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公开(公告)号:US06645915B1
公开(公告)日:2003-11-11
申请号:US09856887
申请日:2001-07-13
申请人: Hans-Jochem Riebel , Akihiko Yanagi , Yukiyoshi Watanabe , Toshio Goto , Kristian Kather , Stefan Lehr , Katharina Voigt , Mark Wilhelm Drewes , Peter Dahmen , Dieter Feucht , Rolf Pontzen
发明人: Hans-Jochem Riebel , Akihiko Yanagi , Yukiyoshi Watanabe , Toshio Goto , Kristian Kather , Stefan Lehr , Katharina Voigt , Mark Wilhelm Drewes , Peter Dahmen , Dieter Feucht , Rolf Pontzen
IPC分类号: C07D25118
CPC分类号: C07D251/18
摘要: The invention relates to novel substituted 1,3,5-triazines of the general formula (I) in which A represents CHR3R4 or represents C1-halogenoalkyl-substituted C3-C6-cycloalkyl, C3-C6-alkinyl or C1-C4-cyanoalkyl, where R1, R2, R3 and R4 are each as defined in the description, and to processes for their preparation, to novel intermediates, including their preparation, and to the use of the compounds of the general formula (I) as herbicides.
摘要翻译: 本发明涉及通式(I)的新的取代的1,3,5-三嗪,其中A表示CHR 3 R 4或表示C 1 - 卤代烷基取代的C 3 -C 6 - 环烷基,C 3 -C 6 - 炔基或 C 1 -C 4 - 氰基烷基,其中R 1,R 2,R 3和R 4各自如说明书中所定义,并且其制备方法,新颖的中间体,包括它们的制备,以及 使用通式(I)的化合物作为除草剂。
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公开(公告)号:US06440903B1
公开(公告)日:2002-08-27
申请号:US09269820
申请日:1999-04-01
申请人: Hans-Jochem Riebel , Stefan Lehr , Uwe Stelzer , Yukiyoshi Watanabe , Markus Dollinger , Seishi Ito , Toshio Goto , Akihiko Yanagi
发明人: Hans-Jochem Riebel , Stefan Lehr , Uwe Stelzer , Yukiyoshi Watanabe , Markus Dollinger , Seishi Ito , Toshio Goto , Akihiko Yanagi
IPC分类号: C07D25148
CPC分类号: A01N43/68 , A01N43/70 , C07C279/26 , C07C311/64 , C07C323/44 , C07D251/18 , C07D251/50 , C07D251/52
摘要: The invention relates to novel substituted 2,4-diamino-1,3,5-triazines of the formula (I) (in which R1, R2, R3, X and Z are each as described in the description), to processes and to novel intermediates for their preparation and to their use as herbicides.
摘要翻译: 本发明涉及式(I)的新型取代的2,4-二氨基-1,3,5-三嗪(其中R1,R2,R3,X和Z各自如说明书所述),以处理和 新型中间体用于制备和用作除草剂。
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公开(公告)号:US5710278A
公开(公告)日:1998-01-20
申请号:US802152
申请日:1997-02-19
申请人: Toshio Goto , Koichi Moriya , Fritz Maurer , Seishi Ito , Katsuaki Wada , Kazuhiro Ukawa , Ryo Watanabe , Asami Ito
发明人: Toshio Goto , Koichi Moriya , Fritz Maurer , Seishi Ito , Katsuaki Wada , Kazuhiro Ukawa , Ryo Watanabe , Asami Ito
IPC分类号: A01N47/38 , C07D401/04 , C07D401/14
CPC分类号: C07D401/04 , A01N47/38
摘要: Herbicidal tetrazolinone derivatives of the formula: ##STR1## in which R.sup.1 is alkyl, haloalkyl, cycloalkyl, alkenyl, haloalkenyl, alkynyl or phenyl, and R.sup.2 is alkyl, haloalkyl, cycloalkyl, alkenyl, haloalkenyl, alkynyl or phenyl, or R.sup.1 and R.sup.2 together with the nitrogen atom to which they are bonded form an optionally benzofused heterocyclic ring, which is optionally substituted by C.sub.1-4 alkyl, n is 0, 1, 2 or 3, and R.sup.3 each independently is nitro, halogen, alkyl, haloalkyl, alkylthio or phenoxy.
摘要翻译: 式中:R 1为烷基,卤代烷基,环烷基,烯基,卤代烯基,炔基或苯基,R 2为烷基,卤代烷基,环烷基,链烯基,卤代烯基,炔基或苯基,或R 1和R 2一起形成的除草四氢唑酮衍生物 与其键合的氮原子形成任选的苯并稠合的杂环,其任选被C 1-4烷基取代,n是0,1,2或3,并且R 3各自独立地是硝基,卤素,烷基,卤代烷基,烷硫基 或苯氧基。
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公开(公告)号:US5650374A
公开(公告)日:1997-07-22
申请号:US553160
申请日:1995-11-07
申请人: Toshio Goto , Yoshinori Kitagawa , Seishi Ito , Katsuhiko Shibuya , Kazuhiro Ukawa , Yoshiko Kyo
发明人: Toshio Goto , Yoshinori Kitagawa , Seishi Ito , Katsuhiko Shibuya , Kazuhiro Ukawa , Yoshiko Kyo
IPC分类号: C07D401/06 , A01N47/38 , C07D257/04 , C07D403/06 , C07D405/12 , A01N43/713 , A01N43/72
CPC分类号: C07D257/04 , A01N47/38
摘要: Herbicidal 1-cyclopropyl tetrazolinones of the formula ##STR1## wherein X represents C.sub.1-3 alkyl, C.sub.2-4 alkenyl or halogen,n represents 0 to 5,R.sup.1 and R.sup.2 each independently represents C.sub.1-6 alkyl, C.sub.2-6 alkenyl, C.sub.2-6 alkynyl, C.sub.3-7 cycloalkyl which may optionally be substituted by C.sub.1-3 alkyl, epoxy-C.sub.3-5 alkan-1-yl, phenyl which may optionally be substituted, or aralkyl which may optionally be substituted, orR.sup.1 and R.sup.2 together with the N-atom to which they are attached, represent a cyclic ring which may be substituted, and some novel intermediates therefor.
摘要翻译: 式(I)的除草1-环丙基四唑啉酮其中X代表C1-3烷基,C2-4烯基或卤素,n代表0-5,R1和R2各自独立地表示C1-6烷基,C2-6烯基 C 2-6炔基,可任选被C 1-3烷基取代的C 3-7环烷基,环烷基-C 3-5烷基-1-基,可任意被取代的苯基或可任意被取代的芳烷基,或R 1和 R2与它们所连接的N-原子一起表示可以被取代的环状环,以及一些新的中间体。
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公开(公告)号:US5641727A
公开(公告)日:1997-06-24
申请号:US498736
申请日:1995-07-06
申请人: Toshio Goto , Koichi Moriya , Fritz Maurer , Seishi Ito , Katsuaki Wada , Kazuhiro Ukawa , Ryo Watanabe , Asami Ito
发明人: Toshio Goto , Koichi Moriya , Fritz Maurer , Seishi Ito , Katsuaki Wada , Kazuhiro Ukawa , Ryo Watanabe , Asami Ito
IPC分类号: A01N47/38 , C07D401/04 , C07D401/14 , A01N43/40
CPC分类号: C07D401/04 , A01N47/38
摘要: Herbicidal tetrazolinone derivatives of the formula: ##STR1## in which R.sup.1 is alkyl, haloalkyl, cycloalkyl, alkenyl, haloalkenyl, alkynyl or phenyl, andR.sup.2 is alkyl, haloalkyl, cycloalkyl, alkenyl, haloalkenyl, alkynyl or phenyl, orR.sup.1 and R.sup.2 together with the nitrogen atom to which they are bonded form an optionally benzofused heterocyclic ring, which is optionally substituted by C.sub.1-4 alkyl,n is 0, 1, 2 or 3, andR.sup.3 each independently is nitro, halogen, alkyl, haloalkyl, alkylthio or phenoxy.
摘要翻译: 式中:R 1为烷基,卤代烷基,环烷基,烯基,卤代烯基,炔基或苯基,R 2为烷基,卤代烷基,环烷基,链烯基,卤代烯基,炔基或苯基,或R 1和R 2一起形成的除草四氢唑酮衍生物 与其键合的氮原子形成任选的苯并稠合的杂环,其任选被C 1-4烷基取代,n是0,1,2或3,并且R 3各自独立地是硝基,卤素,烷基,卤代烷基,烷硫基 或苯氧基。
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公开(公告)号:US5342938A
公开(公告)日:1994-08-30
申请号:US14022
申请日:1993-02-05
申请人: Toyohiko Kume , Toshio Goto , Atsumi Kamochi , Hidenori Hayakawa , Akihiko Yanagi , Tadao Asami
发明人: Toyohiko Kume , Toshio Goto , Atsumi Kamochi , Hidenori Hayakawa , Akihiko Yanagi , Tadao Asami
IPC分类号: A01N43/84 , C07D265/36 , C07D413/04
CPC分类号: C07D413/04 , A01N43/84 , C07D265/36
摘要: Novel benzoxazines of the formula (I) ##STR1## the use of the new compounds as herbicides, and novel compounds of the formula (IX) as intermediates ##STR2## are disclosed.
摘要翻译: 式(I)的新型苯并恶嗪(I)新化合物作为除草剂的使用,以及作为中间体(IX)的式(IX)的新化合物。
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公开(公告)号:US5296454A
公开(公告)日:1994-03-22
申请号:US905944
申请日:1992-06-26
申请人: Toshio Goto , Hidenori Hayakawa , Itsuko Manabe , Akihiko Yanagi
发明人: Toshio Goto , Hidenori Hayakawa , Itsuko Manabe , Akihiko Yanagi
IPC分类号: A01N31/04 , A01N37/22 , A01N43/08 , A01N43/10 , C07C233/15 , C07C233/29 , C07C321/28 , C07C323/41 , C07D307/54 , C07D333/24
CPC分类号: C07C233/29 , A01N37/22 , A01N43/08 , A01N43/10 , C07C233/15 , C07C323/41 , C07D307/54 , C07D333/24
摘要: The invention relates to novel acetanilides of the formula (I) ##STR1## wherein Ar represents phenyl, furyl or thienyl,R.sup.1 represents hydrogen, C.sub.1-5 -alkyl, C.sub.3-6 -cycloalkyl, C.sub.3-6 -cycloalkyl-methyl, C.sub.3-5 alkenyl, C.sub.3-5 -alkynyl, C.sub.1-3 -haloalkyl, C.sub.3-5 -epoxyalkyl, C.sub.1-3 -alkoxy-C.sub.1-4 -alkyl, C.sub.1-3 -alkylthio-C.sub.1-4 -alkyl, C.sub.1-3 -alkoxycarbonyl-C.sub.1-2 -alkyl, cyano-C.sub.1-3 -alkyl, or aralkylR.sup.2 represents hydrogen or C.sub.1-3 -alkyl,R.sup.3 represents hydrogen or C.sub.1-3 -alkyl,X represents halogen, andY represents iso-propyl, tert-butyl, C.sub.1-2 -haloalkyl, C.sub.1-2 -haloalkoxy, C.sub.1-2 -haloalkylthio or C.sub.1-2 -alkylsulfonyl,to processes for their preparation and to their use as herbicides. The invention also relates to novel intermediates and to processes for their preparation.
摘要翻译: 本发明涉及式(I)的新型乙酰苯胺(*化学结构*)(I)其中Ar表示苯基,呋喃基或噻吩基,R1表示氢,C1-5烷基,C3-6环烷基,C3-6- 环烷基 - 甲基,C3-5烯基,C3-5-炔基,C1-3-卤代烷基,C3-5-环氧烷基,C1-3-烷氧基-C1-4-烷基,C1-3-烷硫基-C1-4-烷基 ,C 1-3 - 烷氧基羰基-C 1-2 - 烷基,氰基-C 1-3 - 烷基或芳烷基R 2表示氢或C 1-3 - 烷基,R 3表示氢或C 1-3 - 烷基,X表示卤素,Y表示 异丙基,叔丁基,C 1-2 - 卤代烷基,C 1-2 - 卤代烷氧基,C 1-2 - 卤代烷硫基或C 1-2 - 烷基磺酰基,用于其制备及其作为除草剂的用途。 本发明还涉及新型中间体及其制备方法。
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公开(公告)号:US5266692A
公开(公告)日:1993-11-30
申请号:US900463
申请日:1992-06-18
申请人: Masakuni Okuhara , Hirokazu Tanaka , Toshio Goto , Tohru Kino , Hiroshi Hatanaka
发明人: Masakuni Okuhara , Hirokazu Tanaka , Toshio Goto , Tohru Kino , Hiroshi Hatanaka
IPC分类号: C07D498/18 , C07H19/01 , C12P17/18 , C12P19/44 , C07D498/16 , A61K31/395 , A61K31/695 , C07F7/04
CPC分类号: C07D498/18 , C07H19/01 , C12P17/188 , C12P19/44 , C12R1/465 , C12R1/55
摘要: This invention relates to tricyclo compounds useful for treatment and prevention of resistance by transplantation, graft-versus-host diseases by medulla ossium transplantation, autoimmune diseases, infectious diseases, and the like, which can be represented by the following formula: ##STR1## to a process for their production, to a pharmaceutical composition containing the same and to a use thereof.
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公开(公告)号:US5077401A
公开(公告)日:1991-12-31
申请号:US418001
申请日:1989-10-06
申请人: Toyohiko Kume , Toshio Goto , Atsumi Kamochi , Akihiko Yanagi , Shigeki Yagi , Hiroshi Miyauchi , Katsuhiko Shibuya
发明人: Toyohiko Kume , Toshio Goto , Atsumi Kamochi , Akihiko Yanagi , Shigeki Yagi , Hiroshi Miyauchi , Katsuhiko Shibuya
IPC分类号: A01N43/74 , A01N43/80 , A01N43/82 , A01N43/84 , A01N43/90 , C07D263/58 , C07D265/36 , C07D277/68 , C07D413/06 , C07D413/14 , C07D417/04 , C07D417/06 , C07D417/14 , C07D471/04 , C07D487/04
CPC分类号: C07D263/58 , A01N43/74 , A01N43/80 , A01N43/82 , A01N43/84 , A01N43/90 , C07D265/36 , C07D277/68 , C07D413/06 , C07D413/14 , C07D417/04 , C07D417/06 , C07D417/14 , C07D471/04 , C07D487/04
摘要: Herbicidal benzo-fused cyclic compounds of the formula ##STR1## wherein Q is ##STR2## Y is O or S, W is ##STR3## T is O, S, --NH-- or ##STR4## and R.sup.4 may represent, together with T, chlorine,Z is O or S,X is hydrogen or halogen,n is 0 or 1 andR is C.sub.3-6 cycloalkyl, and optionally substituted 5-membered heterocyclic group or an optionally substituted 6-membered heteroaromatic group which contains one to three nitrogen atoms,and salts thereof.
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公开(公告)号:US5017213A
公开(公告)日:1991-05-21
申请号:US376719
申请日:1989-07-07
申请人: Toyohiko Kume , Toshio Goto , Atsumi Kamochi , Akihiko Yanagi , Hiroshi Miyauchi , Tadao Asami
发明人: Toyohiko Kume , Toshio Goto , Atsumi Kamochi , Akihiko Yanagi , Hiroshi Miyauchi , Tadao Asami
IPC分类号: A01N43/36 , A01N43/38 , A01N43/40 , A01N43/60 , A01N43/653 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/82 , A01N43/824 , A01N43/832 , A01N43/836 , C07D207/32 , C07D207/325 , C07D209/44 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12 , C07D521/00 , C07F7/08
CPC分类号: C07D207/325 , A01N43/36 , A01N43/38 , A01N43/40 , A01N43/80 , A01N43/82 , C07D209/44 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12
摘要: Herbicidal 1-phenylpyrroles of the formula ##STR1## wherein each R.sup.1 represents methyl or together form a tetramethylene group,R.sup.2 represents hydrogen, C.sub.1-6 alkyl, cyclopropylmethyl, C.sub.1-4 alkoxy-C.sub.1-2 alkyl, C.sub.1-4 alkylthio-C.sub.1-2 alkyl, C.sub.1-4 alkylsulfinyl-C.sub.1-2 alkyl, C.sub.1-4 alkylsulfonyl-C.sub.1-2 alkyl, benzyl or phenylethyl which are optionally substituted by halogen, C.sub.3-4 alkenyl, C.sub.3-4 alkynyl, C.sub.3-4 haloalkenyl, C.sub.2-3 cyanoalkyl or carbmoylmethyl, thiocarbamoylmethyl, trimethylsilylmethyl, CH.sub.2 COOR.sup.3, ##STR2## or a C.sub.1-2 alkyl group which is connected with an optionally substituted 5-6 membered heterocyclic group, whereinR.sup.3 represents C.sub.1-6 alkyl or C.sub.5-6 cycloalkyl,R.sup.4 represents hydrogen, methyl, ethyl or cyclopropyl,R.sup.5 represents OR.sup.6 or N(CH.sub.3).sub.2, in whichR.sup.6 represents hydrogen, C.sub.1-5 alkyl, allyl, propargyl or benzyl, andn represents 0 to 1.
摘要翻译: 式(I)的除草性1-苯基吡咯,其中每个R 1表示甲基或一起形成四亚甲基,R 2表示氢,C 1-6烷基,环丙基甲基,C 1-4烷氧基-C 1-2烷基,C 1-4烷硫基 C 1-4烷基,C 1-4烷基亚磺酰基-C 1-2烷基,C 1-4烷基磺酰基-C 1-2烷基,任选被卤素取代的苄基或苯基乙基,C 3-4链烯基,C 3-4炔基,C 3-4卤代烯基 ,C2-3氰基烷基或甲酰甲基,硫代氨基甲酰甲基,三甲基甲硅烷基甲基,CH2COOR3,或与任选取代的5-6元杂环基连接的C 1-2烷基,其中R 3表示C 1-6烷基或C 5-6环烷基 ,R 4表示氢,甲基,乙基或环丙基,R 5表示OR 6或N(CH 3)2,其中R 6表示氢,C 1-5烷基,烯丙基,炔丙基或苄基,n表示0至1。
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