3-Isoxazolylcarbamate derivatives
    2.
    发明授权
    3-Isoxazolylcarbamate derivatives 失效
    3-异恶唑基氨基甲酸酯衍生物

    公开(公告)号:US4116671A

    公开(公告)日:1978-09-26

    申请号:US836237

    申请日:1977-09-23

    CPC分类号: C07D261/14 C07D261/20

    摘要: Isoxazole derivatives represented by the formula: ##STR1## wherein R represents hydrogen, alkyl group, or aryl group, R.sup.1 represents hydrogen, or alkyl group, R.sup.2 represents acyl group, a ##STR2## group [R.sup.3 and R.sup.4 each represent hydrogen, alkyl group, alkenyl group, alkynyl group, aralkyl group, aryl group, alkoxy group, or alkylthio group; or optionally R.sup.3 and R.sup.4 are combined with each other directly or indirectly including another hetero atom (nitrogen, oxygen, or sulfur) to form a nitrogen-containing ring], or a--CO--Y--R.sup.5group [R.sup.5 represents alkyl group, alkenyl group, alkynyl group, aralkyl group, or aryl group, and Y represents oxygen, or sulfur], and X represents hydrogen, alkyl group, or halogen, or R and X are optionally combined each other to form an alkylene group, said alkyl group, aralkyl group, and aryl group each being optionally substituted with one or more members selected from halogen, alkyl group, alkoxy group, nitro group, and hydroxy group, are prepared by eleven routes. The isoxazole derivatives are useful as herbicides.

    Herbicidal compositions containing 3-isoxazolylurea derivatives
    3.
    发明授权
    Herbicidal compositions containing 3-isoxazolylurea derivatives 失效
    含有3-异丙唑基衍生物的除草剂组合物

    公开(公告)号:US4111680A

    公开(公告)日:1978-09-05

    申请号:US836238

    申请日:1977-09-23

    CPC分类号: C07D261/14 C07D261/20

    摘要: Isoxazole derivatives represented by the formula: ##STR1## wherein R represents hydrogen, alkyl group, or aryl group, R.sup.1 represents hydrogen, or alkyl group, R.sup.2 represents acyl group, a ##STR2## group [R.sup.3 and R.sup.4 each represent hydrogen, alkyl group, alkenyl group, alkynyl group, aralkyl group, aryl group, alkoxy group, or alkylthio group; or optionally R.sup.3 and R.sup.4 are combined with each other directly or indirectly including another hetero atom (nitrogen, oxygen, or sulfur) to form a nitrogen-containing ring], or a --CO--Y--R.sup.5 group[R.sup.5 represents alkyl group, alkenyl group, alkynyl group, aralkyl group, or aryl group, and Y represents oxygen, or sulfur], and X represents hydrogen, alkyl group, or halogen, or R and X are optionally combined each other to form an alkylene group, said alkyl group, aralkyl group, and aryl group each being optionally substituted with one or more members selected from halogen, alkyl group, alkoxy group, nitro group, and hydroxy group, are prepared by 11 routes. The isoxazole derivatives are useful as herbicides.

    摘要翻译: 由下式表示的异恶唑衍生物:其中R表示氢,烷基或芳基,R 1表示氢或烷基,R 2表示酰基,基团[R 3和R 4各自表示氢,烷基 烯基,炔基,芳烷基,芳基,烷氧基或烷硫基; 或任选的R 3和R 4彼此直接或间接地包含另外的杂原子(氮,氧或硫)以形成含氮环]或-CO-Y-R 5基[R 5表示烷基,烯基 基团,炔基,芳烷基或芳基,Y表示氧或硫],X表示氢,烷基或卤素,或R和X任选地相互结合形成亚烷基,所述烷基 芳烷基,芳基,芳基,可以被选自卤素,烷基,烷氧基,硝基,羟基中的一个以上的任意一个取代。 异恶唑衍生物可用作除草剂。

    3-Alkylisoxazole derivatives and herbicides containing them
    4.
    发明授权
    3-Alkylisoxazole derivatives and herbicides containing them 失效
    含有它们的3-烷基异恶唑衍生物和除草剂

    公开(公告)号:US4028376A

    公开(公告)日:1977-06-07

    申请号:US615883

    申请日:1975-09-23

    CPC分类号: C07D261/14 C07D261/20

    摘要: 3-ALKYLISOXAZOLE DERIVATIVES REPRESENTED BY THE FORMULA: ##STR1## wherein R represents C.sub.3 -C.sub.6 alkyl or C.sub.3 -C.sub.6 cycloalkyl, R.sup.1 represents hydrogen or C.sub.1 -C.sub.6 alkyl, R.sup.2 represents ##STR2## [in which R.sup.3 and R.sup.4 each represent hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.7 alkenyl, C.sub.1 -C.sub.6 alkoxy, C.sub.2 -C.sub.7 alkoxycarbonyl or C.sub.1 -C.sub.6 alkylthio, or ##STR3## represents morpholino, pyrrolidino or piperidino, and Y represents oxygen or sulfur] or --CO--Y--R.sup.5 [in which R.sup.5 represents C.sub.1 -C.sub.6 alkyl and Y is as defined above] and X represents hydrogen, halogen or C.sub.1 -C.sub.6 alkyl, or R and X are combined to form C.sub.3 -C.sub.6 alkylene, being useful as herbicides, are prepared by several routes.

    摘要翻译: 其中R表示C 3 -C 6烷基或C 3 -C 6环烷基,R 1表示氢或C 1 -C 6烷基,R 2表示其中R 3和R 4各自表示氢,C 1 -C 6烷基,C 1 -C 6烷氧基, C2-C7链烯基,C1-C6烷氧基,C2-C7烷氧基羰基或C1-C6烷硫基,或表示吗啉代,吡咯烷子基或哌啶子基,Y表示氧或硫]或-CO-Y-R5 [其中R5表示C1-C6烷基和 Y如上所定义),X表示氢,卤素或C 1 -C 6烷基,或R和X组合形成可用作除草剂的C 3 -C 6亚烷基,是通过若干途径制备的。

    3-Isoxazolylurea derivatives
    7.
    发明授权
    3-Isoxazolylurea derivatives 失效
    3-异恶唑基脲衍生物

    公开(公告)号:US4062861A

    公开(公告)日:1977-12-13

    申请号:US667033

    申请日:1976-03-15

    IPC分类号: C07D261/14 C07D261/20

    CPC分类号: C07D261/14 C07D261/20

    摘要: Isoxazole derivatives represented by the formula: ##STR1## wherein R represents hydrogen, alkyl group, or aryl group, R.sup.1 represents hydrogen, or alkyl group, R.sup.2 represents acyl group, a ##STR2## group [R.sup.3 and R.sup.4 each represent hydrogen, alkyl group, alkenyl group, alkynyl group, aralkyl group, aryl group, alkoxy group, or alkylthio group; or optionally R.sup.3 and R.sup.4 are combined with each other directly or indirectly including another hetero atom (nitrogen, oxygen, or sulfur) to form a nitrogen-containing ring], or a --CO--Y--R.sup.5 group [R.sup.5 represents alkyl group, alkenyl group, alkynyl group, aralkyl group, or aryl group, and Y represents oxygen, or sulfur], and X represents hydrogen, alkyl group, or halogen, or R and X are optionally combined each other to form an alkylene group, said alkyl group, aralkyl group, and aryl group each being optionally substituted with one or more members selected from halogen, alkyl group, alkoxy group, nitro group, and hydroxy group, are prepared by eleven routes. The isoxazole derivatives are useful as herbicides.

    摘要翻译: 由下式表示的异恶唑衍生物:其中R表示氢,烷基或芳基,R 1表示氢或烷基,R 2表示酰基,基团[R 3和R 4各自表示氢,烷基 烯基,炔基,芳烷基,芳基,烷氧基或烷硫基; 或任选的R 3和R 4彼此直接或间接地包含另外的杂原子(氮,氧或硫)以形成含氮环]或-CO-Y-R 5基[R 5表示烷基,烯基 基团,炔基,芳烷基或芳基,Y表示氧或硫],X表示氢,烷基或卤素,或R和X任选地相互结合形成亚烷基,所述烷基 芳烷基,芳基,芳基,可以被选自卤素,烷基,烷氧基,硝基,羟基中的一个以上的任意一个取代。 异恶唑衍生物可用作除草剂。

    Isoxazole derivatives
    8.
    发明授权
    Isoxazole derivatives 失效
    异恶唑衍生物

    公开(公告)号:US4014876A

    公开(公告)日:1977-03-29

    申请号:US325115

    申请日:1973-01-19

    CPC分类号: C07D261/18 Y10S514/866

    摘要: Isoxazole derivatives represented by the formula: ##STR1## are prepared; wherein R.sup.1 and R.sup.2 each is hydrogen atom, alkyl group of 1 to 8 carbon atoms, or cycloalkyl group of 3 to 10 carbon atoms; R.sup.3 and R.sup.4 each is hydrogen atom, alkyl group of 1 to 8 carbon atoms, cycloalkyl group of 3 to 10 carbon atoms, or phenyl group; or the groupIs morpholino group; and Y is oxo group, thioxo group or imino group; being useful as a hypoglycemic and/or a blood free-fatty-acid normalizing antidiabetic agent.

    摘要翻译: 制备由下式表示的异恶唑衍生物: ; 其中R 1和R 2各自为氢原子,1至8个碳原子的烷基或3至10个碳原子的环烷基; R3和R4各自为氢原子,1〜8个碳原子的烷基,3〜10个碳原子的环烷基或苯基; 或集团IS MORPHOLINO GROUP; 并且Y是氧代基,硫代基或亚氨基; 可用作降血糖和/或血液游离脂肪酸标准化抗糖尿病药。