公开(公告)号：US6037378A

公开(公告)日：2000-03-14

申请号：US229972

申请日：1999-01-14

申请人： Thomas Grote ,  Herbert Bayer ,  Ruth Muller ,  Hubert Sauter ,  Reinhard Kirstgen ,  Volker Harries ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann

发明人： Thomas Grote ,  Herbert Bayer ,  Ruth Muller ,  Hubert Sauter ,  Reinhard Kirstgen ,  Volker Harries ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann

IPC分类号： C07C249/04 ,  A01N35/10 ,  A01N37/36 ,  A01N37/50 ,  C07C20060101 ,  C07C251/34 ,  C07C251/50 ,  C07C251/60 ,  C07C251/62 ,  C07C255/62 ,  C07C255/64 ,  C07C259/04 ,  C07C259/12 ,  C07C317/16 ,  C07C317/26 ,  C07C323/10 ,  C07C323/47 ,  C07C327/38 ,  C07C327/58 ,  C07C381/00 ,  A01N33/24 ,  C07C251/32 ,  C07C255/10

CPC分类号： A01N37/50 ,  C07C251/60

摘要： Phenylacetic acid derivatives of the formula I ##STR1## where the substituents and the index have the following meanings: X is NOCH.sub.3, CHOCH.sub.3, CHCH.sub.3 ;Y is O, NRR.sup.1,R independently of one another are hydrogen and C.sub.1 -C.sub.4 -alkyl;R.sup.2 is cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy;m is 0, 1 or 2, it being possible for the radicals R.sup.2 to be different when m is 2;R.sup.3 is hydrogen, cyano, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl;R.sup.4, R.sup.5 and R.sup.6 have the meanings given in claim 1,and their salts, a process and intermediates for the preparation of these compounds, and compositions comprising them for controlling animal pests and harmful fungi.

摘要翻译： 其中取代基和指数具有以下含义的式I的苯乙酸衍生物：X为NOCH 3，CHOCH 3，CHCH 3; Y是O，NR R 1，R 2彼此独立地是氢和C 1 -C 4 - 烷基; R2是氰基，硝基，三氟甲基，卤素，烷基和烷氧基; m为0,1或2，当m为2时，基团R2可能不同; R3是氢，氰基，C1-C4-烷基，C1-C4卤代烷基，C3-C6-环烷基; R4，R5和R6具有权利要求1中给出的含义，其盐，制备这些化合物的方法和中间体，以及包含它们的用于控制动物害虫和有害真菌的组合物。

公开(公告)号：US06380231B1

公开(公告)日：2002-04-30

申请号：US09287274

申请日：1999-04-07

申请人： Bernd Müller ,  Reinhard Kirstgen ,  Hartmann König ,  Michael Rack ,  Klaus Oberdorf ,  Franz Röhl ,  Hubert Sauter ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Volker Harries

发明人： Bernd Müller ,  Reinhard Kirstgen ,  Hartmann König ,  Michael Rack ,  Klaus Oberdorf ,  Franz Röhl ,  Hubert Sauter ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Volker Harries

IPC分类号： A01N43653

CPC分类号： C07D401/04 ,  A01N43/56 ,  A01N43/653 ,  C07D231/20 ,  C07D249/12

摘要： Compounds of formula I wherein n is 0, 1, 2, 3, or 4; R is nitro, cyano, halogen, unsubstituted or substituted alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy or two adjacent radicals R form an optionally substituted three or four membered bridge; R1, R2 are C1-C4-alkyl; and R3 is a substituted pyrazole or triazole ring; their preparation and intermediates adapted therefore, and their use for controlling animal and fungal pests.

摘要翻译： 式I的化合物是0,1,2,3或4; R是硝基，氰基，卤素，未取代或取代的烷基，烯基，炔基，烷氧基，烯氧基，炔氧基或两个相邻基团R形成任选取代的三或四个 R1，R2是C1-C4烷基; 和R 3是取代的吡唑或三唑环;其制备和中间体因此适应，以及它们用于控制动物和真菌害虫的用途。

公开(公告)号：US06255352B1

公开(公告)日：2001-07-03

申请号：US09423860

申请日：1999-11-17

申请人： Wassilios Grammenos ,  Ruth Müller ,  Hubert Sauter ,  Herbert Bayer ,  Thomas Grote ,  Andreas Gypser ,  Reinhard Kirstgen ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Ruth Müller ,  Hubert Sauter ,  Herbert Bayer ,  Thomas Grote ,  Andreas Gypser ,  Reinhard Kirstgen ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann

IPC分类号： A01N3324

CPC分类号： A01N35/10

摘要： A method for control of harmful fungi is provided by treating the fungi, or the materials, plants, the soil or seeds to be protected against fungal infection, with an effective amount of a bisoxime of the formula I or a salt or adduct thereof, the index and the substituents having the following meanings: R1 is halogen, alkyl or haloalkyl; R2 is cyano, nitro, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, alkylamino, dialkylamino, alkylaminocarbonyl, substituted or unsubstituted phenyl, phenoxy or phenylthio; n is 0, 1, 2 or 3; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl or phenylalkyl.

摘要翻译： 通过用有效量的式I的二肟或其盐或其加合物处理真菌或材料，植物，待保护的土壤或种子免受真菌感染，提供有害真菌的控制方法，指数 并且具有以下含义的取代基：R 1是卤素，烷基或卤代烷基; R 2是氰基，硝基，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，烷基氨基，二烷基氨基，烷基氨基羰基，取代或未取代的苯基，苯氧基或苯硫基; n 为0,1,2或3; R3为烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基或苯基烷基。

公开(公告)号：US06583090B1

公开(公告)日：2003-06-24

申请号：US09623178

申请日：2000-08-29

申请人： Markus Gewehr ,  Roland Götz ,  Thomas Grote ,  Hubert Sauter ,  Norbert Götz ,  Herbert Bayer ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries ,  Oliver Cullmann

发明人： Markus Gewehr ,  Roland Götz ,  Thomas Grote ,  Hubert Sauter ,  Norbert Götz ,  Herbert Bayer ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries ,  Oliver Cullmann

IPC分类号： A01N4356

CPC分类号： C07D231/12 ,  C07D231/16 ,  C07D233/56 ,  C07D233/64 ,  C07D233/68 ,  C07D249/08 ,  C07D249/10 ,  C07D249/12 ,  C07D261/08 ,  C07D261/10 ,  C07D261/12 ,  C07D263/32 ,  C07D263/34 ,  C07D403/12 ,  C07D413/12

摘要： The invention relates to hetaryl-substituted benzyl phenyl ethers of formula (I) in which the substituents have the following meanings: (Q): C(═CHOCH3)—COOCH3, C(═CHCH3)—COOCH3, C(═NOCH3)—COOCH3, C(═NOCH3)—CONHCH3, N(—OCH3)—COOCH3 or a group F, G, H or J, whereby # characterizes the bond with the phenyl ring, and (X) five-linked heteroaryl which is optionally substituted by a group Y2p and which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom. The invention also relates to the salts of the inventive hetaryl-substituted benzyl phenyl ethers, to the production of compounds (I), and to the use of compounds (I) for combating harmful fungi and animal pests.

摘要翻译： 本发明涉及式（I）的杂芳基取代的苄基苯基醚，其中取代基具有以下含义：（Q）：C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C（= NOCH 3） - COOCH 3，C（= NOCH 3）-CONHCH 3，N（-OCH 3）-COOCH 3或基团F，G，H或J，其中＃表示与苯环的键，和（X）任选取代的五连接杂芳基 由Y2P组成，其中含有1-4个氮原子或一至三个氮原子和一个硫或氧原子。 本发明还涉及本发明的杂芳基取代的苄基苯基醚的盐，涉及化合物（I）的生产，以及化合物（I）用于防治有害真菌和动物害虫的用途。

公开(公告)号：US06232339B1

公开(公告)日：2001-05-15

申请号：US09358474

申请日：1999-07-21

申请人： Andreas Gypser ,  Thomas Grote ,  Hubert Sauter ,  Herbert Bayer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Arne Ptock ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries ,  Franz Röhl

发明人： Andreas Gypser ,  Thomas Grote ,  Hubert Sauter ,  Herbert Bayer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Arne Ptock ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries ,  Franz Röhl

IPC分类号： C07C27128

CPC分类号： C07C271/28 ,  A01N47/24 ,  C07C2601/02

摘要： Phenylcarbamates of the formula I where: R1 is C1-C4-alkyl; R2 is cyano, nitro, trifluoromethyl, halogen, C1-C4-alkyl and C1-C4-alkoxy; m is 0, 1 or 2, where the radicals R2 may be different if m is 2; R3 is hydrogen, cyano, C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl; R4, R5 and R6 are each as defined in claim 1, and salts thereof, a process and intermediates for preparing these compounds and compositions comprising them for controlling animal pests and harmful fungi are described.

摘要翻译： 式I的苯基氨基甲酸酯其中：R1是C1-C4烷基; R2是氰基，硝基，三氟甲基，卤素，C1-C4-烷基和C1-C4-烷氧基; m是0,1或2，其中基团R2可以是 如果m是2，则R 3是氢，氰基，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 3 -C 6环烷基; R 4，R 5和R 6各自如权利要求1所定义， 描述了制备这些化合物的中间体和包含它们的用于控制动物害虫和有害真菌的组合物。

公开(公告)号：US06537989B1

公开(公告)日：2003-03-25

申请号：US09806608

申请日：2001-04-02

申请人： Markus Gewehr ,  Wassilios Grammenos ,  Hubert Sauter ,  Herbert Bayer ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries

发明人： Markus Gewehr ,  Wassilios Grammenos ,  Hubert Sauter ,  Herbert Bayer ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries

IPC分类号： A61K3155

CPC分类号： C07D273/00 ,  A01N43/88

摘要： The present invention relates to azadioxacycloalkenes of the formula I in which the substituents R1 to R5 and X, the index n and the bridge member W have the following meanings: R1 is C1-C4-alkyl, halogen, C1-C4-haloalkyl, C3-C6-cycloalkyl; R2 is C1-C4-alkyl, C1-C4-haloalkyl, C3-C4-alkenyl, C3-C4-haloalkenyl, C3-C4-alkynyl or C3-C4-haloalkynyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl or unsubstituted or substituted phenyl; R4 is ═CRaRb, —CRd═CRaRb or ═N—ORc, where Ra, Rb, Rc and Rd are each as defined in claim 1; R5 is nitro, cyano, halogen, C1-C6-alkyl or, in the case that n is 2, additionally a bridge which is attached to two adjacent ring atoms; n is 0, 1, 2, 3 or 4, where the substituents R1 may be different if n is greater than 1; X is C1-C4-alkoxy-N═, C1-C4-alkoxy-CH═ or R6—CH═, where R6 is as defined in claim 1 W is unsubstituted or substituted C1-C3-alkylene.

摘要翻译： 本发明涉及取代基R1至R5和X，指数n和桥连构件W具有以下含义的式Iin的二恶唑环烯烃：R1为C1-C4烷基，卤素，C1-C4卤代烷基，C3- C6-环烷基; R2是C1-C4-烷基，C1-C4卤代烷基，C3-C4-烯基，C3-C4-卤代烯基，C3-C4-炔基或C3-C4-卤代炔基; R3是氢，C1-C4- 烷基，C1-C4卤代烷基或未取代或取代的苯基; R4是= CRaRb，-CRd = CRaRb或= N-ORc，其中Ra，Rb，Rc和Rd分别如权利要求1中所定义; R5是硝基，氰基， 卤素，C 1 -C 6 - 烷基，或在n为2的情况下，另外是连接到两个相邻环原子上的桥; n为0,1,2,3或4，其中如果n 大于1; X为C 1 -C 4 - 烷氧基-N =，C 1 -C 4 - 烷氧基-CH =或R 6 -CH =，其中R 6如权利要求1W中所定义，为未取代或取代的C 1 -C 3 - 亚烷基。

公开(公告)号：US06200997B1

公开(公告)日：2001-03-13

申请号：US09236108

申请日：1999-01-25

申请人： Andreas Gypser ,  Hubert Sauter ,  Herbert Bayer ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Roland Götz ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Volker Harries ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Andreas Gypser ,  Hubert Sauter ,  Herbert Bayer ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Roland Götz ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Volker Harries ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： A01N4382

CPC分类号： C07D263/44 ,  A01N43/76 ,  C07D249/12

摘要： The present invention relates to heterocyclyl-substituted phenyl compounds of the formula I, where the substituents have the following meanings: Y is halogen, C1-C4-alkyl, C1-C4-haloalkyl or C1-C4-alkoxy; n is 0, 1 or 2, where the radicals Y may be different if n=2; E is a group A or B,  where # denotes the bond to the phenyl ring, and G R&agr;, R&bgr;, Y, n, T and Z are each as defined in the description.

摘要翻译： 本发明涉及式I的杂环基取代的苯基化合物，其中取代基具有以下含义：Y为卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基或C 1 -C 4 - 烷氧基; n为0,1 或2，其中如果n = 2，基团Y可以不同; E是基团A或B，其中＃表示与苯环的键，G Ralpha，Rbeta，Y，n，T和Z各自定义 在说明中。

公开(公告)号：US06372766B1

公开(公告)日：2002-04-16

申请号：US09529806

申请日：2000-04-20

申请人： Wassilios Grammenos ,  Klaus Oberdorf ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Markus Gewehr ,  Thomas Grote ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Gerhard Hamprecht ,  Norbert Götz ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Klaus Oberdorf ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Markus Gewehr ,  Thomas Grote ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Gerhard Hamprecht ,  Norbert Götz ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： A01N4340

CPC分类号： C07D213/64 ,  A01N43/40

摘要： Substituted 2-(2′-pyridyloxy)phenylacetamides I, where R1 is fluorine, chlorine, CH3 or halomethyl; R2 is fluorine, bromine, alkyl or halomethyl; R3 is hydrogen or one of the radicals mentioned under R2; and R2 is 6-chloro if R3 is hydrogen, R3 is 5-chloro if R2 is fluorine and the compound in which R1, R2 and R3 are each chlorine with the proviso that R1 may not be chlorine if R2 is 5-trifluoromethyl and R3 is hydrogen, and processes for their preparation and their use for controlling harmful fungi and animal pests are described.

摘要翻译： 取代的2-（2'-吡啶基氧基）苯基乙酰胺I，其中R 1是氟，氯，CH 3或卤代甲基; R 2是氟，溴，烷基或卤代甲基; R 3是氢或在R 2下提及的一个基团; 如果R 3为氢，R 2为6-氯，如果R 2为氟，则R 3为5-氯，并且其中R 1，R 2和R 3各自为氯的化合物，条件是如果R 2为5-三氟甲基并且R 3为氢，则R 1可不为氯， 并描述了其制备方法及其用于控制​​有害真菌和动物害虫的用途。

公开(公告)号：US06414031B1

公开(公告)日：2002-07-02

申请号：US09674533

申请日：2000-11-02

申请人： Herbert Bayer ,  Roland Götz ,  Michael Keil ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Eberhard Ammermann ,  Thomas Grote ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries

发明人： Herbert Bayer ,  Roland Götz ,  Michael Keil ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Eberhard Ammermann ,  Thomas Grote ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries

IPC分类号： A01N3718

CPC分类号： C07C251/60 ,  C07C2601/14

摘要： There are disclosed bisoxime ether derivatives of the formula I in which the variables have the following meanings: R1 is halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; n is 1 to 5, it being possible for the radicals R1 to be different if n is other than 1; R2 is C1-C4-alkyl, C3-C6-alkenyl or C3-C6-alkynyl, it being possible for these groups to be partially or fully halogenated; Q is C(═CHOCH3)—COOCH3, C(═CHCH3)—COOCH3, C(═NOCH3)—COOCH3 or C(═NOCH3)13 CONHCH3; and salts thereof, processes and intermediates for the preparation of these compounds, and their use for controlling animal pests and harmful fungi.

摘要翻译： 公开了式Iin的双肟醚衍生物，其变量具有以下含义：R 1是卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 卤代烷氧基; n是1至 5，如果n不是1，则基团R1可能是不同的; R2是C1-C4-烷基，C3-C6-烯基或C3-C6-炔基，这些基团可能是部分或完全的 卤素; Q是（C 1 -C 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C（= NOCH 3）-COOCH 3或C（= NOCH 3）13 CONHCH 3;及其盐，用于制备这些化合物的方法和中间体， 及其用于控制​​动物害虫和有害真菌的用途。

公开(公告)号：US06232317B1

公开(公告)日：2001-05-15

申请号：US09463435

申请日：2000-01-27

申请人： Wassilios Grammenos ,  Herbert Bayer ,  Hubert Sauter ,  Thomas Grote ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Norbert Götz ,  Eberhard Ammermann ,  Volker Harries ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Herbert Bayer ,  Hubert Sauter ,  Thomas Grote ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Norbert Götz ,  Eberhard Ammermann ,  Volker Harries ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： A01N43653

CPC分类号： A01N43/80 ,  A01N43/653 ,  C07D249/12

摘要： Imino-substituted phenyl compounds of the formula I where the substituents have the following meanings: z is a group A or B  where  # denotes the bond with the phenyl ring and  Ra is halogen, alkyl or alkoxy; y is halogen, alkyl, haloalkyl or alkoxy; n is 0, 1 or 2, it being possible for the radicals Y to be different if n=2; R1 is halogen, haloalkyl or alkoxy; R2 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl; R3 is cyano, alkyl, haloalkyl, alkoxy, cycloalkoxy, alkoxyalkyl;  unsubstituted or substituted cycloalkyl, aryl, aryloxy or arylmethylene, heteroaryl, heterocyclyl,  C(R3a)═N—OR3b or C(R3a)═CR3cR3d, where R3a, R3b, R3c, R3d independently of one another are hydrogen, alkyl or unsubstituted or substituted phenyl, processes for their preparation, and their use.

摘要翻译： 取代基具有以下含义：Z是A或B基团，其中＃表示与苯环的键，Ra是卤素，烷基或烷氧基; y是卤素，烷基，卤代烷基或烷氧基 n为0,1或2，如果n = 2，则基团Y可能不同; R1为卤素，卤代烷基或烷氧基; R2为烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基; R3为氰基， 烷基，卤代烷基，烷氧基，环烷氧基，烷氧基烷基; 未取代或取代的环烷基，芳基，芳氧基或芳基亚甲基，杂芳基，杂环基，C（R3a）= N-OR3b或C（R3a）= CR3cR3d，其中R3a，R3b，R3c，R3d彼此独立地为氢，烷基或未取代或取代的 苯基，其制备方法及其用途。