N-P-Cyanoaryl nitrogen-containing heterocycles having pendent sulfur-containing groups
    73.
    发明授权
    N-P-Cyanoaryl nitrogen-containing heterocycles having pendent sulfur-containing groups 失效
    含有含硫基团的N-P-氰基芳基含氮杂环

    公开(公告)号:US06339044B1

    公开(公告)日:2002-01-15

    申请号:US09049447

    申请日:1998-03-27

    IPC分类号: C07D23954

    CPC分类号: C07D239/56 A01N43/54

    摘要: N-Cyanoaryl nitrogen heterocycles having sulfur-containing groups of the formula (1), in which Q1 represents oxygen or sulfur, R1 represents hydrogen or halogen, R2 represents halogen, cyano, nitro, amino or the grouping —N(A1)SO2A, in which A represents, in each case, optionally substituted alkyl, alkenyl, alkinyl, dialkylamino, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl, and A1 represents hydrogen, formyl or, in each case optionally substituted, alkyl, alkenyl, alkinyl, alkylcarbonyl, alkoxycarbonyl or alkylsulphonyl, or together with A represents alkanediyl, R3 represents hydrogen, halogen, cyano or optionally substituted alkyl, R4 represents optionally substituted alkyl or together with R3 represents alkanediyl, and Z represents one of the groups in which Q2 represents oxygen or sulfur and R5 represents hydrogen or, in each case optionally substituted, alkyl, alkenyl, alkinyl or alkylcarbonyl, and salts of compounds of the formula (1) with the proviso that at least one of the groupings Q1 or Q2 represents sulfur. Several processes are disclosed for preparing these compounds which are useful as herbicides and insecticides.

    摘要翻译: 具有式(1)的含硫基团的N-氰基芳基氮杂环,其中Q1表示氧或硫,R1表示氢或卤素,R2表示卤素,氰基,硝基,氨基或-N(A1)SO2A基团, 在任何情况下,A表示任选取代的烷基,烯基,炔基,二烷基氨基,环烷基,环烷基烷基,芳基或芳基烷基,A表示氢,甲酰基或在各种情况下任选取代的烷基,烯基,炔基,烷基羰基,烷氧基羰基或烷基磺酰基,或 与A一起表示烷二基,R 3表示氢,卤素,氰基或任选取代的烷基,R 4表示任选取代的烷基或与R 3表示烷二基,Z表示其中Q 2表示氧或硫并且R 5表示氢的基团之一, 取代的,烷基,烯基,炔基或烷基羰基,以及式(1)化合物的盐,条件是至少一个分组Q1或 Q2代表硫。公开了用于制备可用作除草剂和杀虫剂的这些化合物的几种方法。

    Substituted 2,4-diamino-1,3,5-triazines as herbicides
    77.
    发明授权
    Substituted 2,4-diamino-1,3,5-triazines as herbicides 失效
    取代的2,4-二氨基-1,3,5-三嗪作为除草剂

    公开(公告)号:US06399541B1

    公开(公告)日:2002-06-04

    申请号:US09381442

    申请日:1999-10-18

    IPC分类号: A01N4368

    CPC分类号: A01N43/68 C07D251/18

    摘要: The invention relates to novel substituted 2,4-diamino-1,3,5-triazines of the formula (I) in which R1 represents (in each case unsubstituted) phenyl or naphthyl R2 represents alkyl, R3 represents hydrogen, represents halogen or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl or alkylsulphonyl, R4 represents hydrogen, represents halogen or represents optionally substituted alkyl, R5 represents hydrogen, represents halogen or represents optionally substituted alkyl, and R6 represents hydrogen or represents in each case optionally substituted alkyl, alkylcarbonyl or alkylsulphonyl, (but where the compound 2-amino-4-(1-phenyl-ethylamino)-6-trifluoromethyl-1,3,5-triazine is excluded), to processes for preparing the novel compounds and to their use as herbicides.

    摘要翻译: 本发明涉及式(I)的新的取代的2,4-二氨基-1,3,5-三嗪,其中R 1表示(在每种情况下未被取代的)苯基或萘基,R 2表示烷基,R 3表示氢,表示卤素,或各自表示 任选取代的烷基,烷氧基,烷硫基,烷基亚磺酰基或烷基磺酰基,R 4表示氢,表示卤素,或表示任选取代的烷基,R 5表示氢,表示卤素或表示任选取代的烷基,R 6表示氢或表示任意取代的烷基,烷基羰基 或烷基磺酰基(但不包括化合物2-氨基-4-(1-苯基 - 乙基氨基)-6-三氟甲基-1,3,5-三嗪)),制备新化合物的方法及其作为除草剂的用途 。

    Herbicidal sulphonylamino(thio) carbonyl compounds
    78.
    再颁专利
    Herbicidal sulphonylamino(thio) carbonyl compounds 失效
    除草磺酰氨基(硫)羰基化合物

    公开(公告)号:USRE39607E1

    公开(公告)日:2007-05-01

    申请号:US10603997

    申请日:2003-06-25

    IPC分类号: A01N43/653 C07D249/12

    摘要: The invention relates to novel sulphonylamino(thio) carbonyl compounds of the formula (I), in which A represents a single bond, oxygen, sulphur or the group N—R, in which R represents hydrogen, alkyl, alkenyl, alkinyl or cycloalkyl, Q represents oxygen or sulphur, R1 represents hydrogen or formyl or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, cycloalkyl, cycloalkylcarbonyl or cycloalkylsulphonyl, R2 represents cyano or halogen or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy or alkinyloxy, and R3 represents in each case optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulphur or nitrogen and from one to three further ring members can be nitrogen, and salts of compounds of the formula (I), the previously known compounds 4,5-dimethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one, 4,5-diethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one and N-(2,5-dimethoxy-phenylsulphonyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide being excluded by disclaimer; and also to processes and novel intermediates for the preparation of the novel substances and to their use as herbicides.

    摘要翻译: 本发明涉及式(I)的新型磺酰基氨基(硫代)羰基化合物,其中A表示单键,氧,硫或基团NR,其中R表示氢,烷基,烯基,炔基或环烷基,Q表示 氧或硫,R 1表示氢或甲酰基,或在各种情况下表示任选取代的烷基,烯基,炔基,烷基羰基,烷氧基羰基,烷基磺酰基,环烷基,环烷基羰基或环烷基磺酰基,R 2 >表示氰基或卤素,或表示在各种情况下任选取代的烷基,烯基,炔基,烷氧基,烯氧基或烷氧基,R 3表示在每种情况下任选取代的具有5个环成员的杂环基,其中至少一个 是氧,硫或氮,并且一至三个其它的环成员可以是氮,并且式(I)化合物的盐,先前已知的化合物4,5-二甲氧基-2-(2,5-二甲氧基 - 苯基磺酰基氨基羰基) -2,4-二氢-3H- 1,2,4-三唑-3-酮,4,5-二乙氧基-2-(2,5-二甲氧基 - 苯基磺酰基氨基羰基)-2,4-二氢-3H-1,2,4-三唑-3-酮和 通过免责声明排除N-(2,5-二甲氧基 - 苯基磺酰基)-1,5-二甲基-1H-吡唑-3-甲酰胺; 以及用于制备新物质及其作为除草剂的用途的方法和新型中间体。