公开(公告)号：US20070129380A1

公开(公告)日：2007-06-07

申请号：US10565656

申请日：2004-07-03

申请人： Frank Schieweck ,  Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Scholf ,  Maria Scherer ,  Reinhard Stierl

发明人： Frank Schieweck ,  Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Scholf ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/505 ,  C07D239/42

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and these substituents R1, R2 and R3 are as defined in the description and R4 is as defined below: R4 corresponds to one of the formulae where Ra is hydrogen, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C3-C6-cycloalkyl or C1-C4-alkoxy and R5 is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C4-alkyloxy-C1-C2-alkyl, phenyl-C1-C2-alkyl or phenyloxy-C1-C2-alkyl, to processes for preparing these compounds, to compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和这些取代基R 1，R 2和R 3是 如在说明书中所定义的，R 4是如下定义的：R 4对应于下式之一其中R a a是氢，C 1〜 C 1 -C 6烷基，C 2 -C 8 - 烯基，C 2 - 亚烷基，C 2 -C 6 - C 1 -C 8 - 炔基，C 3 -C 6 - 环烷基或C 1 -C 6 - 4 - 烷氧基和R 5是氢，C 1 -C 6 - 烷基，C 2〜 C 1 -C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 6 - 4 - 烷氧基-C 1 -C 2 - 烷基，苯基-C 1 -C 2 - 亚烷基 烷基或苯氧基-C 1 -C 2 - 烷基，用于制备这些化合物的方法，包含这些化合物的组合物及其作为农药的用途。

公开(公告)号：US20060058326A1

公开(公告)日：2006-03-16

申请号：US10541386

申请日：2004-01-28

申请人： Bernd Muller ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Tormo I Blasco ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Bernd Muller ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Tormo I Blasco ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/513

CPC分类号： C07D239/56 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/653 ,  A01N43/707 ,  A01N43/78 ,  A01N43/82 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04

摘要： Pyrimidines of the formula I in which Ln is as defined in the description and the substituents R1, R2 and R3 are as defined below: R1 is C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl, phenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S; R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl; R3 is a five- or six-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S; and processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的嘧啶

公开(公告)号：US20070054929A1

公开(公告)日：2007-03-08

申请号：US10555894

申请日：2004-05-10

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/506 ,  C07D403/04

CPC分类号： C07D239/48 ,  A01N43/56 ,  C07D403/04

摘要： The present invention relates to pyrimidines of the formula I in which the index n and the substituents L, R1-R3 are as defined in the description and R4 corresponds to one of the formulae and to processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的嘧啶，其中指数n和取代基L，R 1〜R 3如说明书中所定义， 4对应于一个公式，以及制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060211711A1

公开(公告)日：2006-09-21

申请号：US10550571

申请日：2004-03-30

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR2, cyano, S(O)nA1 or C(O)A2; R=alkyl or alkylcarbonyl, A1=hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A2=alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R1=hydrogen or alkyl; R2=alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-烷基氨基 - 三唑并嘧啶类，其中取代基具有以下含义：L =卤素，烷基，卤代烷基，烷氧基，氨基，NHR，NR 2，氰基，S（O） 或者C（O）A 2 O 2。 R =烷基或烷基羰基，A 1〜H 2，羟基，烷基，烷基氨基或亚烷基氨基; n = 0,1或2; 链烯基，烷氧基，卤代烷氧基或A 1中引用的基团之一; m = 1,2,3,4或5，其中至少一个基团L存在于与三唑并嘧啶骨架的键的邻位; X =卤素，氰基，烷基，卤代烷基或烷氧基; R 1 =氢或烷基; R 2 =炔基，其可以是未取代的或根据描述取代的。 本发明还涉及生产所述化合物的方法，含有所述化合物的试剂及其用于对抗有害植物病原真菌的用途。

公开(公告)号：US06919485B2

公开(公告)日：2005-07-19

申请号：US10469688

申请日：2002-03-09

申请人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Norbert Götz ,  Karl Eicken ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Norbert Götz ,  Karl Eicken ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N35/04 ,  C07C45/46 ,  C07C49/84 ,  C07C45/00 ,  A01N35/00

CPC分类号： C07C49/84 ,  A01N35/04 ,  C07C45/46

摘要： The invention relates to benzophenones of formula (I), in which the substituents have the following meanings: X represents halogen; R1 represents hydrogen, halogen, C1-C6 alkyl, halo-C1-C2 alkyl, C1-C4 alkoxy, oxyhalomethyl or nitro, and; R2 represents hydrogen, C1-C6 alkyl, benzyl, cyclohexylmethyl or C3-C6 alkenyl. The invention also relates to the production of these benzophenones and to their use as fungicides

摘要翻译： 本发明涉及式（I）的二苯甲酮，其中取代基具有以下含义：X表示卤素; R 1表示氢，卤素，C 1 -C 6烷基，卤代C 1 -C 3 烷基，C 1 -C 4烷氧基，氧卤甲基或硝基，和; R 2表示氢，C 1 -C 6烷基，苄基，环己基甲基或C 3 -C 3 > 6个烯基。 本发明还涉及这些二苯甲酮的制备及其作为杀真菌剂的用途

公开(公告)号：US20080221177A1

公开(公告)日：2008-09-11

申请号：US12101175

申请日：2008-04-11

申请人： Wassilios GRAMMENOS ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Wassilios GRAMMENOS ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/40 ,  A01P3/00

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2′ and R3′, R2′, R3′ are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， '和R 3'，R 2'，R 3'是氢，卤素，烷基，烷氧基或卤代甲基; 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 被C（R 6） - - NOR 7取代的苯基，其中R 6是烷基，R 7是 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070135453A1

公开(公告)日：2007-06-14

申请号：US10579395

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; L1, L2, L3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的6-（2,4,6-三卤代苯基）三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基， 卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2 R 1是氢或R 1，R 2和R 2中所提及的基团之一，与它们的氮原子一起 还可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个其它由O，N和S组成的组的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; L 1，L 2，L 3 3是氯或氟，其中至少一个基团是氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050107619A1

公开(公告)日：2005-05-19

申请号：US10507605

申请日：2003-03-12

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07B61/00 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C233/73

CPC分类号： C07C235/34 ,  A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C233/22 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14

摘要： Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X=H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R1=alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R2=H, alkyl, haloalkyl, allyl, propargyl or CH2C≡C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests.

摘要翻译： 式（I）的Z-取代的丙烯酰胺，其中取代基具有以下含义：X = H，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，其中X为3-或4-位，n = 1或2，其中 如果n = 2，则X可以不同，R 1 =烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，氮丙啶和环氧乙烷，R 2 = H，烷基，卤代烷基，烯丙基 炔丙基或CH 2C≡C-烷基。 其制备方法，包含上述物质及其用于治疗植物致病性真菌害虫的用途。

公开(公告)号：US20050181948A1

公开(公告)日：2005-08-18

申请号：US10509112

申请日：2003-03-27

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： C07D213/56 ,  C07D213/61 ,  C07D263/10 ,  A01N43/60 ,  A01N43/40 ,  A01N43/54

CPC分类号： C07D263/10 ,  C07D213/56 ,  C07D213/61

摘要： The present invention relates to novel phenethylacrylamides of the formula I in which the substituents R1, R2, R3 and R4 have the following meanings: R1 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C3-C8-cycloalkyl, C1-C4-haloalkoxy or C1-C4-haloalkyl; R2 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C3-C10-cycloalkyl, C1-C4-haloalkoxy or C1-C4-haloalkyl; R3 is C1-C4-alkyl, C1-C4-haloalkyl, propargyl, C3-C4-alkenyl or a radical of the formula —H2C—C≡C—C(Ra, Ra)—Rc, wherein Ra, Rb independently of one another are hydrogen or methyl and Rc is hydrogen or C1-C4-alkyl; R4 is methyl or C1-haloalkyl; and Het is a 5- or 6-membered heteroaromatic ring, to processes for their preparation, and to the use of phenethylacrylamides of the formula I for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的新的苯乙基丙烯酰胺，其中取代基R 1，R 2，R 3和R 4 具有以下含义：R 1是氢，卤素，C 1 -C 4 - 烷基，C 1 C 1 -C 4 - 烷氧基，C 3 -C 8 - 环烷基，C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷基; R 2是氢，卤素，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 烷氧基，C 3 -C 10 - 环烷基，C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷基; R 3是C 1 -C 4 - 烷基，C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4 - 烷基，炔丙基，C 3 -C 4 - 烯基或式-H 2C≡CC（R 0）的基团 其中R a，R b，R b独立地为C 1 -C 4，其中R a，R b， 另一个是氢或甲基，R c是氢或C 1 -C 4 - 烷基; R 4是甲基或C 1 - 卤代烷基; 并且Het是5或6元杂芳环，用于其制备方法，以及使用式I的苯乙基丙烯酰胺来控制植物病原性有害真菌。

公开(公告)号：US20060079537A1

公开(公告)日：2006-04-13

申请号：US10531898

申请日：2003-11-14

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(═O)-A or S(═O)pA′; A and A′ are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR1R2 or S(O)nR31, where n and R31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，-C（ - O） - 取代的取代基如下： -A或S（-O） A'; A和A'如说明书所定义; p为0,1或2; m为0,1,2,3,4或5; X是氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 - 至十元饱和的，部分不饱和的或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1和R 2连同 它们所连接的氮原子也可以形成可被来自O，N和S的原子间隔的五元或六元环，其中R 1和/或 R 2可以如说明书中定义的取代; 和R 3是氰基，羟基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，NR 1 R 2或S（O）n 其中n和R 31如在说明书中所定义的; 描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。