公开(公告)号：US4116674A

公开(公告)日：1978-09-26

申请号：US597572

申请日：1975-07-21

申请人： Raymond Leo Sunley ,  Geoffrey David Snowling

发明人： Raymond Leo Sunley ,  Geoffrey David Snowling

IPC分类号： C07D239/47 ,  A01N43/54 ,  C07D239/42 ,  C07D239/46 ,  C07D239/48 ,  C07D239/56 ,  A01N9/22

CPC分类号： C07D239/47 ,  C07D239/42 ,  C07D239/46 ,  C07D239/48 ,  C07D239/56

摘要： A process of severely damaging or killing unwanted plants, which comprises applying to the plants, or to the growth medium thereof, a herbicidally effective amount of pyrimidine compound of the formula: ##STR1## or a herbicidal acid addition salt thereof, wherein R.sup.1 is an alkyl radical of 1 to 6 carbon atoms, cycloalkyl or alkenyl; R is a hydrogen atom or an alkyl or alkenyl radical of from 1 to 12 carbon atoms, which may be substituted by a phenyl radical; or R.sup.1 and R taken together form a trimethylene or tetramethylene radical; X is either (a) an --NR.sup.3 R.sup.4 radical wherein each of the groups R.sup.2 and R.sup.4 is a hydrogen atom or an alkyl or alkenyl radical of 1 to 3 carbon atoms or cycloalkyl, or --NR.sup.3 R.sup.4 constitutes a pyrrolidinyl, piperidinyl or morpholinyl ring; or (b) a group --OR.sup.5 wherein R.sup.5 is an alkyl or alkenyl radical of 1 to 10 carbon atoms or cycloalkyl; and R.sup.6 and R.sup.7 each represent hydrogen or an alkyl or alkenyl radical of 1 to 8 carbon atoms, or cycloalkyl, or R.sup.6 and R.sup.7, taken together with the nitrogen atom to which they are attached constitute a pyrrolidinyl, piperidinyl, or morpholinyl ring; provided that R may be hydrogen only when X is an OR.sup.5 group.

摘要翻译： 一种严重破坏或杀死有害植物的方法，其包括向植物或其生长培养基施用除草有效量的下式嘧啶化合物或其除草酸加成盐，其中R1为 1至6个碳原子的烷基，环烷基或链烯基; R是氢原子或具有1至12个碳原子的烷基或烯基，其可被苯基取代; 或R 1和R一起形成三亚甲基或四亚甲基; X是（a）-NR 3 R 4基团，其中基团R 2和R 4各自是氢原子或1至3个碳原子的烷基或烯基或环烷基，或-NR 3 R 4构成吡咯烷基，哌啶基或吗啉基; 或（b）基团-OR5，其中R5是1-10个碳原子的烷基或烯基或环烷基; 并且R 6和R 7各自表示氢或1〜8个碳原子的烷基或烯基，或环烷基，或者R 6和R 7与它们所连接的氮原子一起构成吡咯烷基，哌啶基或吗啉基; 条件是只有当X是OR 5基团时，R可以是氢。