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1.
公开(公告)号:US20070142393A1
公开(公告)日:2007-06-21
申请号:US11668906
申请日:2007-01-30
申请人: Kristof Emelen , Janine Arts , Leo Backx , Hans De Winter , Sven Van Brandt , Marc Verdonck , Lieven Meerpoel , Isabelle Pilatte , Virginie Poncelet , Alexey Dyatkin , Jimmy Van heusden
发明人: Kristof Emelen , Janine Arts , Leo Backx , Hans De Winter , Sven Van Brandt , Marc Verdonck , Lieven Meerpoel , Isabelle Pilatte , Virginie Poncelet , Alexey Dyatkin , Jimmy Van heusden
IPC分类号: A61K31/506 , C07D403/04
CPC分类号: C07D413/12 , A61K31/40 , A61K31/402 , A61K31/435 , A61K31/4427 , A61K31/454 , A61K31/4545 , A61K31/472 , A61K31/495 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K31/55 , A61K45/06 , C07D207/09 , C07D207/14 , C07D207/277 , C07D207/28 , C07D211/14 , C07D211/58 , C07D213/78 , C07D213/81 , C07D213/82 , C07D217/02 , C07D217/04 , C07D217/16 , C07D233/90 , C07D239/42 , C07D241/04 , C07D241/24 , C07D243/08 , C07D261/10 , C07D295/155 , C07D295/22 , C07D295/26 , C07D307/68 , C07D307/79 , C07D333/34 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12 , C07D405/06 , C07D409/04 , C07D409/12 , C07D409/14 , C07D413/04 , C07D413/14 , C07D471/04 , C07D471/10 , C07D513/04 , C12Q1/34 , C12Q1/48 , G01N33/573 , G01N2333/91
摘要: This invention comprises the novel compounds of formula (I) wherein n, m, t, R1, R2, R3, R4, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
摘要翻译: 本发明包括新的式(I)化合物,其中n,m,t,R 1,R 2,R 3,R 3, 具有组氨酸脱乙酰酶抑制酶活性的含义; 其制剂,含有它们的组合物及其作为药物的用途。
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2.
公开(公告)号:US20080108601A1
公开(公告)日:2008-05-08
申请号:US11926759
申请日:2007-10-29
申请人: Kristof Van Emelen , Janine Arts , Leo-Jacobus Backx , Hans De Winter , Sven Van Brandt , Marc Verdonck , Lieven Meerpoel , Isabelle Pilatte , Virginie Poncelet , Alexey Dyatkin , Jimmy Van heusden
发明人: Kristof Van Emelen , Janine Arts , Leo-Jacobus Backx , Hans De Winter , Sven Van Brandt , Marc Verdonck , Lieven Meerpoel , Isabelle Pilatte , Virginie Poncelet , Alexey Dyatkin , Jimmy Van heusden
IPC分类号: A61K31/551 , A61K31/495 , A61K31/501 , C07D241/04 , C07D403/04 , C12Q1/00 , C07D413/14 , C07D243/08 , A61K31/506 , A61K31/5355
CPC分类号: C07D413/12 , A61K31/40 , A61K31/402 , A61K31/435 , A61K31/4427 , A61K31/454 , A61K31/4545 , A61K31/472 , A61K31/495 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K31/55 , A61K45/06 , C07D207/09 , C07D207/14 , C07D207/277 , C07D207/28 , C07D211/14 , C07D211/58 , C07D213/78 , C07D213/81 , C07D213/82 , C07D217/02 , C07D217/04 , C07D217/16 , C07D233/90 , C07D239/42 , C07D241/04 , C07D241/24 , C07D243/08 , C07D261/10 , C07D295/155 , C07D295/22 , C07D295/26 , C07D307/68 , C07D307/79 , C07D333/34 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12 , C07D405/06 , C07D409/04 , C07D409/12 , C07D409/14 , C07D413/04 , C07D413/14 , C07D471/04 , C07D471/10 , C07D513/04 , C12Q1/34 , C12Q1/48 , G01N33/573 , G01N2333/91
摘要: This invention comprises the novel compounds of formula (I) wherein n, m, t, R1, R2, R3, R4, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
摘要翻译: 本发明包括新的式(I)化合物,其中n,m,t,R 1,R 2,R 3,R 3, 具有组氨酸脱乙酰酶抑制酶活性的含义; 其制剂,含有它们的组合物及其作为药物的用途。
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