公开(公告)号：US06737383B1

公开(公告)日：2004-05-18

申请号：US09869771

申请日：2001-06-29

申请人： Gary David Annis ,  George Chih-Shu Chiang ,  David Raymond Forney ,  Kanu Maganbhai Patel ,  Morris Padgett Rorer ,  William Francis Smith, III ,  Thomas Martin Stevenson ,  King-Mo Sun ,  Chi-Ping Tseng

发明人： Gary David Annis ,  George Chih-Shu Chiang ,  David Raymond Forney ,  Kanu Maganbhai Patel ,  Morris Padgett Rorer ,  William Francis Smith, III ,  Thomas Martin Stevenson ,  King-Mo Sun ,  Chi-Ping Tseng

IPC分类号： C07D27107

CPC分类号： A01N47/38 ,  C07D271/07 ,  C07D413/04 ,  C07D413/06 ,  C07D413/12 ,  C07D417/04 ,  C07D417/06

摘要： Compounds of Formula (1) and processes for their preparation, their N-oxides and agriculturally suitable salts, are disclosed which are useful for controlling undesired vegetation wherein Q, X1, X2, X3, R1, R2, R6 and R7 are as defined in the disclosure. Also disclosed are novel intermediates of Formula (5), Formula (8) and Formula (20) wherein R27 is —(CR6R7)q—Q; R6, R7, q, Q, X1 and X2 are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula (1) and a method for controlling undesired vegetation which involves contacting the vegetation or its environment with an effective amount of a compound of Formula (1).

摘要翻译： 公开了式（1）化合物及其制备方法，其N-氧化物和农业上合适的盐，其可用于控制不期望的植物，其中Q，X 1，X 2，X 3， R 1，R 2，R 6和R 7如本公开所定义。 还公开了式（5），式（8）和式（20）的新中间体，其中R 27是 - （CR 6 R 7）q -Q; R 6，R 7，q，Q，X 1和X 2如本公开所定义。 还公开了含有式（1）化合物和控制不期望植物的方法的组合物，其涉及将植物或其环境与有效量的式（1）化合物接触。

公开(公告)号：US6096895A

公开(公告)日：2000-08-01

申请号：US952384

申请日：1997-11-13

申请人： Richard James Brown ,  Dilon Jancey Daniel ,  Deborah Ann Frasier ,  Michael Henry Howard, Jr. ,  Gerard Michael Koether ,  Morris Padgett Rorer

发明人： Richard James Brown ,  Dilon Jancey Daniel ,  Deborah Ann Frasier ,  Michael Henry Howard, Jr. ,  Gerard Michael Koether ,  Morris Padgett Rorer

IPC分类号： A01N43/653 ,  A01N43/82 ,  A01N55/00 ,  C07D249/12 ,  C07D401/04 ,  C07D401/14 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D413/04 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F7/08 ,  A01N43/647

CPC分类号： C07D401/04 ,  A01N43/653 ,  A01N43/82 ,  A01N55/00 ,  C07D401/14 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F7/0812

摘要： Compounds of Formula I, and their N-oxides and agriculturally suitable salts, are disclosed which are useful as fungicides ##STR1## In said formula, E is a ring system selected from certain 5- to 12-membered monocyclic and fused bicyclic aromatic heterocyclic ring systems, or an optionally substituted naphthalene ring as defined in the disclosure;A is O; S; N; NR.sup.5 ; or CR.sup.14 ;G is C or N; provided that when G is C, then A is O, S or NR.sup.5 and the floating double bond is attached to G; and when G is N, then A is N or CR.sup.14 and the floating double bond is attached to A;W is O; S; NH; N(C.sub.1 -C.sub.6 alkyl); or NO(C.sub.1 -C.sub.6 alkyl);X is OR.sup.1 ; S(O).sub.m R.sup.1 ; or halogen;R.sup.1 is C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.6 haloalkyl; C.sub.2 -C.sub.6 alkenyl; C.sub.2 -C.sub.6 haloalkenyl; C.sub.2 -C.sub.6 alkynyl; C.sub.2 -C.sub.6 haloalkynyl; C.sub.3 -C.sub.6 cycloalkyl; C.sub.2 -C.sub.4 alkylcarbonyl; or C.sub.2 -C.sub.4 alkoxycarbonyl;R.sup.2 is H; C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.6 haloalkyl; C.sub.2 -C.sub.6 alkenyl; C.sub.2 -C.sub.6 haloalkenyl; C.sub.2 -C.sub.6 alkynyl; C.sub.2 -C.sub.6 haloalkynyl; C.sub.3 -C.sub.6 cycloalkyl; C.sub.2 -C.sub.4 alkylcarbonyl; C.sub.2 -C.sub.4 alkoxycarbonyl; hydroxy; C.sub.1 -C.sub.2 alkoxy; or acetyloxy;R.sup.5 is H; C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.6 haloalkyl; C.sub.2 -C.sub.6 alkenyl; C.sub.2 -C.sub.6 haloalkenyl; C.sub.2 -C.sub.6 alkynyl; C.sub.2 -C.sub.6 haloalkynyl; C.sub.3 -C.sub.6 cycloalkyl; C.sub.2 -C.sub.4 alkylcarbonyl; or C.sub.2 -C.sub.4 alkoxycarbonyl; andY, Z, R.sup.14 and m are as defined in the disclosure.Also disclosed are compositions containing the compounds of Formula I and a method for controlling plant diseases caused by fungal plant pathogens which involves applying an effective amount of a compound of Formula I.

摘要翻译： PCT No.PCT / US96 / 06533 Sec。 371日期：1997年11月13日 102（e）日期1997年11月13日PCT提交1996年5月8日PCT公布。 WO96 / 36633 PCT公开号 日期：1996年11月21日公开了式I化合物及其N-氧化物和农业上合适的盐，其可用作杀真菌剂。在所述式中，E是选自某些5-至12-元单环和稠合双环芳族 杂环体系或本公开中所定义的任选取代的萘环; A是O S; N; NR5; 或CR14; G为C或N; 条件是当G为C时，A为O，S或NR5，浮动双键连接至G; 当G为N时，A为N或CR14，浮选双键为A; W是O; S; NH; N（C 1 -C 6烷基）; 或NO（C 1 -C 6烷基）; X为OR1; S（O）mR1; 或卤素; R1是C1-C6烷基; C1-C6卤代烷基; C2-C6烯基; C2-C6卤代烯基; C2-C6炔基; C 2 -C 6卤代炔基; C3-C6环烷基; C 2 -C 4烷基羰基; 或C 2 -C 4烷氧基羰基; R2为H; C1-C6烷基; C1-C6卤代烷基; C2-C6烯基; C2-C6卤代烯基; C2-C6炔基; C 2 -C 6卤代炔基; C3-C6环烷基; C 2 -C 4烷基羰基; C 2 -C 4烷氧基羰基; 羟基; C1-C2烷氧基; 或乙酰氧基; R5是H; C1-C6烷基; C1-C6卤代烷基; C2-C6烯基; C2-C6卤代烯基; C2-C6炔基; C 2 -C 6卤代炔基; C3-C6环烷基; C 2 -C 4烷基羰基; 或C 2 -C 4烷氧基羰基; 和Y，Z，R 14和m如本公开中所定义。 还公开了含有式I化合物的组合物和控制由真菌植物病原体引起的植物病害的方法，其涉及施用有效量的式I化合物。