2-(2-imidazolin-2-ylthio)-acetanilides
    52.
    发明授权
    2-(2-imidazolin-2-ylthio)-acetanilides 失效
    2-(2-咪唑烷-2-基) - 乙酰胺

    公开(公告)号:US3711505A

    公开(公告)日:1973-01-16

    申请号:US3711505D

    申请日:1971-01-25

    申请人: WANDER AG DR A

    发明人: BREAM J PICARD C READ D

    CPC分类号: C07D233/84 C07D233/42

    摘要: THE INVENTION CONCERNS A COMPOUND OF THE FORMULA

    2-((R1,R2-PHENYL)-NH-CO-CH2-S-),4-R3,5-R4-IMIDAZOLINE

    WHEREIN R1 AND R2 ARE EACH HYDROGEN, HALOGEN OR ALKYL OF 1 TO 3 CARBON ATOMS, AND EITHER EACH OF R3 AND R4 IS HYDROGEN, OR ONE OF R3 AND R4 IS ALKYL OF 1 TO 3 CARBON ATOMS OE HYDROXY AND THE OTHER IS HYDROGEN, OR A PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALT THEREOF.

    Process for 5 h-imidazo(2,1-a)isoindoles
    54.
    发明授权
    Process for 5 h-imidazo(2,1-a)isoindoles 失效
    5 H-IMIDAZO(2,1-A)ISOINDOLES的方法

    公开(公告)号:US3699119A

    公开(公告)日:1972-10-17

    申请号:US3699119D

    申请日:1971-02-16

    申请人: SANDOZ AG

    IPC分类号: C07D209/46 C07D49/34

    CPC分类号: C07D209/46

    摘要: PROCESS FOR PREPARING 5-HYDROXY-5-ARYL-2,3-DIHYDRO5H-IMIDAZO(2,1-A)ISOINDOLES, E.G., 5-(P-CHLOROPHENYL)-5HYDROXY-2,3-DIHYDRO-5H-IMIDAZO(2,1-A)ISOINDOLE. AN APPROPARIATELY SUBSTITUTED 3-ARYL PHTHALIMIDINE IS TREATED WITH TRIETHYLOXONIUM BORONETRAFLUORIDE TO PROVIDE AN INTERMEDIATE 3-ETHOXY-1H-ISOINDOLE WHICH IS CONVERTED TO THE FINAL PRODUCT BY TREATMENT WITH ETHYLENEIMINE HYDROTETRAFLUOROBORATE AND CONTACTING THE RESULTING PRODUCT WITH AIR OR OXYGEN. THESE COMPOUNDS ARE USEFUL AS PSYCHIC ENERGIZERS AND ANORETICS.

    2-carbamyl-2-imidazolines and method for their production
    55.
    发明授权
    2-carbamyl-2-imidazolines and method for their production 失效
    2-卡马来-2-咪唑啉及其生产方法

    公开(公告)号:US3681379A

    公开(公告)日:1972-08-01

    申请号:US3681379D

    申请日:1970-04-22

    申请人: BASF AG

    CPC分类号: C07D233/28 D06M13/35

    摘要: Production of 2-carbamyl-2-imidazolines by reacting haloacetamides with 1,2-alkylene diamines and elementary sulfur, and the 2-carbamyl-2-imidazolines. The new compounds are auxiliaries for the textile and leather industries, plant protection agents and valuable starting material for the manufacture of textile and leather auxiliaries and plant protection agents.

    摘要翻译: 卤代乙酰胺与1,2-亚烷基二胺和元素硫反应生成2-氨基甲酰基-2-咪唑啉,2-氨基甲酰基-2-咪唑啉。

    2-(substituted benzyl)methyl-2-imidazolines
    57.
    发明授权
    2-(substituted benzyl)methyl-2-imidazolines 失效
    2-(取代苄基)甲基-2-咪唑烷

    公开(公告)号:US3660423A

    公开(公告)日:1972-05-02

    申请号:US3660423D

    申请日:1970-02-13

    申请人: DOW CHEMICAL CO

    IPC分类号: C07D233/24 C07D49/34

    CPC分类号: C07D233/24

    摘要: 2 - (SUBSTITUTED BENZYL) - 2 - IMIDAZOLINE COMPOUNDS SUCH AS 2-(4-AMINO-3-CHLOROBENZYL)-2-IMIDAZOLINE, AND THEIR PHARMACEUTICALLY-ACCEPTABLE SALTS SUCH AS THE MONOAND DIHYDROCHLORIDES ARE PREPARED BY CLASSICAL PROCEDURES. THE COMPOUNDS ARE ACTIVE AS ANTIDEPRESSANTS.