Herbicidal 1-substituted methyl-tetrazolinones
    1.
    发明授权
    Herbicidal 1-substituted methyl-tetrazolinones 失效
    除草剂1-取代的甲基 - 四唑啉酮

    公开(公告)号:US06262275B1

    公开(公告)日:2001-07-17

    申请号:US09368475

    申请日:1999-08-04

    IPC分类号: C07D41306

    CPC分类号: C07D257/04 A01N47/38

    摘要: Novel 1-substituted methyltetrazolinones of the formula (I) wherein R1 represents a 5-membered heterocyclic radical which has 1 to 3 heteroatoms selected arbitrarily from the group consisting of N, O and S and which is optionally substituted by halogen and/or C1-4 alkyl, or represents oxiran-2-yl, optionally chloro-substituted pyridyl or C1-4 alkyl-S(O)m— wherein m represents 0, 1 or 2, or represents a C3-6 alicyclic hydrocarbon radical; R2 and R3 represent, independently of one another, C1-6 alkyl, C3-7 cycloalkyl or optionally substituted phenyl, or R2 and R3 may form, together with the N-atom to which they are bonded, an optionally substituted ring; R4 represents a hydrogen atom or methyl; and n represents 0 or 1; as well as for their preparation processes and novel intermediates in their production. The inventive compounds of formula (I) are used as herbicides.

    摘要翻译: 式(I)的新的1-取代的甲基四唑啉酮,其中R 1表示具有1至3个杂原子的5元杂环基,其任选地由N,O和S组成,并且任选被卤素和/或C 1-4取代 烷基,或表示环氧乙烷-2-基,任选氯取代的吡啶基或C 1-4烷基-S(O)m - ,其中m表示0,1或2,或表示C 3-6脂族烃基; R 2和R 3彼此独立地表示C 1-6烷基,C 3-7环烷基或任选取代的苯基,或者R 2和R 3可以与它们所键合的N-原子一起形成任选取代的环; R4表示氢原子或甲基; n表示0或1; 以及它们的制备过程和新型中间体的生产。 本发明式(I)化合物用作除草剂。

    Herbicidal 1-substituted methyl-tetrazolinones
    2.
    发明授权
    Herbicidal 1-substituted methyl-tetrazolinones 失效
    除草剂1-取代的甲基 - 四唑啉酮

    公开(公告)号:US6017853A

    公开(公告)日:2000-01-25

    申请号:US890432

    申请日:1997-07-09

    CPC分类号: C07D257/04 A01N47/38

    摘要: Novel 1-substituted methyltetrazolinones of the formula (I) ##STR1## wherein R.sup.1 represents a 5-membered heterocyclic radical which has 1 to 3 heteroatoms selected arbitrarily from the group consisting of N, O and S and which is optionally substituted by halogen and/or C.sub.1-4 alkyl, or represents oxiran-2-yl, optionally chloro-substituted pyridyl or C.sub.1-4 alkyl-S(O).sub.m --wherein m represents 0, 1 or 2, or represents a C.sub.3-6 alicyclic hydrocarbon radical; R.sup.2 and R.sup.3 represent, independently of one another, C.sub.1-4 alkyl, C.sub.3-7 cycloalkyl or optionally substituted phenyl, or R.sup.2 and R.sup.3 may form, together with the N-atom to which they are bonded, an optionally substituted ring; R.sup.4 represents a hydrogen atom or methyl; and n represents 0 or 1; as well as for their preparation processes and novel intermediates in their production. The inventive compounds of formula (I) are used as herbicides.

    摘要翻译: 式(I)的新型1-取代的甲基四唑啉酮,其中R 1表示具有1至3个杂原子的5元杂环基,其任选地由N,O和S组成的组中选择,并且其任选被卤素和/或C1- 或烷基,或表示环氧乙烷-2-基,任选氯取代的吡啶基或C 1-4烷基-S(O)m - ,其中m表示0,1或2,或表示C 3-6脂环族烃基; R 2和R 3彼此独立地表示C 1-4烷基,C 3-7环烷基或任选取代的苯基,或者R 2和R 3可以与它们所键合的N-原子一起形成任选取代的环; R4表示氢原子或甲基; n表示0或1; 以及它们的制备过程和新型中间体的生产。 本发明式(I)化合物用作除草剂。

    Tetrazolinones
    3.
    发明授权
    Tetrazolinones 失效
    四唑啉酮

    公开(公告)号:US5605920A

    公开(公告)日:1997-02-25

    申请号:US618954

    申请日:1996-03-20

    摘要: Disclosed are herbicidal tetrazolinone derivatives, selective in paddy fields of the formula ##STR1## wherein X represents C.sub.1-4 alkyl,n represents 1, 2, 3 or 4,R.sup.1 and R.sup.2 each independently represents C.sub.1-6 alkyl, C.sub.2-4 alkenyl, C.sub.2-6 alkynyl, C.sub.3-8 cycloalkyl, aryl which may optionally be substituted (wherein the substituent is at least one radical selected from the group consisting of halogen, C.sub.1-4 alkyl, C.sub.1-2 haloalkyl, C.sub.1-2 haloalkoxy, C.sub.1-2 haloalkylthio, acyl, nitro and cyano) or aralkyl optionally substituted by halogen orR.sup.1 and R.sup.2 form, together with the N-atom to which they are bonded, a cyclic ring which may be substituted. Also, disclosed are novel intermediates useful in the preparation of the compounds of formula (I).

    摘要翻译: 公开了除草性四唑啉酮衍生物,其在式(I)的水田中是选择性的,其中X表示C1-4烷基,n表示1,2,3或4,R1和R2各自独立地表示C1-6烷基,C2- 4链烯基,C 2-6炔基,C 3-8环烷基,可任选取代的芳基(其中取代基是至少一个选自卤素,C 1-4烷基,C 1-2卤代烷基,C 1-2卤代烷氧基 ,C 1-2卤代烷硫基,酰基,硝基和氰基)或任选被卤素或R 1和R 2形式取代的芳烷基与它们所键合的N-原子一起可以被取代的环状基团。 还公开了可用于制备式(I)化合物的新型中间体。

    Herbicidal 1-cyclopropyl tetrazolinones
    5.
    发明授权
    Herbicidal 1-cyclopropyl tetrazolinones 失效
    除草1-环丙基四唑啉酮

    公开(公告)号:US5650374A

    公开(公告)日:1997-07-22

    申请号:US553160

    申请日:1995-11-07

    CPC分类号: C07D257/04 A01N47/38

    摘要: Herbicidal 1-cyclopropyl tetrazolinones of the formula ##STR1## wherein X represents C.sub.1-3 alkyl, C.sub.2-4 alkenyl or halogen,n represents 0 to 5,R.sup.1 and R.sup.2 each independently represents C.sub.1-6 alkyl, C.sub.2-6 alkenyl, C.sub.2-6 alkynyl, C.sub.3-7 cycloalkyl which may optionally be substituted by C.sub.1-3 alkyl, epoxy-C.sub.3-5 alkan-1-yl, phenyl which may optionally be substituted, or aralkyl which may optionally be substituted, orR.sup.1 and R.sup.2 together with the N-atom to which they are attached, represent a cyclic ring which may be substituted, and some novel intermediates therefor.

    摘要翻译: 式(I)的除草1-环丙基四唑啉酮其中X代表C1-3烷基,C2-4烯基或卤素,n代表0-5,R1和R2各自独立地表示C1-6烷基,C2-6烯基 C 2-6炔基,可任选被C 1-3烷基取代的C 3-7环烷基,环烷基-C 3-5烷基-1-基,可任意被取代的苯基或可任意被取代的芳烷基,或R 1和 R2与它们所连接的N-原子一起表示可以被取代的环状环,以及一些新的中间体。

    1-cycloalkenyltetrazolinones
    7.
    发明授权
    1-cycloalkenyltetrazolinones 失效
    1-环烯基四唑啉酮

    公开(公告)号:US5654257A

    公开(公告)日:1997-08-05

    申请号:US601748

    申请日:1996-02-15

    CPC分类号: C07D257/04 A01N47/38

    摘要: 1-cycloalkenyltetrazolinone derivatives of the following herbicidal formula ##STR1## R.sup.1 is cycloalkenyl which may optionally be substituted by halogen C.sub.1-4 alkyl, or bicycloalkenyl which may optionally be substituted by halogen or C.sub.1-4 alkyl, andR.sup.2 and R.sup.3 each independently is alkyl, cycloalkyl, phenyl (optionally substituted by a member selected from the group consisting of nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and alkylthio), alkenyl and alkynyl,orR.sup.2 and R.sup.3 together with the N-atom to which they are bonded form, a 5- or 6-membered heterocyclic ring which may optionally contain a further hetero atom, said heterocyclic ring optionally being benzo-condensed, or a C-.sub.1-4 alkyl,and intermediates therefore of the formula ##STR2##

    摘要翻译: 以下除草式R 1的1-环烯基四唑啉酮衍生物是可任选被卤素C 1-4烷基取代的环烯基,或可任意被卤素或C 1-4烷基取代的双环烯基,R 2和R 3各自独立地为烷基 ,环烷基,苯基(任选被选自硝基,氰基,卤素,烷基,卤代烷基,烷氧基,卤代烷氧基和烷硫基的成员取代),烯基和炔基,或者R 2和R 3与它们的N-原子一起 键合形式,可任选地含有另外的杂原子的所述5或6元杂环,所述杂环任选地被苯并稠合,或C 1-4烷基,因此具有下式的中间体: