogen, m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ib) by reacting a compound of the formula Ib with a compound of the formula R5—X, wherein R5 is as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R5 is chlorine, bromine or iodine, m is 1 or 2, and n is 1, and the other substituents are defined as in claim 1, formula (Ic) by reacting a compound of the formula 1e with an N-halosuccinimide and an oxidising agent.

    摘要翻译： 其中取代基如权利要求1中所定义的式（I）化合物适合用作除草剂。 还要求保护的是制备式I化合物的方法，其中m为2且n为1，其它取代基如权利要求1，式（Ia）所定义，通过使式Ia化合物在单一 与式R 5 -X和/或R 6 -X的化合物相继步骤或逐步进行，其中R 5和R 0 > 6 如权利要求1中所定义，X是离去基团，以及制备式I化合物的方法，其中R 6为C 1 烷基或卤素，m是2，n是1，其它取代基如权利要求1式（Ib）所定义，通过使式Ib化合物与 式R 5 -X的化合物，其中R 5如权利要求1中所定义，X为离去基团，和其制备方法 式I其中R 5为氯，溴或碘，m为1或2，n为1，其它取代基定义如下： m 1，式（Ic）通过使式1e的化合物与N-卤代琥珀酰亚胺和氧化剂反应。

    Use of cyclic depsipeptides having 12 ring atoms for combating endoparasites, new cyclic despipeptides having 12 ring atoms, and processes for their preparation
    35.
    发明授权
    Use of cyclic depsipeptides having 12 ring atoms for combating endoparasites, new cyclic despipeptides having 12 ring atoms, and processes for their preparation 失效
    具有12个环原子的环状缩水甘油醚与具有12个环原子的新环状脱磷酸酯的反应的内源寄生虫的使用及其制备方法

    公开(公告)号：US5663140A

    公开(公告)日：1997-09-02

    申请号：US372543

    申请日：1995-01-13

    申请人： Jurgen Scherkenbeck ,  Peter Jeschke ,  Andrew Plant ,  Achim Harder ,  Norbert Mencke

    发明人： Jurgen Scherkenbeck ,  Peter Jeschke ,  Andrew Plant ,  Achim Harder ,  Norbert Mencke

    IPC分类号： A61K31/33 ,  A61K31/38 ,  A61K31/41 ,  A61K38/00 ,  A61P33/00 ,  A61P33/10 ,  C07D273/00 ,  C07D273/08 ,  C07D413/06 ,  C07K11/02 ,  A61K35/78

    CPC分类号： C07D273/00 ,  A61K31/33 ,  A61K31/38 ,  C07D413/06

    摘要： The present invention relates to the use of cyclic depsipeptides having 12 ring atoms of the general formula (I) ##STR1## in which R.sup.1 and R.sup.4 independently of one another represent hydrogen, straight-chain or branched alkyl, cycloalkyl, aralkyl, aryl, heteroaryl or heteroarylalkyl, each of which is optionally substituted,R.sup.2, R.sup.3, R.sup.5 and R.sup.6 independently of one another represent hydrogen, straight-chain or branched alkyl having up to 8 carbon atoms, halogenoalkyl, hydroxyalkyl, alkanoyloxyalkyl, alkoxyalkyl, aryloxyalkyl, mercaptoalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, carboxyalkyl, alkoxycarbonylalkyl, arylalkoxycarbonylalkyl, carbamoylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, guanidinoalkyl which can optionally be substituted by one or two benzyloxycarbonyl radicals or by one, two, three or four alkyl radicals, alkoxycarbonylaminoalkyl, 9-fluorenylmethoxycarbonyl(Fmoc)aminoalkyl, alkenyl, cycloalkyl, cycloalkylalkyl, and optionally substituted aryl, arylalkyl, heteroaryl and heteroarylalkyl, and their optical isomers and racemates,in medicine and veterinary medicine for combating endoparasites, to new depsipeptides having 12 ring atoms, and to processes for their preparation.

    摘要翻译： 本发明涉及具有通式（I）的12个环原子的环状缩水甘油酯的用途，其中R 1和R 4彼此独立地表示氢，直链或支链烷基，环烷基，芳烷基， 芳基，杂芳基或杂芳基烷基，其各自任选被取代，R 2，R 3，R 5和R 6彼此独立地表示氢，具有至多8个碳原子的直链或支链烷基，卤代烷基，羟烷基，烷酰氧基烷基，烷氧基烷基，芳氧基烷基， 烷基磺酰基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，羧基烷基，烷氧基羰基烷基，芳基烷氧基羰基烷基，氨基甲酰基烷基，氨基烷基，烷基氨基烷基，二烷基氨基烷基，胍基烷基，其可以任选被一个或两个苄氧基羰基取代或被一个，二个，三个或四个烷基取代，烷氧基羰基氨基烷基， 芴基甲氧基羰基（Fmoc）氨基烷基，烯基，环烷基，环烷基烷基和任选取代的a 芳基烷基，杂芳基和杂芳基烷基，以及它们的光学异构体和外消旋体，在用于抗内寄生物的医药和兽医学中，具有12个环原子的新的缩肽，以及它们的制备方法。