-
公开(公告)号：US20090186924A1
公开(公告)日：2009-07-23
申请号：US12407365
申请日：2009-03-19
申请人： Denis Billen , Jessica Boyle , Douglas James Critcher , David Morris Gethin , Kim Thomas Hall , Graham Michael Kyne
发明人： Denis Billen , Jessica Boyle , Douglas James Critcher , David Morris Gethin , Kim Thomas Hall , Graham Michael Kyne
IPC分类号： A61K31/415 , A61K31/4439 , A61K31/427 , C07D401/12 , C07D417/06 , C07D403/12 , C07D231/38 , C07D231/14 , A61P33/00
CPC分类号： C07D231/38 , A01N53/00 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/40 , C07D401/04 , C07D401/12 , C07D403/12 , C07D405/12 , C07D413/06 , C07D413/12 , C07D417/06 , C07D417/12 , C07D417/14 , C07D487/04
摘要： This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which the cyclopropyl ring is substituted at the angular position, and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.
摘要翻译： 本发明涉及其中环丙基环在角位置被取代的1-芳基-4-环丙基吡唑的范围及其药学上可接受的盐和溶剂化物，包括这些化合物的组合物，其合成方法及其作为杀寄生虫剂的用途。
-
公开(公告)号：US20090137524A1
公开(公告)日：2009-05-28
申请号：US12364879
申请日：2009-02-03
申请人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
发明人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
IPC分类号： A01N43/16 , C07D403/04 , A01N43/40 , A01P1/00 , A01N43/56 , C07D231/14
CPC分类号： C07D401/04 , A61K31/415 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/12 , C07D403/12 , C07D413/04 , A61K2300/00
摘要： This invention relates to a combination product comprising a compound of formula I wherein X, R1, R2, R3, R4, R5, R6, R7 and R9 are as described herein, and one or more further biologically active compounds as described herein, particularly anti-parasitic agents.
摘要翻译： 本发明涉及包含式I化合物的组合产品，其中X，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 9如本文所述，以及本文所述的一种或多种其它生物活性化合物， - 寄生虫剂。
-
公开(公告)号：US07968584B2
公开(公告)日：2011-06-28
申请号：US12407365
申请日：2009-03-19
申请人： Denis Billen , Jessica Boyle , Douglas James Critcher , David Morris Gethin , Kim Thomas Hall , Graham Michael Kyne
发明人： Denis Billen , Jessica Boyle , Douglas James Critcher , David Morris Gethin , Kim Thomas Hall , Graham Michael Kyne
IPC分类号： A61K31/415 , C07D231/10
CPC分类号： C07D231/38 , A01N53/00 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/40 , C07D401/04 , C07D401/12 , C07D403/12 , C07D405/12 , C07D413/06 , C07D413/12 , C07D417/06 , C07D417/12 , C07D417/14 , C07D487/04
摘要： This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which the cyclopropyl ring is substituted at the angular position, and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.
摘要翻译： 本发明涉及其中环丙基环在角位置被取代的1-芳基-4-环丙基吡唑的范围及其药学上可接受的盐和溶剂化物，包括这些化合物的组合物，其合成方法及其作为杀寄生虫剂的用途。
-
公开(公告)号：US20090312371A1
公开(公告)日：2009-12-17
申请号：US11917389
申请日：2006-06-06
申请人： Denis Billen , Nathan Anthony Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Walshe
发明人： Denis Billen , Nathan Anthony Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Walshe
IPC分类号： A61K31/4439 , A61K31/415 , A61P33/00
CPC分类号： C07D401/04 , A61K31/415 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/12 , C07D403/12 , C07D413/04 , A61K2300/00
摘要： This invention relates to a combination product comprising a range of 1-aryl-4-cyclopropylpyrazoles in which there is at least one fluorine attached to the cyclopropyl ring, and one o more further therapeutic agents, particularly anti-parasitic agents.
摘要翻译： 本发明涉及包含一系列1-芳基-4-环丙基吡唑的组合产品，其中至少一个氟连接到环丙基环上，另外还有一种还有更多的治疗剂，特别是抗寄生虫剂。
-
公开(公告)号：US07538134B2
公开(公告)日：2009-05-26
申请号：US11453053
申请日：2006-06-14
申请人： Denis Billen , Jessica Boyle , Douglas James Critcher , David Morris Gethin , Kim Thomas Hall , Graham Michael Kyne
发明人： Denis Billen , Jessica Boyle , Douglas James Critcher , David Morris Gethin , Kim Thomas Hall , Graham Michael Kyne
IPC分类号： A61K31/415 , C07D231/10
CPC分类号： C07D231/38 , A01N53/00 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/40 , C07D401/04 , C07D401/12 , C07D403/12 , C07D405/12 , C07D413/06 , C07D413/12 , C07D417/06 , C07D417/12 , C07D417/14 , C07D487/04
摘要： This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which the cyclopropyl ring is substituted at the angular position, and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.
摘要翻译： 本发明涉及其中环丙基环在角位置被取代的1-芳基-4-环丙基吡唑的范围及其药学上可接受的盐和溶剂化物，包括这些化合物的组合物，其合成方法及其作为杀寄生虫剂的用途。
-
公开(公告)号：US07514464B2
公开(公告)日：2009-04-07
申请号：US11153103
申请日：2005-06-15
申请人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
发明人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
IPC分类号： A61K31/4439 , C07D231/10
CPC分类号： C07D401/04 , A61K31/415 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/12 , C07D403/12 , C07D413/04 , A61K2300/00
摘要： This invention relates to a combination product comprising a compound of formula I wherein X, R1, R2, R3, R4, R5, R6, R7 and R9 are as described herein, and one or more further biologically active compounds as described herein, particularly anti-parasitic agents.
摘要翻译： 本发明涉及包含式I化合物的组合产品，其中X，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 9如本文所述，以及本文所述的一种或多种其它生物活性化合物， - 寄生虫剂。
-
公开(公告)号：US07435753B2
公开(公告)日：2008-10-14
申请号：US11013176
申请日：2004-12-15
申请人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
发明人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
IPC分类号： A61K31/4439 , C07D231/10
CPC分类号： A01N43/56 , A61K31/415 , A61K31/416 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/04 , C07D401/12 , C07D413/04
摘要： This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which there is at least one fluorine attached to the cyclopropyl ring, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.
摘要翻译： 本发明涉及其中存在至少一个与环丙基环连接的氟的1-芳基-4-环丙基吡唑的范围，包含这些化合物的组合物，其合成方法及其作为杀寄生物的用途。
-
公开(公告)号：US20050148649A1
公开(公告)日：2005-07-07
申请号：US11013176
申请日：2004-12-15
申请人： Denis Billen , Nathan Chubb , David Gethin , Kim Hall , Lee Roberts , Nigel Walshe
发明人： Denis Billen , Nathan Chubb , David Gethin , Kim Hall , Lee Roberts , Nigel Walshe
IPC分类号： A01N43/56 , A61K31/415 , A61K31/416 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/04 , C07D401/12 , C07D403/12 , C07D413/04 , C07D43/02
CPC分类号： A01N43/56 , A61K31/415 , A61K31/416 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/04 , C07D401/12 , C07D413/04
摘要： This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which there is at least one fluorine attached to the cyclopropyl ring, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.
摘要翻译： 本发明涉及其中存在至少一个与环丙基环连接的氟的1-芳基-4-环丙基吡唑的范围，包含这些化合物的组合物，其合成方法及其作为杀寄生物的用途。
-
公开(公告)号：US08084486B2
公开(公告)日：2011-12-27
申请号：US13089423
申请日：2011-04-19
申请人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
发明人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
IPC分类号： A61K31/415 , C07D231/10
CPC分类号： C07D401/04 , A61K31/415 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/12 , C07D403/12 , C07D413/04 , A61K2300/00
摘要： This invention relates to a combination product comprising a compound of formula I wherein X, R1, R2, R3, R4, R5, R6, R7 and R9 are as described herein, and one or more further biologically active compounds as described herein, particularly anti-parasitic agents.
摘要翻译： 本发明涉及包含式I化合物的组合产品，其中X，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 9如本文所述，以及本文所述的一种或多种其它生物活性化合物， - 寄生虫剂。
-
公开(公告)号：US07960426B2
公开(公告)日：2011-06-14
申请号：US12364879
申请日：2009-02-03
申请人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
发明人： Denis Billen , Nathan Anthony Logan Chubb , David Morris Gethin , Kim Thomas Hall , Lee Richard Roberts , Nigel Derek Arthur Walshe
IPC分类号： A61K31/415 , C07D231/10
CPC分类号： C07D401/04 , A61K31/415 , A61K31/4439 , C07D231/38 , C07D231/40 , C07D401/12 , C07D403/12 , C07D413/04 , A61K2300/00
摘要： This invention relates to a combination product comprising a compound of formula I wherein X, R1, R2, R3, R4, R5, R6, R7 and R9 are as described herein, and one or more further biologically active compounds as described herein, particularly anti-parasitic agents.
-
-
-
-
-
-
-
-
-
搜索结果
23 条记录 (耗时 0.038 秒)
