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    N-thiolated 2-oxazolidinone-derived antibiotics
    1.
    发明授权
    N-thiolated 2-oxazolidinone-derived antibiotics 有权
    N-硫醇化2-恶唑烷酮衍生的抗生素

    公开(公告)号：US07482467B2

    公开(公告)日：2009-01-27

    申请号：US11948073

    申请日：2007-11-30

    Applicant: Edward Turos ,  Rajesh Kumar Mishra

    Inventor： Edward Turos ,  Rajesh Kumar Mishra

    IPC: C07D263/02

    CPC classification number: C07D263/26 ,  C07D263/52

    Abstract: This invention describes the discovery and synthesis of N-thiolated 2-oxazolidinones as a new class of anti bacterial agents. These compounds can be synthesized from 2-oxazolidinones by Ndeprotection and N-sulfenylation. These new substances were found to exhibit potent anti-bacterial activity, including bacteriostatic properties against Staphylococcus spp., including methicillin resistant Staphylococcus aureus (MRSA), and Bacillus spp., including Bacillus anthracis.

    Abstract translation: 本发明描述了N-硫醇化的2-恶唑烷酮作为新类抗细菌剂的发现和合成。 这些化合物可以通过Nd保护和N-亚磺酰化由2-恶唑烷酮合成。 发现这些新物质显示出有效的抗细菌活性，包括对葡萄球菌属的抑菌性，包括耐甲氧西林金黄色葡萄球菌（MRSA）和芽孢杆菌属（Bacillus spp。），包括炭疽芽孢杆菌。

    N-thiolated 2 oxazolidone antibiotics
    2.
    发明授权
    N-thiolated 2 oxazolidone antibiotics 有权
    N-硫醇化2恶唑烷酮抗生素

    公开(公告)号：US07332611B2

    公开(公告)日：2008-02-19

    申请号：US11382157

    申请日：2006-05-08

    Applicant: Edward Turos ,  Rajesh Kumar Mishra

    Inventor： Edward Turos ,  Rajesh Kumar Mishra

    IPC: C07D263/02

    CPC classification number: C07D263/26 ,  C07D263/52

    Abstract: This invention describes the discovery and synthesis of N-thiolated 2-oxazolidinones as a new class of anti bacterial agents. These compounds can be synthesized from 2-oxazolidinones by Ndeprotection and N-sulfenylation. These new substances were found to exhibit potent anti-bacterial activity, including bacteriostatic properties against Staphylococcus spp., including methicillin resistant Staphylcoccus aureus (MRSA), and Bacillus spp., including Bacillus anthracis.

    Abstract translation: 本发明描述了N-硫醇化的2-恶唑烷酮作为新类抗细菌剂的发现和合成。 这些化合物可以通过Nd保护和N-亚磺酰化由2-恶唑烷酮合成。 发现这些新物质显示出有效的抗细菌活性，包括对葡萄球菌属的抑菌性，包括耐甲氧西林金黄色葡萄球菌（MRSA）和芽孢杆菌属（Bacillus spp。），包括炭疽芽孢杆菌。

    Derivative N-thiolated 2-oxazolidinone antibiotics
    3.
    发明授权
    Derivative N-thiolated 2-oxazolidinone antibiotics 失效
    衍生N-硫醇化2-恶唑烷酮抗生素

    公开(公告)号：US08703963B2

    公开(公告)日：2014-04-22

    申请号：US12028460

    申请日：2008-02-08

    Applicant: Edward Turos ,  Rajesh Kumar Mishra ,  Kevin Revell

    Inventor： Edward Turos ,  Rajesh Kumar Mishra ,  Kevin Revell ,  Cristina M. Coates

    IPC: C07D263/26

    CPC classification number: C07D263/26 ,  C07D263/52

    Abstract: This invention describes the discovery and synthesis of N-thiolated 2-oxazolidinones as a new class of anti bacterial agents. These compounds can be synthesized from 2-oxazolidinones by Ndeprotection and N-sulfenylation. These new substances were found to exhibit potent anti-bacterial activity, including bacteriostatic properties against Staphylococcus spp., including methicillin resistant Staphylcoccus aureus (MRSA), and Bacillus spp., including Bacillus anthracis.

    Abstract translation: 本发明描述了N-硫醇化的2-恶唑烷酮作为新类抗细菌剂的发现和合成。 这些化合物可以通过Nd保护和N-亚磺酰化由2-恶唑烷酮合成。 发现这些新物质显示出有效的抗细菌活性，包括对葡萄球菌属的抑菌性，包括耐甲氧西林金黄色葡萄球菌（MRSA）和芽孢杆菌属（Bacillus spp。），包括炭疽芽孢杆菌。

    IMPLEMENTING A SCALABLE TEST ENVIRONMENT
    4.
    发明申请
    IMPLEMENTING A SCALABLE TEST ENVIRONMENT 审中-公开
    实施可扩展的测试环境

    公开(公告)号：US20130238668A1

    公开(公告)日：2013-09-12

    申请号：US13414175

    申请日：2012-03-07

    Applicant: Kalambur Subramaniam ,  Rajesh Kumar Mishra ,  Mandar Nanivadekar ,  Prakash B. Angadi ,  Albrecht Schroth

    Inventor： Kalambur Subramaniam ,  Rajesh Kumar Mishra ,  Mandar Nanivadekar ,  Prakash B. Angadi ,  Albrecht Schroth

    IPC: G06F7/00

    CPC classification number: G06F11/3664 ,  G06F16/188

    Abstract: An embodiment provides a system and method for implementing a scalable test environment. The method includes modeling, within a file system environment creator executing on a computing device, a structure of a file system used by an application and intercepting a system call from the application to the file system at the file system environment creator. The method also includes generating a content of the file system dynamically within the file system environment creator based on the system call and the structure of the file system.

    Abstract translation: 实施例提供了用于实现可扩展测试环境的系统和方法。 该方法包括在计算设备上执行的文件系统环境创建器内建模应用程序使用的文件系统的结构，并在文件系统环境创建者处拦截系统调用从应用程序到文件系统。 该方法还包括基于系统调用和文件系统的结构在文件系统环境创建器内动态生成文件系统的内容。

    N-THIOLATED 2-OXAZOLIDINONE -DERIVED ANTIBIOTICS
    5.
    发明申请
    N-THIOLATED 2-OXAZOLIDINONE -DERIVED ANTIBIOTICS 有权
    N-巯基-2-氧杂环己烷 - 抗坏血酸

    公开(公告)号：US20080119533A1

    公开(公告)日：2008-05-22

    申请号：US11948073

    申请日：2007-11-30

    Applicant: Edward Turos ,  Rajesh Kumar Mishra

    Inventor： Edward Turos ,  Rajesh Kumar Mishra

    IPC: A61K31/421 ,  C07D263/20 ,  A61P31/04

    CPC classification number: C07D263/26 ,  C07D263/52

    Abstract: This invention describes the discovery and synthesis of N-thiolated 2-oxazolidinones as a new class of anti bacterial agents. These compounds can be synthesized from 2-oxazolidinones by Ndeprotection and N-sulfenylation. These new substances were found to exhibit potent anti-bacterial activity, including bacteriostatic properties against Staphylococcus spp., including methicillin resistant Staphylococcus aureus (MRSA), and Bacillus spp., including Bacillus anthracis.

    Abstract translation: 本发明描述了N-硫醇化的2-恶唑烷酮作为新类抗细菌剂的发现和合成。 这些化合物可以通过Nd保护和N-亚磺酰化由2-恶唑烷酮合成。 发现这些新物质显示出有效的抗细菌活性，包括对葡萄球菌属的抑菌性，包括耐甲氧西林金黄色葡萄球菌（MRSA）和芽孢杆菌属（Bacillus spp。），包括炭疽芽孢杆菌。

    DERIVATIVE N-THIOLATED 2-OXAZOLIDINONE ANTIBIOTICS
    6.
    发明申请
    DERIVATIVE N-THIOLATED 2-OXAZOLIDINONE ANTIBIOTICS 失效
    衍生的N-巯基2-氧杂环丁烷酮抗生素

    公开(公告)号：US20120149911A1

    公开(公告)日：2012-06-14

    申请号：US12028460

    申请日：2008-02-08

    Applicant: Edward Turos ,  Rajesh Kumar Mishra

    Inventor： Edward Turos ,  Rajesh Kumar Mishra

    IPC: C07D263/26

    CPC classification number: C07D263/26 ,  C07D263/52

    Abstract: This invention describes the discovery and synthesis of N-thiolated 2-oxazolidinones as a new class of anti bacterial agents. These compounds can be synthesized from 2-oxazolidinones by Ndeprotection and N-sulfenylation. These new substances were found to exhibit potent anti-bacterial activity, including bacteriostatic properties against Staphylococcus spp., including methicillin resistant Staphylcoccus aureus (MRSA), and Bacillus spp., including Bacillus anthracis.

    Abstract translation: 本发明描述了N-硫醇化的2-恶唑烷酮作为新类抗细菌剂的发现和合成。 这些化合物可以通过Nd保护和N-亚磺酰化由2-恶唑烷酮合成。 发现这些新物质显示出有效的抗细菌活性，包括对葡萄球菌属的抑菌性，包括耐甲氧西林金黄色葡萄球菌（MRSA）和芽孢杆菌属（Bacillus spp。），包括炭疽芽孢杆菌。

    DERIVATIVE N-THIOLATED 2-OXAZOLIDINONE ANTIBIOTICS
    7.
    发明申请
    DERIVATIVE N-THIOLATED 2-OXAZOLIDINONE ANTIBIOTICS 审中-公开
    衍生的N-巯基2-氧杂环丁烷酮抗生素

    公开(公告)号：US20090156654A1

    公开(公告)日：2009-06-18

    申请号：US12339174

    申请日：2008-12-19

    Applicant: Edward Turos ,  Rajesh Kumar Mishra

    Inventor： Edward Turos ,  Rajesh Kumar Mishra

    IPC: A61K31/421 ,  A61P31/04

    CPC classification number: C07D263/26 ,  C07D263/52

    Abstract: This invention describes the discovery and synthesis of N-thiolated 2-oxazolidinones as a new class of anti bacterial agents. These compounds can be synthesized from 2-oxazolidinones by Ndeprotection and N-sulfenylation. These new substances were found to exhibit potent anti-bacterial activity, including bacteriostatic properties against Staphylococcus spp., including methicillin resistant Staphylococcus aureus (MRSA), and Bacillus spp., including Bacillus anthracis.

    Abstract translation: 本发明描述了N-硫醇化的2-恶唑烷酮作为新类抗细菌剂的发现和合成。 这些化合物可以通过Nd保护和N-亚磺酰化由2-恶唑烷酮合成。 发现这些新物质显示出有效的抗细菌活性，包括对葡萄球菌属的抑菌性，包括耐甲氧西林金黄色葡萄球菌（MRSA）和芽孢杆菌属（Bacillus spp。），包括炭疽芽孢杆菌。

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