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81 条记录 (耗时 0.052 秒)

    Method for producing alkenyl-substituted bis(oxime ether) derivatives
    74.
    发明授权
    Method for producing alkenyl-substituted bis(oxime ether) derivatives 失效
    烯基取代的双（肟醚）衍生物的制备方法

    公开(公告)号：US06417388B1

    公开(公告)日：2002-07-09

    申请号：US09831412

    申请日：2001-05-09

    申请人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Norbert Götz ,  Roland Götz

    发明人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Norbert Götz ,  Roland Götz

    IPC分类号： C07C22900

    CPC分类号： C07C249/12 ,  C07C251/60

    摘要： The process for preparing alkenyl-substituted bis(oxime ether) derivatives of the formula I where: R1 is unsubstituted C1-C4-alkyl or C2-C4-alkenyl-, C2-C4-alkynyl- or phenyl-substituted methyl; R2, R4 independently of one another are hydrogen or methyl; R3, R5 independently of one another are hydrogen or C1-C4-alkyl, trifluoromethyl or phenyl and X is —C(═CHCH3)—COOCH3, —C(═CHOCH3)—COOCH3, —C(═NOCH3)—COOCH3, —C(═NOCH3)—CONHCH3 or —N(OCH3)—COOCH3, and intermediates which are obtainable by this process are described. Alkenyl-substituted bis(oxime ether) derivatives of the formula I are described in the literature as interesting crop protection agents.

    摘要翻译： 制备式I的烯基取代的双（肟醚）衍生物的方法，其中：R1是未取代的C1-C4-烷基或C2-C4-烯基 - ，C2-C4-炔基或苯基取代的甲基; R2，R4独立地 其中R 3，R 5彼此独立地是氢或C 1 -C 4烷基，三氟甲基或苯基，X是-C（= CHCH 3）-COOCH 3，-C（= CHOCH 3）-COOCH 3，-C（ = NOCH 3）-COOCH 3，-C（= NOCH 3）-CONHCH 3或-N（OCH 3）-COOCH 3，并且可以通过该方法获得的中间体。 式I的烯基取代的双（肟醚）衍生物在文献中描述为有趣的作物保护剂。

    Fungicidal 5-Hydroxypyrazolines, Method for Producing the Same and Agents Comprising the Same
    75.
    发明申请
    Fungicidal 5-Hydroxypyrazolines, Method for Producing the Same and Agents Comprising the Same 审中-公开
    杀真菌剂5-羟基吡唑啉，其制备方法及其制剂

    公开(公告)号：US20080194405A1

    公开(公告)日：2008-08-14

    申请号：US11915989

    申请日：2006-05-24

    申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    IPC分类号： A01N43/56 ,  C07D231/08 ,  A01P3/00

    CPC分类号： A01N43/56

    摘要： The present invention relates to novel 5-hydroxypyrazolines of the formula I in which the substituents are as defined below: B is phenyl, naphthyl or 5- or 6-membered hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; A is C═O, C═S or SO2; R1 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, phenyl, 5- or 6-membered heterocyclyl or hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; R2 is alkyl, haloalkyl, alkenyl, haloalkyl, alkynyl, haloalkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, phenyl, 5- or 6-membered hetaryl or heterocyclyl which contains one to four heteroatoms from the group consisting of O, N and S; R3 is hydrogen, nitro, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, haloalkenyl, alkynyl, haloalkynyl or NR′2, where R′ independently of one another are hydrogen or alkyl; R4 is hydrogen, halogen, nitro, cyano, NR′2, alkyl, haloalkyl, COOR′ or 5- or 6-membered hetaryl or heterocyclyl; where the variables mentioned above may be substituted according to the description; processes for their preparation, their use for controlling harmful fungi and compositions comprising them.

    摘要翻译： 本发明涉及式I的新的5-羟基吡唑啉，其中取代基如下所定义：B是苯基，萘基或5-或6-元杂芳基，其含有一至四个由O，N和 S; A是C-O，C-S或SO 2。 R 1是烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基，环烷基，环烯基，环炔基，苯基，5-或6-元杂环基或杂芳基，其含有一至四个 O，N和S; R 2是烷基，卤代烷基，烯基，卤代烷基，炔基，卤代炔基，环烷基，环烯基，环炔基，苯基，5-或6-元杂芳基或杂环基，其含有一至四个 O，N和S; R 3是氢，硝基，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，卤代烯基，炔基，卤代炔基或NR'2，其中R'彼此独立地 是氢或烷基; R 4是氢，卤素，硝基，氰基，NR'2，烷基，卤代烷基，COOR'或5-或6-元杂芳基或杂环基; 其中上述变量可以根据描述被替代; 其制备方法，它们用于控制有害真菌的用途和包含它们的组合物。

    Bicyclic 5-Hydroxypyrazolines, Method For Producing the Same and Agents Comprising the Same
    76.
    发明申请
    Bicyclic 5-Hydroxypyrazolines, Method For Producing the Same and Agents Comprising the Same 审中-公开
    双环5-羟基吡唑啉，其制备方法和包含其的试剂

    公开(公告)号：US20080227840A1

    公开(公告)日：2008-09-18

    申请号：US11916201

    申请日：2006-05-24

    申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    IPC分类号： A01N43/56 ,  C07D231/54 ,  A01N25/26 ,  A01P3/00

    CPC分类号： C07D401/12 ,  A01N43/56 ,  C07D231/56

    摘要： Bicyclic 5-hydroxypyrazolines of the formula I in which the substituents are as defined below: B is phenyl, naphthyl or 5- or 6-membered hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; A is C═O, C═S or SO2; R1 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, phenyl, 5- or 6-membered heterocyclyl or hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; R2 together with R1 or R4 is C3-C4-alkylene or C3-C4-alkenylene, which groups may be defined according to the description, R3 is hydrogen, nitro, cyano, NR″2, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, haloalkenyl, alkynyl or haloalkynyl, where R″ independently of one another are hydrogen or alkyl; R4 is hydrogen, halogen, nitro, cyano, NR″2, alkyl, haloalkyl, COOR″, hetaryl or heterocyclyl; where the variables mentioned above may be substituted according to the description; processes for their preparation, their use for controlling harmful fungi and compositions comprising them.

    摘要翻译： 其中取代基如下定义的式I的双环5-羟基吡唑啉：B是含有一至四个由O，N和S组成的组的杂原子的苯基，萘基或5-或6-元杂芳基; A是C-O，C-S或SO 2。 R 1是烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基，环烷基，环烯基，环炔基，苯基，5-或6-元杂环基或杂芳基，其含有一至四个 O，N和S; R 2与R 1或R 4一起是C 3 -C 4烷基， - 亚烷基或C 3 -C 4 - 亚烯基，这些基团可以根据描述定义，R 3是氢，硝基，氰基 ，NR“2，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，卤代烯基，炔基或卤代炔基，其中R”彼此独立地是氢或烷基; R 4是氢，卤素，硝基，氰基，NR“2，烷基，卤代烷基，COOR”，杂芳基或杂环基; 其中上述变量可以根据描述被替代; 其制备方法，它们用于控制有害真菌的用途和包含它们的组合物。

    Fungicidal N-Benzyl-5-Hydroxy-5-Phenylpryrazolines, Processes For Their Preparation and Compositions Comprising Them
    77.
    发明申请
    Fungicidal N-Benzyl-5-Hydroxy-5-Phenylpryrazolines, Processes For Their Preparation and Compositions Comprising Them 审中-公开
    杀真菌剂N-苄基-5-羟基-5-苯基吡唑啉，其制备方法及其组合

    公开(公告)号：US20080214642A1

    公开(公告)日：2008-09-04

    申请号：US11916233

    申请日：2006-05-24

    申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    IPC分类号： A01N43/56 ,  C07D231/08 ,  A01P3/00

    CPC分类号： C07D231/08 ,  A01N43/56

    摘要： N-benzoyl-5-hydroxy-5-phenylpyrazolines of the formula I in which the substituents are as defined below: L1, L2 are hydrogen, halogen, haloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl; L3, L4, L5 are alkyl or one of the groups mentioned under L1 and L2; X is oxygen or sulfur; R1 is halogen, nitro, cyano, NR′2, alkyl, haloalkyl, alkoxy, alkenyl, haloalkyl, alkynyl, haloalkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, phenyl, 5- or 6-membered heterocyclyl or hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; R′ independently of one another are hydrogen or alkyl; m is 1, 2, 3, 4 or 5; R2 is hydrogen or alkyl; R3 is hydrogen, nitro, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, haloalkenyl, alkynyl, haloalkynyl or NR′2, where R4 is hydrogen, halogen, nitro, cyano, NR′2, alkyl, haloalkyl, COOR′ or 5- or 6-membered heterocyclyl or hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; where the variables mentioned above may be substituted according to the description; processes for their preparation, their use for controlling harmful fungi and compositions comprising them.

    摘要翻译： 其中取代基如下定义的式I的N-苯甲酰基-5-羟基-5-苯基吡唑：L 1，L 2是氢，卤素，卤代烷基， 烯基，卤代烯基，炔基或卤代炔基; L 3，L 4，L 5是烷基或在L 1和L 2之间提及的基团之一， SUP> 2 ; X是氧或硫; R 1是卤素，硝基，氰基，NR'2，烷基，卤代烷基，烷氧基，烯基，卤代烷基，炔基，卤代炔基，环烷基，环烯基，环炔基，苯基，5 - 或6元杂环基或杂芳基，其含有一至四个由O，N和S组成的组的杂原子; R'彼此独立地是氢或烷基; m为1,2,3,4或5; R 2是氢或烷基; R 3是氢，硝基，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，卤代烯基，炔基，卤代炔基或NR'2，其中R 4， / SUP>是氢，卤素，硝基，氰基，NR'2，烷基，卤代烷基，COOR'或5-或6-元杂环基或杂芳基，其含有一至四个由以下组成的组的杂原子： O，N和S; 其中上述变量可以根据描述被替代; 其制备方法，它们用于控制有害真菌的用途和包含它们的组合物。

    Fungicidal 5-Hydroxypyrazolines, Processes for their Preparation and Comprising Them
    78.
    发明申请
    Fungicidal 5-Hydroxypyrazolines, Processes for their Preparation and Comprising Them 审中-公开
    杀真菌剂5-羟基吡唑啉，其制备方法及其组成

    公开(公告)号：US20080182886A1

    公开(公告)日：2008-07-31

    申请号：US11915779

    申请日：2006-05-24

    申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Andreas Gypser ,  Matthias Niedenbruck

    IPC分类号： A01N43/56 ,  C07D231/06 ,  A01P3/00 ,  A01N25/26

    CPC分类号： A01N43/56 ,  C07D231/06

    摘要： Novel 5-hydroxypyrazolines of the formula I in which the substituents are as defined below: B is phenyl, naphthyl or 5- or 6-membered hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; A is C═O, C═S or SO2; W is CX1X2; X1, X2 are hydrogen, fluorine, chlorine or bromine; R1 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, phenyl, 5- or 6-membered heterocyclyl or hetaryl which contains one to four heteroatoms from the group consisting of O, N and S; R2 is hydrogen or alkyl; R3 is hydrogen, nitro, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, haloalkenyl, alkynyl, haloalkynyl or NR′2, where R′ independently of one another are hydrogen or alkyl; R4 is hydrogen, halogen, nitro, cyano, NR′2, alkyl, haloalkyl, COOR′ or 5- or 6-membered hetaryl or heterocyclyl; where the variables mentioned above may be substituted according to the description; processes for their preparation, their use for controlling harmful fungi and compositions comprising them.

    摘要翻译： 式I的新型5-羟基吡唑啉，其中取代基如下所定义：B是苯基，萘基或含有一至四个由O，N和S组成的组的杂原子的5-或6-元杂芳基; A是C-O，C-S或SO 2。 W是CX 1，X 2， X 1，X 2是氢，氟，氯或溴; R 1是烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基，环烷基，环烯基，环炔基，苯基，5-或6-元杂环基或杂芳基，其含有一至四个 O，N和S; R 2是氢或烷基; R 3是氢，硝基，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，卤代烯基，炔基，卤代炔基或NR'2，其中R'彼此独立地 是氢或烷基; R 4是氢，卤素，硝基，氰基，NR'2，烷基，卤代烷基，COOR'或5-或6-元杂芳基或杂环基; 其中上述变量可以根据描述被替代; 其制备方法，它们用于控制有害真菌的用途和包含它们的组合物。

    5-phenypyrimidines their preparation compositions comprising them and their use
    80.
    发明申请
    5-phenypyrimidines their preparation compositions comprising them and their use 失效

    公开(公告)号：US20060148764A1

    公开(公告)日：2006-07-06

    申请号：US10495280

    申请日：2002-11-15

    申请人： Andreas Gypser

    发明人： Andreas Gypser

    IPC分类号： A61K31/655 ,  A61K31/513 ,  A61K31/506 ,  A61K31/505 ,  C07D239/47 ,  C07D403/02

    CPC分类号： C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

    摘要： 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C(═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.