2- (2-pyridyl) -5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi
    52.
    发明申请
    2- (2-pyridyl) -5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi 失效
    2-(2-吡啶基)-5-苯基-6-氨基嘧啶,用于生产和用于对抗有害真菌的方法和中间产物

    公开(公告)号:US20050107401A1

    公开(公告)日:2005-05-19

    申请号:US10505146

    申请日:2003-02-06

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(2-pyridyl)-5-phenyl-6-amninopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

    摘要翻译: 本发明涉及式I的2-(2-吡啶基)-5-苯基-6-脒嘧啶,其中取代基和指数具有以下含义:R 1表示卤素,羟基,杂环基, 烷氧基,烷氧基羰基,氨基甲酰基,烷基氨基羰基,二烷基氨基羰基,吗啉代羰基,吡咯烷基羰基,烷基羰基氨基,烷基氨基。 二烷基氨基,烷硫基,烷基亚磺酰基,烷基磺酰基,羟基磺酰基,氨基磺酰基,烷基氨基磺酰基,二烷基氨基磺酰基; m = 0或1-4; R 2表示氢,卤素,氰基,烷基,卤代烷基或烷氧基; R 3,R 4表示氢,烷基,卤代烷基,环烷基,卤代烷基,烯基,卤代烯基,环烯基,炔基,卤代炔基或环炔基,R 3 O 和R 4与它们连接的氮原子一起形成5或6元环,其被来自基团O,N或S的原子和/或可被取代 根据说明; R 5表示卤素,烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7,R 8表示氢,卤素,烷基或卤代烷基; R 9表示氢,卤素,羟基,氰基,烷基,烷氧基,环烷氧基,卤代烷氧基,烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物,除了其用于对抗不期望的植物之外。

    5-Halogen-6-phenyl-7-fluoroalkylamino-triazolopyrimidines as fungicides
    55.
    发明授权
    5-Halogen-6-phenyl-7-fluoroalkylamino-triazolopyrimidines as fungicides 失效
    作为杀真菌剂的5-卤代-6-苯基-7-氟烷基氨基 - 三唑并嘧啶

    公开(公告)号:US07105664B2

    公开(公告)日:2006-09-12

    申请号:US10474460

    申请日:2002-04-06

    IPC分类号: C07D487/04 A01N43/90

    CPC分类号: C07D487/04

    摘要: 5-Halogen-6-phenyl-7-fluoroalkylamino-triazolopyrimidines of formula I: (I) in which R1 is hydrogen, fluoro, alkyl, alkenyl, alkynyl, alkadienyl, where the carbon chains of these radicals may be unsubstituted or substituted as defined in the description; R2 is hydrogen, alkyl, alkenyl, alkynyl, alkadienyl, where these radicals may be unsubstituted or substituted; R3 is fluoroalkyl or fluoroalkenyl; X is halogen; n is 0 or an integer from 1 to 4; L each independently is halogen, nitro, alkyl, haloalkyl, alkoxy or haloalkoxy. Processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

    摘要翻译: 式I的5-卤代-6-苯基-7-氟烷基氨基 - 三唑并嘧啶:其中R 1是氢,氟,烷基,烯基,炔基,链二烯基,其中这些的碳链 基团可以是未取代的或如说明书中所定义的取代基; R 2是氢,烷基,烯基,炔基,链二烯基,其中这些基团可以是未取代的或取代的; R 3是氟代烷基或氟代烯基; X是卤素; n为0或1至4的整数; L各自独立地为卤素,硝基,烷基,卤代烷基,烷氧基或卤代烷氧基。 其制备方法,含有它们的组合物及其用于对抗植物病原真菌的用途。