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公开(公告)号:US20050043533A1
公开(公告)日:2005-02-24
申请号:US10807884
申请日:2004-03-24
申请人: Kevin Babiak , Terri Boehm , Pierre-Jean Colson , Payman Farid , Donald Gallagher , Christian Huber , Russell Linderman , Chin Liu , Eduardo Mar , Murad Newaz , Daniel Pippel , Claire Przybyla , Christopher Robb , Glenn Stahl , Ravindra Topgi , Gerald Weisenburger , Edward Yonan
发明人: Kevin Babiak , Terri Boehm , Pierre-Jean Colson , Payman Farid , Donald Gallagher , Christian Huber , Russell Linderman , Chin Liu , Eduardo Mar , Murad Newaz , Daniel Pippel , Claire Przybyla , Christopher Robb , Glenn Stahl , Ravindra Topgi , Gerald Weisenburger , Edward Yonan
IPC分类号: A61K20060101 , C07D43/02
CPC分类号: C07D335/02 , C07D211/54 , C07D309/08 , C07D401/04 , C07D401/06 , C07D401/14 , C07D405/06 , C07D405/12 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/04 , C07D417/12 , C07D417/14
摘要: This invention is directed generally to a process for making α-substituted hydroxamic acids (including salts thereof) generally corresponding in structure to Formula (I): wherein n, Z, Z3, A, R, E, and Y are as defined in this patent. This invention also is directed to compounds that may, for example, be used as intermediates in such a process, as well as processes for making such compounds.
摘要翻译: 本发明一般涉及在通式(I)结构中对应制备α-取代的异羟肟酸(包括其盐)的方法:其中n,Z,Z 3,A,R,E和Y为 在该专利中定义。 本发明还涉及可以例如在这种方法中用作中间体的化合物以及制备这些化合物的方法。